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18 Cards in this Set
- Front
- Back
Short Acting Beta 2 Agonists;
Meds; MOA; ADR; CI; Dose; Monitoring; |
*Drug of choice for mld/mod asthma, COPD*
Albuterol, Maxair (pirbuterol), Xopenex, Alupent (metaproterenol) MOA; relaxes bronchial smooth muscle by action on beta 2 receptors. ADR; angina, HTN, palpitation, nausea, diarrhea, dizziness, irritability, CNS stimulation, asthma exacerbation, hyperglycemia, hypokalemia, allergy. *ADR more pronounced w/po med, use spacer* Precautions; CV dz, glaucoma, hyperthyroidism, DM, preg cat C (po terbutaline used to prevent labor) CI; Hypersensitivity Dose; Acute 4-8 puffs or neb 2.5mg q 20mins. Chronic; 1-2 puffs q 4-6hrs/max 12 puffs qd. PO; 2-4mg 3-4X day/max 32mg qd. Prophylaxis; 2 puffs 30mins prior to exercise. Monitoring; PFT's, BP, HR, Gulcose, K. |
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Long Acting Beta 2 Agonists;
Meds; ADR; CI; Dose; Monitoring; Warnings; |
Serevent (salmeterol, Foradil (formoterol), Brovana (arformoterol.
*Not for acute attacks, maintence med only* ADR; HA, HTN, tachycardia, CNS stimulation, dizziness, insomnia, asthma, bronchoconstriction, allergy. CI; hypersensitivity, acute tx. Monitoring; PFT's, BP, HR, CNS stim, glucose, k, asthma sx. Warning; long acting may ↑ asthma related deaths, CV, DM, glaucoma, hyperthyroidism, hypokalemia, seizures, animal studies show dose dep. |
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Cortidosteroids;
Meds & strength; MOA; ADR; Warning; CI; Dose; Conversion Oral to inhaled; |
Inhaled or systemic *1st choice for moderate/severe asthma or COPD
Aerobid (flunisolide)250mcg/puff, Asmacort (triamcinolone) 100mcg/puff, Asmanex (mometasone) 220mcg/puff, Beconase, QVar (beclomethasone) 40,80mcg/puff, Flovent HFA (fluticasone) 110mcg/puff, Pulmicort (budesonide) 90, 180 mcg/puff, Combo; Advair (fluticasone/salmeterol 100/50, 250/50, 500/50mcg/dose, Symbicort (budesonide/formoterol), Prednisone, methylprednisone, given during acute attacks IV or PO MOA; decrease immune response to allergens, irritants, cold & exercise (macrophages, T lymph, eosinophils) ADR;(minimized w/spacer)HA, resp tract infection, throat irritation, sinus infection, cough, thrush, dizziness, insomnia, mood swings, bronchospasm, ↓ growth w/peds. Warning; HPA suppression in children, viral infections, preg cat C. CI; hypersensitivity, acute broncho-spasm. Dose; use lowest strength to start, 1-2inh bid Conversion; oral to inhaled, must taper off oral 10days p starting inhaled. |
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Mast Cell Stablizers;
Meds; MOA; Use; ADR; Precautions; CI; Dose; |
Intal (cromolyn), Tilade (nedocromil)
MOA; prevent mast cell release of histamine & leukotrienes. Use; preventitive, must be used @ regular intervals for 2-4wks, prophylaxis;10-15mins prior. ADR; bad taste, HA, dizziness, drowsiness, n/v, cough. Precautions; not for <6yrs, Preg cat B. CI; hypersensitivity, acute bronchospasm. Dose; 2puffs 3-4 X qd |
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Cholinergic Antagonist
Meds; MOA; Use; ADR; Precaution; CI; Dose; |
Meds; Atrovent (ipratropium)
MOA; blocks vagally mediated contraction of smooth muscle. Use; bronchospasm, COPD ADR; bronchitis, palpitation, dizziness, nausea, sinusitis, glaucoma, urinary retention, dry eyes, dry mouth. Precaution; not for acute attack, glaucoma, BPH/bladder obstruction. CI; hypersensitivity to ipratropium or atropine. Dose; 2puffs qid |
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Methylxanthines, Theophylline;
Meds; MOA; Use; ADR; Precaution; CI; Dose; |
Theo24, Uniphyl, Elixophyllin
MOA; ↑ epinephrine release & then bronchodilation. Use; Asthma, bronchitis, COPD ADR;dose dependent, Serum 15-25mcg/ml: n/v, diarrhea, insomnia, nervousness, dizziness, HA, muscle cramps. Serum 25-35mcg/ml:tachycardia Serum <35mcg/ml: Vtach, PVC, seizure. *Narrow therapeutic index, drug interactions, replaced by albuterol & corticosteroids* Precautions; vomiting, draw level & hold dose, hyperthroidism, seizures, hypertension & arrhythmias, smoking, avoid dietary stimulants, preg cat C CI; hypersensitivity Dose; wt based not to exceed 900mg qd (tablets, liquid, IV) |
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Anti-leukotrienes Drugs;
What are Leukotrienes? Meds; MOA; Use; ADR; Precaution; CI; Dose; |
Leukotrienes cause eoxinophil migration, neutrophil/monocyte aggregation, ↑ cap permeability, S/M contraction, edema, muccous secretion & bronchoconstriction.
