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18 Cards in this Set

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  • Back
Lunesta
Eszopiclone
Sedative Class 4
No generic
Tabs(1,2,3mg)
Dosing: 1mg elderly, 2mg nonelderly BEFORE BEDTIME
Tx: insomnia
MoA: cyclopyrrolone (pyrrolopyrazine), gaba agonist
Di's: inc cns depression with cns depressants; cyp3a4 inhibitors/inducers
Ci's: insomnia > 10 days may be sign of phyical or psychiatric disorder
Ae's: drowsy, headache, taste
PxCx: Take at bedtime, on empty stomach, drowsy/machinery/alertness, avoid alcohol, WARNING:habit forming, withdrawls with sudden d/c
Ambien
Zolpidem tartrate
Sedative Class 4
Tabs(5,10mg)
Tabs CR(6.25,12.5mg)
Dosing: one tab before bedtime
Tx: insomnia
MoA: imidazopyradine, gaba agonist
Di's: inc cns depression with cns depressants
Ci's: <nothing memorable>
Ae's: drowsy, headache, nausea
PxCx: drowsy/machinery/alertness, avoid alcohol, WARNING:habit forming, swallow ambien CR whole
Trileptal
Oxcarbazepine
Antiepileptic
Tabs(150,300,600mg)
Susp(60mg/5ml)
Dosing: start with 300mg BID
Tx: Partial seizures
MoA: Na+ channel blocker
Di's: phenobarbital, phenytoin, valproic acid, cyp3a4/5 induction
Ci's: hypersensitivity rxns
Ae's: dizzy, somnolence, fatigue, ataxia, abnormal vision, n&v
PxCx: drowsy/machinery/alertness, avoid alcohol, shake susp well, take w/wo meals
Keppra
Levetiracetam
Anticonvulsant
Tabs(250,500,750,1000mg), tabs ER, soln
Dosing: 500mg BID
Tx: Partial seizures
MoA: pyrolidine deriv
Di's: none significant
Ci's: dec slowly to avoid triggering seizure
Ae's: dizzy, somnolence, asthenia, infection, hostility
PxCx: drowsy/machinery/alertness, dont d/c, taper off slowly
Topamax
Topiramate
Antiepileptic
Sprinkle caps(15, 25mg), tabs
Dosing: 100-200mg BID
Tx: seizures, migraines
MoA: Na+ channel blocker, gaba agonist
Di's: inc cns depression with cns depressants; estrogen, metformin, phenytoin, carbamazepine, valproic acid, hctz
Ci's: hyperchloremia, metabolic acidosis, glaucoma
Ae's: fatigue, nervousness, concentration, confusion, depression, dec weight
PxCx: contact doc if ocular pain and/or dec acuity, drowsy/machinery/alertness, avoid alcohol, hydrate well to avoid kidney stones, dont chew sprinkles
Dilantin, Kapseals
Phenytoin sodium (extended)
Antiepileptic
Caps(30,100mg)
Dosing: 100mg TID
Tx: tonic-clonic and psychomotor seizures
MoA: inc Na+ ion extrusion from neurons and cardiac myocytes
Di's: amiodarone, chloramphenicol, cimetidine, disulfiram, isoniazid, oral anticoagulants, sulfonamides, fluconazole, trimethazole, antineoplastics, carbamazepine, rifampin, sucralfate, disopyramide, theophillines, oral contraceptives, and many others!
Ci's: d/c if rash appears
Ae's: Ataxia, slurred speech, mental confusion, rash
PxCx: drowsy/machinery/alertness, call doc if rash appears, dont d/c w/o consult, take w/ food, diabetics monitor blood glucose
Lamictal
Lamotrigine
Antiepileptic
Tabs, chewable(5,25mg), odt, er
Dosing: 25-200mg QD
Tx: seizures
MoA: Na+ channel blocker
Di's: phenytoin, carbamazepine, phenobarbital, rifampin, valproic acid, oral contraceptives
Ci's: life threatening rashes during first 2 weeks
Ae's: dizzy, ataxia, somnolence, headache, rash, n&v, blurred vision, diplopia(double vision)
PxCx: report rash/hypersensitivity, drowsy/machinery/alertness, report if pregnant, dont change dosage w/o consult
Tegretol, Carbatrol, Equetrol
Carbamazepine
Anticonvulsant
Tabs(200mg), chewables(100mg), er, caps, susp
Dosing: 800-1200mg 3-4 dd's
Tx: seizures, trigeminal neuralgia pain
MoA: dec synaptic response/potential
Di's: oral anticoags, valproic acid, pancuronium, cimetidine, isoniazid, diltiazem, fluoxetine, propoxyphene, verapamil, macrolides, hydantoins, doxycycline, haloperidol, lithium, grapefruit juice
Ci's: bone marrow depression, moa-i, many other states...
