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121 Cards in this Set
- Front
- Back
Bethanechol (Urecholine)
|
muscarinic
|
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Pilocarpine (Salagen)
|
muscarinic
|
|
Carbachol
|
muscarinic
|
|
Cevimiline (Evoxac)
|
muscarinic
|
|
Atropine
|
anti-muscarinic
|
|
Tropicamide (Mydriacyl)
|
anti-muscarinic
|
|
Cyclopentolate (Cyclogyl)
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anti-muscarinic
|
|
Glycopyrrolate
|
anti-muscarinic
|
|
Mepenzolate
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anti-muscarinic
|
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Propantheline
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anti-muscarinic
|
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Clidinium
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anti-muscarinic
|
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Dicyclomine (Bentyl)
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anti-muscarinic
|
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Hyoscyamine (Levsin)
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anti-muscarinic
|
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Scopolamine (Transderm Scop)
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anti-muscarinic
|
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Belladonna
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anti-muscarinic
|
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Ipratropium (Flovent)
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anti-muscarinic
|
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Tiotropium (Spiriva)
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anti-muscarinic
|
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Tolterodine (Detrol/Detrol LA)
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anti-muscarinic
|
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Fesoterodine (Toviaz)
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anti-muscarinic
|
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Oxybutynin (Ditropan/Ditropan XL)
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anti-muscarinic
|
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Darifenacin (Enablex)
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anti-muscarinic
|
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Solfenacin (Vesicare)
|
anti-muscarinic
|
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Trospium (Sanctura)
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anti-muscarinic
|
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Flavoxate (Urispas)
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anti-muscarinic
|
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Neostigmine
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AChE inhibitor
|
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Physostigmine
|
AChE inhibitor
|
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Pyridostigmine (Mestinon)
|
AChE inhibitor
|
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Ambenonium (Mytelase)
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AChE inhibitor
|
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Malathion (Ovide)
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AChE inhibitor
|
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Edrophonium
|
AChE inhibitor
|
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Echothiophate (Phospholine Iodide)
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AChE inhibitor
|
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Pralidoxime (2-PAM)
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Oxime. (Reverses neurotoxic effects of organophosphate inactivated acetylcholinesterase.)
|
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Varenicline (Chantix)
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Partial CNS Nicotinic Agonist
|
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Mecamylamine
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Ganglionic Blocker (used for severe hypertension--blocks SANS innervation of vessels)
|
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Pancuronium
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Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Vecuronium
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Muscle nicotinic receptor antagonist (competitive/polarizing)
|
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Atracurium
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Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Doxacurium
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Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Cisatracurium
|
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Rocuronium
|
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Mivacurium
|
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Rapacuronium
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Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
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Pipecuronium
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Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
|
|
Succinylcholine
|
Muscle nicotinic receptor agonist (depolarizing neuromuscular blocker) (NOTE: risk of malignant hyperthermia)
|
|
Oxymetazoline (Afrin)
|
Alpha-1 Agonist
|
|
Phenylephrine (Neo-Synephrine)
|
Alpha-1 Agonist
|