Meds; Singulair qd(montelukast), Accolate bid(zafirlukast) MOA; blocks leukotriene receptors responsible for secretions & edema in asthma. Use; prophylaxis & chronic tx of asthma. ADR; HA, dizziness, n/v/d, pain, weakness, hepatitis, infection. Precaution; acute bronchospasm, liver dysfunction, preg cat B CI; hypersensitivity Dose; Singulair 10mg po qd >6mos, Accolate 20mg po bid >5yrs |
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Leukotriene Inhibitors;
Meds; MOA; Use; ADR; Precaution; CI; Dose; |
Med; Zyflo (zileuton)
MOA; inhibits leukoriene formation. Use; asthma ADR; HA, pain, nausea, ↑ liver enzymes. Precaution; liver dysfunction, peds <12, preg cat C, interacts w/theophylline & warfarin CI; hypersensitivity, active liver dz Dose; 600 mg qid |
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Monoclonal Antibody;
Meds; MOA; Use; ADR; Precaution; CI; Dose; |
Meds; Xolair (omalizumab)
MOA; IgG monoclonal antibody, decreases IgE mediated response to allergies. Use;Mod/Severe allergic asthma not respondent to corticosteroids. ADR;HA, injection pain, URT infxn, viral infxn, sinusitis, dermatitis, anaphylaxis. Precaution; monitor IgE levels, delayed allergic reaction CI; hypersensitivity, acute bronchospasm, status asthmaticus. Dose; based on wt & IgE levels, 150-400 units sugQ q 2-4wks, stays in body for 1yr. |
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Myambutol (ethambutol);
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB
MOA;inhibits RNA synthesis ADR;optic neuritis, hepatotoxicity, myocarditis, n/v, gout, blood dyscrasias, renal failure. Precaution; liver, kidney dysfunction (↓ dose), preg C. CI; hypersensitivity Dose; daily, twice or three X a wk based on wt. Monitoring; baseline & monthly visual tests, renal hepatic & blood test. |
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Isoniazid (INH)
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use;TB
MOA; Disruption of cell wall synthesis ADR; liver failure, vision loss, HTN, palp, tachy, dizziness, rash, hyperglycemia, n/v, blood dyscrasias, hepatitis, peripheral neuropathy. Precaution; boxed warning fatal hepatitis, liver dysfunction, eye problems, preg C CI; hypersensitivity, acute liver dz. Dose; 300mg qd for 6-9mos Monitoring; 650mg/qd pridoxine to ↓ risk of peripheral neuropathy, LFT's, S/Sx of hepatitis. |
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Pyrazinamide;
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB
MOA; converted to pyrazinoic acid, ↓ pH. ADR; malaise, n/v, myalgia, hepatotoxicity, kidney toxicity, gout. Precaution; renal or liver failure, gout, DM, preg C CI; hypersensitivity, acute gout, severe liver dx. Dose; 1000-3000 qd based on wt, ↓ w/renal impairment. Monitoring; LFT, uric acid, kidney fxn tests. |
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Rifampin;
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB
MOA; inhibist RNA synthesis, ABX. ADR; dedema, flushing, ataxia, mental ▲s, dizziness, blood dyscrasias, acute renal failure, rash, n/v/d, pancreatitis, ↑LFT, flu sx. Precaution; liver impairment, caution w/pyrazinamide/alcholism, discolors urine, saliva, sweat & tears, drug interactions, preg C CI; hypersensitivity, pretease inhibitors Dose; 10mg/kg/day Monitoring; LFT, CBC, mental status |
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Streptomycin;
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB
MOA; inhibits bacterial protein synthesis, aminoglycoside ABX. ADR; hypotension, neurotoxicity, n/v, ototoxicity, nephrotoxicity. Precaution; Black box warning for above ADR, renal impairment, nerve disorders, hearing loss, bacterial super infection. CI; hypersensitivity, PREGNANCY. Dose; 15mg/kg/day Monitoring; hearing/tinnitus, Bun Cr, drug level |
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Aminosalicylic Acid;
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; adjunctive tx in TB
MOA; competitive antagonist w/PABA ADR; n/v, blood dyscrasias, hepatitis, optic neuritis Precaution; hepatic/renal dysfunction, ulcer, nasal polyps, asthma, preg C. CI; hypersensitivity Dose; 150mg/kg/day in 2-3 doses. Monitoring; adverse rxns |
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Capastat (capreomycin);
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB
MOA; ABX, exact MOA unknown ADR; ototoxicity, nephrotoxicity, eosinophillia, hypokalemia Precaution; Box warning of above ADR, preg C, treatogenic CI; hypersensitivity Dose; 1gm/day for 60-120days, then 1gm 2-3 X q week Monitoring; hearing tests, renal fxn, LFT, K. |
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Seromycin (cycloserine);
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; adjunctive tx for TB
MOA; inhibits bacterial cell wall formation, ABX. ADR; arrhythmia, drowsiness, HA, dizziness, vertigo, seizure, psychosis, vit b12 folate defiency. Precaution; epilepsy, depression, anxiety, psychosis, renal impairment, alcoholism, preg C. CI; hypersensitivity Dose; 250 mg q 12hrs for 2wks, then 500mg-1gm for 18-24mos Monitoring; renal, hepatic, blood tests, cycloserine level. |
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Trecator (ethionamide);
Use; MOA; ADR; Precaution; CI; Dose; Monitoring; |
Use; TB tx when 1st line tx have failed.
MOA; inhibits peptide synthesis. ADR; hypotension, depression, dizziness, rash, hypoglycemia, hypothyroidism, n/v, impotence, hepatitiis, peripheral neuritis, optic neuritis Precaution; DM, cycloserine/isoniazid Dose; 15-20mg/kg/day Monitoring; LFT, thyroid fxn test, eye exam |