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121 Cards in this Set

  • Front
  • Back
Bethanechol (Urecholine)
muscarinic
Pilocarpine (Salagen)
muscarinic
Carbachol
muscarinic
Cevimiline (Evoxac)
muscarinic
Atropine
anti-muscarinic
Tropicamide (Mydriacyl)
anti-muscarinic
Cyclopentolate (Cyclogyl)
anti-muscarinic
Glycopyrrolate
anti-muscarinic
Mepenzolate
anti-muscarinic
Propantheline
anti-muscarinic
Clidinium
anti-muscarinic
Dicyclomine (Bentyl)
anti-muscarinic
Hyoscyamine (Levsin)
anti-muscarinic
Scopolamine (Transderm Scop)
anti-muscarinic
Belladonna
anti-muscarinic
Ipratropium (Flovent)
anti-muscarinic
Tiotropium (Spiriva)
anti-muscarinic
Tolterodine (Detrol/Detrol LA)
anti-muscarinic
Fesoterodine (Toviaz)
anti-muscarinic
Oxybutynin (Ditropan/Ditropan XL)
anti-muscarinic
Darifenacin (Enablex)
anti-muscarinic
Solfenacin (Vesicare)
anti-muscarinic
Trospium (Sanctura)
anti-muscarinic
Flavoxate (Urispas)
anti-muscarinic
Neostigmine
AChE inhibitor
Physostigmine
AChE inhibitor
Pyridostigmine (Mestinon)
AChE inhibitor
Ambenonium (Mytelase)
AChE inhibitor
Malathion (Ovide)
AChE inhibitor
Edrophonium
AChE inhibitor
Echothiophate (Phospholine Iodide)
AChE inhibitor
Pralidoxime (2-PAM)
Oxime. (Reverses neurotoxic effects of organophosphate inactivated acetylcholinesterase.)
Varenicline (Chantix)
Partial CNS Nicotinic Agonist
Mecamylamine
Ganglionic Blocker (used for severe hypertension--blocks SANS innervation of vessels)
Pancuronium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Vecuronium
Muscle nicotinic receptor antagonist (competitive/polarizing)
Atracurium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Doxacurium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Cisatracurium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Rocuronium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Mivacurium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Rapacuronium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Pipecuronium
Muscle nicotinic receptor antagonist (competitive/non-depolarizing)
Succinylcholine
Muscle nicotinic receptor agonist (depolarizing neuromuscular blocker) (NOTE: risk of malignant hyperthermia)
Oxymetazoline (Afrin)
Alpha-1 Agonist
Phenylephrine (Neo-Synephrine)
Alpha-1 Agonist
Midodrine (ProAmatine)
Alpha-1 Agonist
Pseudoephedrine (Sudafed)
Alpha-1 Agonist
Prazosin (Minipress)
Alpha-1 ANTagonist
Terazosin (Hytrin)
Alpha-1 ANTagonist
Doxazosin (Cardura)
Alpha-1 ANTagonist
Alfuzosin (Uroxatral)
Alpha-1 ANTagonist
Tamsulosin (Flomax)
Alpha-1 ANTagonist
(subtype 1a specific)
(less 1st dose effect)
Phenoxybenzamine (Dibenzyline)
Alpha blocker
(non-specific, irreversible)
Phentolamine (Regitine)
Alpha blocker
(non-selective, reversible)
Dobutamine
Beta-1 Agonist
(selective)
(inotropic effect > chronotropic effect)
@ higher doses = weak Beta-2 activity
Clonidine (Catapres)
Alpha-2 agonist
Methyldopa
Alpha-2 agonist
(pro-drug)
Guanabenz
Alpha-2 agonist
Guanfacine (Tenex)
Alpha-2 agonist
Dexmedetomidine
Alpha-2 agonist
Brimonidine (Alphagan)
Alpha-2 agonist
Apraclonidine
Alpha-2 agonist
Yohimbine
Alpha-2 ANTagonist
Isoproterenol
Beta agonist
(non-selective)
Acebutolol (Sectral)
Beta-1 ANTagonist
(selective)
(ISA = intrinsic sympathomimetic activity, that is, it has partial agonist activity)
(best choice for COPD/asthma pt who needs a Beta blocker)
Atenolol (Tenormin)
Beta-1 ANTagonist
Betaxolol (Betoptic)
Beta-1 ANTagonist
Bisoprolol (Zebeta)
Beta-1 ANTagonist
Esmolol (Brevibloc)
Beta-1 ANTagonist
Metoprolol (Lopressor/Toprol XL)
Beta-1 ANTagonist
Propranolol (Inderal/Inderal LA)
Beta ANTagonist
(non-selective)
Nadolol (Corgard)
Beta ANTagonist
(non-selective)
Pindolol
Beta ANTagonist
(non-selective)
Sotalol (Betapace/Sotacor)
Beta ANTagonist
(non-selective)
Timolol (Timoptic)
Beta ANTagonist
(non-selective)
Levobunolol (Betegan)
Beta ANTagonist
(non-selective)
Carvedilol (Coreg/Coreg CR)
Beta ANTagonist (non-selective)
Alpha-1 (selective) ANTagonist
Labetalol (Trandate)
Beta ANTagonist (non-selective)
Alpha-1 (selective) ANTagonist
Albuterol (Salbutamol)
Beta-2 agonist
(tocolytic drug)
Bitolterol (Tornalate)
Beta-2 agonist
Formoterol (Foradil)
Beta-2 agonist
Isoetharine
Beta-2 agonist
Levalbuterol (Xopenex)
Beta-2 agonist
Metaproterenol (Alupent)
Beta-2 agonist
Pibuterol (Maxair)
Beta-2 agonist
Salmeterol (Serevent)
Beta-2 agonist
Terbutaline
Beta-2 agonist
(fast acting for status asthmaticus)
(IV)
(tocolytic drug)
Ritodrine
Beta-2 agonist
(tocolytic drug)
Fenoldopam
D1 weak agonist
Causes vasodilation of the renal/coronary arteries/arterioles
Tx: severe HTN
Indapamide (Lozol)
Thiazide-like diuretic