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Midodrine (ProAmatine)
|
Alpha-1 Agonist
|
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Pseudoephedrine (Sudafed)
|
Alpha-1 Agonist
|
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Prazosin (Minipress)
|
Alpha-1 ANTagonist
|
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Terazosin (Hytrin)
|
Alpha-1 ANTagonist
|
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Doxazosin (Cardura)
|
Alpha-1 ANTagonist
|
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Alfuzosin (Uroxatral)
|
Alpha-1 ANTagonist
|
|
Tamsulosin (Flomax)
|
Alpha-1 ANTagonist
(subtype 1a specific) (less 1st dose effect) |
|
Phenoxybenzamine (Dibenzyline)
|
Alpha blocker
(non-specific, irreversible) |
|
Phentolamine (Regitine)
|
Alpha blocker
(non-selective, reversible) |
|
Dobutamine
|
Beta-1 Agonist
(selective) (inotropic effect > chronotropic effect) @ higher doses = weak Beta-2 activity |
|
Clonidine (Catapres)
|
Alpha-2 agonist
|
|
Methyldopa
|
Alpha-2 agonist
(pro-drug) |
|
Guanabenz
|
Alpha-2 agonist
|
|
Guanfacine (Tenex)
|
Alpha-2 agonist
|
|
Dexmedetomidine
|
Alpha-2 agonist
|
|
Brimonidine (Alphagan)
|
Alpha-2 agonist
|
|
Apraclonidine
|
Alpha-2 agonist
|
|
Yohimbine
|
Alpha-2 ANTagonist
|
|
Isoproterenol
|
Beta agonist
(non-selective) |
|
Acebutolol (Sectral)
|
Beta-1 ANTagonist
(selective) (ISA = intrinsic sympathomimetic activity, that is, it has partial agonist activity) (best choice for COPD/asthma pt who needs a Beta blocker) |
|
Atenolol (Tenormin)
|
Beta-1 ANTagonist
|
|
Betaxolol (Betoptic)
|
Beta-1 ANTagonist
|
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Bisoprolol (Zebeta)
|
Beta-1 ANTagonist
|
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Esmolol (Brevibloc)
|
Beta-1 ANTagonist
|
|
Metoprolol (Lopressor/Toprol XL)
|
Beta-1 ANTagonist
|
|
Propranolol (Inderal/Inderal LA)
|
Beta ANTagonist
(non-selective) |
|
Nadolol (Corgard)
|
Beta ANTagonist
(non-selective) |
|
Pindolol
|
Beta ANTagonist
(non-selective) |
|
Sotalol (Betapace/Sotacor)
|
Beta ANTagonist
(non-selective) |
|
Timolol (Timoptic)
|
Beta ANTagonist
(non-selective) |
|
Levobunolol (Betegan)
|
Beta ANTagonist
(non-selective) |
|
Carvedilol (Coreg/Coreg CR)
|
Beta ANTagonist (non-selective)
Alpha-1 (selective) ANTagonist |
|
Labetalol (Trandate)
|
Beta ANTagonist (non-selective)
Alpha-1 (selective) ANTagonist |
|
Albuterol (Salbutamol)
|
Beta-2 agonist
(tocolytic drug) |
|
Bitolterol (Tornalate)
|
Beta-2 agonist
|
|
Formoterol (Foradil)
|
Beta-2 agonist
|
|
Isoetharine
|
Beta-2 agonist
|
|
Levalbuterol (Xopenex)
|
Beta-2 agonist
|
|
Metaproterenol (Alupent)
|
Beta-2 agonist
|
|
Pibuterol (Maxair)
|
Beta-2 agonist
|
|
Salmeterol (Serevent)
|
Beta-2 agonist
|
|
Terbutaline
|
Beta-2 agonist
(fast acting for status asthmaticus) (IV) (tocolytic drug) |
|
Ritodrine
|
Beta-2 agonist
(tocolytic drug) |
|
Fenoldopam
|
D1 weak agonist
Causes vasodilation of the renal/coronary arteries/arterioles Tx: severe HTN |
|
Indapamide (Lozol)
|
Thiazide-like diuretic
Possible hypokalemia |
|
Triamterene
|
K+ sparing diuretic
|
|
Hydrochlorothiazide
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Thiazide diuretic
Possible hypokalemia |
|
Dyazide (HCTZ + Triamterene)
|
Thiazide/K+ sparing diuretic combo
|
|
Metolazone (Zaroxolyn)
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Thiazide-like diuretic
|
|
Chlorthalidone (Hygroton)
|
Thiazide-like diuretic
|
|
Chlorothiazide
|
Thiazide diuretic
|
|
Verapamil (Calan)
|
Calcium Channel Blocker (CCB)
Non-DHP Phenylalkylamine |
|
Diltiazem (Cardizem)
|
Calcium Channel Blocker (CCB)
Non-DHP Benzothiazepine |
|
Amlodipine (Norvasc)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Felodipine (Plendil)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Isradipine (Dynacirc)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Nicardipine (Cardene)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Nifedipine (Adalat CC, Procardia XL)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Nimodipine (Nimotop)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Nisoldipine (Sular)
|
Calcium Channel Blocker (CCB)
DHP Affects blood vessels only! |
|
Methazolamide (Neptazane)
|
Carbonic anhydrase inhibitor
(sends Na+ and HCO3- downstream from the proximal convoluted tubule) |
|
Acetazolamide (Diamox)
|
Carbonic anhydrase inhibitor
(sends Na+ and HCO3- downstream from the proximal convoluted tubule) |
|
Dorzolamide (Trusopt)
|
Carbonic anhydrase inhibitor
(sends Na+ and HCO3- downstream from the proximal convoluted tubule) |
|
Amiloride
|
Na channel inhibitor
"K+ sparing" |
|
Triamterene
|
Na channel inhibitor
"K+ sparing" |
|
Eplerenone (Inspra)
|
Aldosterone antagonist
Very low efficacy due to location in late distal tubule and collecting duct |
|
Spironolactone
|
Aldosterone antagonist
Very low efficacy due to location in late distal tubule and collecting duct |
|
Vasopressin (ADH)
|
Agonist at V2 receptor.
SOA: In collecting duct. Increases insertion of water channels (aquaporins) into lumenal membrane. |
|
Desmopressin
|
DDAVP - V2 selective agonist
SOA: In collecting duct. Increases insertion of water channels (aquaporins) into lumenal membrane. |
|
Ethacrynic Acid
|
Loop diuretic
|
|
Furosemide
|
Loop diuretic
|
|
Bumetanide (Bumex)
|
Loop diuretic
|
|
Torsemide
|
Loop diuretic
|
|
Conivaptan
|
V1, V2 receptor antagonist
Promotes water loss!! Tx: euvolemic hyponatremia |
|
Tolvaptan
|
V1, V2 receptor antagonist
Promotes water loss!! Tx: euvolemic hyponatremia |