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34 Cards in this Set

  • Front
  • Back

Acetylcholine

Direct Acting


Cholinergic Agonist


1)Decrease HR


2)Decrease BP


3)Increase salivary/intestinal Secretions


4)Increase bronchioar secreations


5)Increase tone of detrusor urinae muscle


6)Constriction of sphincter pupillae


7) Stimulate cillary muscle

Bethanecol

Urecholine


Urinary Retention and Increase GI motility


Direct acting


Cholinergic Agonist

Carbachol

Direct Acting


Cholinergic Agonist


Constricts Pupils


Eye Surgery


Pilocarpine

Direct Acting


Cholinergic Agonist


Acute Glucoma (Lowers Intraocular pressure)

Ambenonium

Mytelase


indirect reversible


Cholinergic Agonist

Donepezil

Aricept


Alzhimers


Indirect reversible


Cholinergic Agonist

Galantamine

Razadyne


alzhimers tx


Indirect reversible


Cholinergic Agonist

Neostigmine

Prostigmin


indirect reversible


Cholinergic Agonist


Myastinia Gravis


Prevents Post Abdominal Distention

Physostigmine

Antrilirum


Cholinergic Agonist


indirect reversible


Increase intestinal and bladder motility


Miosis


Glucoma Treatment

Pyridostigmine

Mestinon


Cholinergic Agonist


indirect reversible


A cholinesterase inhibitor used in chronic management of myasthenia gravis

Rivastigmine

Exelon


alzhimers tx


indirect reversible


Cholinergic Agonist

Echothiophate

Phospholine Iodide


perminetly inactivates acetylcholinesterase


Indirect irreversible


Cholinergic Agonist

Isoflurophate

Indirect irreversible


Cholinergic Agonist


Atropine

Cholinergic Antagonist


Antimuscarinic Agent


Mydriasis, Reduce GI activity, reduce hypermotility in Urinary Tract, Increase HR at High doses, lower HR in lower doses. Blocks salivary glands


Scopolamine

Transderm-Scop


Antimuscarinic Agent


Cholinergic Antagonist


anti-motion sickness

Ipratropium

Atrovent


Cholinergic Antagonist


Antimuscarinic Agent


Treating asthma and COPD


Nicotine

Cholinergic Antagonist


Ganglionic Blocker


Increase BP, Increase HR, Increase peristalsis and secretions.



At higher doses the BP fall due to ganglionic blockade.

Benztropine

Congentin


Antimuscarinic Agent


Cholinergic Antagonist

Oxybutynin

Ditropan


Antimuscarinic Agent


Cholinergic Antagonist

Triotropium

Spiriva


Antimuscarinic Agent


Cholinergic Antagonist



Trihexyphenidyl

Artane


Antimuscarinic Agent


Cholinergic Antagonist

Albuterol

Adrenergic Antagonist


Direct Acting


Bronchodilator

Dobutamine

Dobutrex


Adrenergic Agonist


Direct Acting


Increase Cardiac Output in CHF pt's


Epinephrine

Adrenergic Agonist


Direct Acting


Increase Myocardial contractility, Increase HR, Cardiac Output Increases, and heart oxygen demand Increases Bronchodilation


Hyperglycemia, Lipolysis


Tx: Acute Asthma, Anaphylatic shock, Glaucoma, Anesthetics


Dopamine

Adrenergic Agonist


Direct Acting


Cardio: Inotropic (force) and chronotropic (rate) effects


Renal/Visceral: Increase blood flow to kidneys


Tx : Shock

Norepinephrine

Adrenergic Agonist


Direct Acting


Increase peripheral resistance (vasocontriction)

Isoproterernol

Isuprel


Adrenergic Agonist


Direct Acting


increase Myocardial contractility, Increase HR, Cardiac Output Increases


Phenylephrine

Sudafed


Adrenergic Agonist


Direct Acting


Vasoconstrictor that raises BP, Nasal Decongestant, used topically on nasal mucosa

Formoterol

Adrenergic Agonist


Direct Acting


Broncho-dilation


long lasting B2 agonist (Albuterol x3 days)

Salmeterol

Adrenergic Agonist


Direct Acting


Broncho-dilation


long lasting B2 agonist (Albuterol x3 days)

AMPHETAMINE

Adderall


indirect acting Adrenergic Agonist


Increase BP,


Tx: Hyperactivity in children, narcolepsy, appetite control


Adverse Effects: Arrhythmia, HA, insomnia, tremors

Cocaine

indirect acting Adrenergic Agonist


Reuptake inhibitor

Trebutaline

Brethine


Adrenergic Agonist


Direct Acting

Ephedrine

Adrenergic Agonist


Direct and Indirect Acting