Possible hypokalemia
Triamterene
K+ sparing diuretic
Hydrochlorothiazide
Thiazide diuretic

Possible hypokalemia
Dyazide (HCTZ + Triamterene)
Thiazide/K+ sparing diuretic combo
Metolazone (Zaroxolyn)
Thiazide-like diuretic
Chlorthalidone (Hygroton)
Thiazide-like diuretic
Chlorothiazide
Thiazide diuretic
Verapamil (Calan)
Calcium Channel Blocker (CCB)
Non-DHP
Phenylalkylamine
Diltiazem (Cardizem)
Calcium Channel Blocker (CCB)
Non-DHP
Benzothiazepine
Amlodipine (Norvasc)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Felodipine (Plendil)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Isradipine (Dynacirc)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Nicardipine (Cardene)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Nifedipine (Adalat CC, Procardia XL)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Nimodipine (Nimotop)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Nisoldipine (Sular)
Calcium Channel Blocker (CCB)
DHP

Affects blood vessels only!
Methazolamide (Neptazane)
Carbonic anhydrase inhibitor

(sends Na+ and HCO3- downstream from the proximal convoluted tubule)
Acetazolamide (Diamox)
Carbonic anhydrase inhibitor

(sends Na+ and HCO3- downstream from the proximal convoluted tubule)
Dorzolamide (Trusopt)
Carbonic anhydrase inhibitor

(sends Na+ and HCO3- downstream from the proximal convoluted tubule)
Amiloride
Na channel inhibitor

"K+ sparing"
Triamterene
Na channel inhibitor

"K+ sparing"
Eplerenone (Inspra)
Aldosterone antagonist

Very low efficacy due to location in late distal tubule and collecting duct
Spironolactone
Aldosterone antagonist

Very low efficacy due to location in late distal tubule and collecting duct
Vasopressin (ADH)
Agonist at V2 receptor.

SOA: In collecting duct. Increases insertion of water channels (aquaporins) into lumenal membrane.
Desmopressin
DDAVP - V2 selective agonist

SOA: In collecting duct. Increases insertion of water channels (aquaporins) into lumenal membrane.
Ethacrynic Acid
Loop diuretic
Furosemide
Loop diuretic
Bumetanide (Bumex)
Loop diuretic
Torsemide
Loop diuretic
Conivaptan
V1, V2 receptor antagonist

Promotes water loss!!
Tx: euvolemic hyponatremia
Tolvaptan
V1, V2 receptor antagonist

Promotes water loss!!
Tx: euvolemic hyponatremia