Ae's: dizzy/drowsy, n&v, unsteadiness
PxCx: drowsy/machinery/alertness, avoid alcohol, shake susp well, take w/ food/milk, swallow er whole, call doc if rash/fever/ulcers/bruising, drink with full glass of water for chewable
Lyrica
Pregabalin
Anticonvulsant/antineuralgic
Class 5
Caps, soln(20mg/ml)
Dosing: 150mg in 2-3 dd's
Tx: diabetic neuropathy, postherpetic neuralgia, partial seizures, fibromyalgia
MoA: alpha2-delta agonist in cns tissue
Di's: inc cns depression with cns depressants, thiazolidinedione antidiabetics may inc edema
Ci's: rare rhabdomyolysis/myopathy
Ae's: dizzy, somnolence, dry mouth
PxCx: taper off gradually, drowsy/machinery/alertness, avoid alcohol, dont suddenly d/c, take w/wo meals, report muscle pain/fever, soln must be used w/in 45 days of opening
Neurontin
Gabapentin
Anticonvulsant/antineuralgic
Caps, tabs(600, 800mg), soln(250/5ml)
Dosing: 900-1800mg in 3 dd's
Tx: partial seizures, postherpetic neuralgia
MoA: unknown
Di's: Antacids dec BA
Ci's: caution with kids < 12
Ae's: somnolence, dizzy, ataxia, fatigue, nystagmus
PxCx: dont d/c suddenly(taper), drowsy/machinery/alertness, avoid alcohol, take w/wo meals
Depakote
Divalproex sodium
Anticonvulsant/antipsychotic
Tabs coated, er, sprinkle caps(125mg)
Dosing: 250mg TID
Tx: petit mals, partials, mania/bipolar, migraine prophylaxis
MoA: inc's gaba
Di's: aspirin, carbamazepine, dicumarol, phenobarbital, phenytoin, clonazepam
Ci's: (contra)hepatic disease, life threatening pancreatitis, suicide ideation
Ae's: n&v, asthenia, somnolence, dizzy, diarrhea
PxCx: dont d/c suddenly, drowsy/machinery/alertness, take w/ food/milk if gi upset, dont chew sprinkles, contact doc if facial edema/weakness/malaise
Geodon
Ziprasidone HCL
Antipsychotic
No generic
Caps, inj(20mg/ml)
Dosing: 40-80mg BID
Tx: schizophrenia, mania/bipolar
MoA: antagonist of dopamine d2, serotonin 5ht2, histamine h1, and alpha1 rx's
Di's: carbamazepine, ketoconazole, quinidine, antiarrys, and many others
Ci's: (contra)demetia related psychosis, qt prolongation, recent mi, heart failure, and many cautions
Ae's: drowsy/dizzy, nausea, constipation, cold symptoms, asthenia, dry mouth
PxCx: can cause serious arrys, inform doc of every med you take, take w/ food, drowsy/machinery/alertness, avoid alcohol, dont d/c suddenly
Abilify
Aripiprazole
Antipsychotic
No generic
Tabs, odt, inj, soln(1mg/ml)
Dosing: 10-15mg QD
Tx: schizophrenia, mania/bipolar
MoA: partial agonist at dopamine d2 and serotonin 5ht1a, antagonist at 5ht2a rx's
Di's: cyp3a4 inhibitors and inducers affect plasma levels
Ci's: (contra)dementia related psychosis, many cautions
Ae's: headache, anxiety, insomnia, asthenia, n&v, constipation, drowsy, tardive dyskinesia
PxCx: drowsy/machinery/alertness, avoid alcohol
Risperdal
Risperidone
Antipsychotic
Tabs, odt, powder for inj, soln(1mg/ml)
Dosing: start with 1mg QD
Tx: schizophrenia, mania/bipolar, autistic anger
MoA: antagonist of dopamine d2 and serotonin 5ht2 rx's
Di's: levodopa, carbamazepine, fluoxetine, clozapine(antischizophrenia drug)
Ci's: (contra)dementia related psychosis
Ae's: extrapyramidal symptoms, insomnia, agitation, anxiety, n&v, tachycardia, rash
PxCx: may cause fainting initially so get up slowly, may impair judgement, avoid alcohol, take with food/milk if gi upset, avoid excess heat/sunlight, dont take otc's w/o consult
Zyprexa
Olanzapine
Antipsychotic
Tabs, odt, powder for susp and for inj
Dosing: 10-15mg
Tx: psychotic disorders, mania/bipolar, schizophrenia
MoA: antagonist of dopamine, serotonin, muscarinic, histamine, and alpha1 rx's
Di's: inc cns depression with cns depressants; omeprazole, rifampin, activated charcoal, carbamazepine
Ci's: (contra)dementia related psychosis
Ae's: somnolence, agitation, nervousness, hostility, dizzy, constipation
PxCx: may cause fainting initially so get up slowly, drowsy/machinery/alertness, w/wo meals, dont change dosage, zydis(odt) tabs must be used immediately once opened
Seroquel
Quetiapine fumerate
Antipsychotic
Tabs, er
Dosing: 300-400mg in 2-3 dd's
Tx: schizophrenia, bipolar depression, mania/bipolar, major depressive disorder(ER tabs only)
MoA: antagonist of dopamine, serotonin, histamine, alpha1&2 rx's
Di's: inc cns depression with cns depressants
Ci's: (contra)dementia related psychosis, suicide ideation
Ae's: somnolence, dizzy, constipation, dry mouth
PxCx: may cause fainting initially so get up slowly, drowsy/machinery/alertness, take w/wo meals, dont change dosage, swallow ER whole
BuSpar
Buspirone HCL
Antianxiety agent
Tabs(5,10,15,30mg)
Dosing: 5-10mg QID
Tx: anxiety
MoA: inc metab of norepi, presynaptic dopamine agonist, serotonin agonist
Di's: MAO-i inc bp, grapefruit juice inc's plasma levels
Ci's: caution with hepatic and renal impairment
Ae's: skin rash, tachycardia, nervousness, insomnia, headache, fatigue, dizzy/drowsy
PxCx: drowsy/machinery/alertness, report involuntary movement of tongue or face(may cause parkinsons or tardive dyskinesia), avoid grapefruit juice
Prozac
Fluoxetine HCL
Antidepressant
Tabs(10,20mg),caps(10,20,40mg),caps er,liquid
Dosing: 10-40mg
Tx: depression, ocd, bulimia nervosa, panic disorder
MoA: SSRI
Di's: MOA-i(serious), thioridazine, tca, benazodiazepines, phenytoin, carbamazepine, tryptophan, sumatriptan, aspirin, nsaid
Ci's: (contra)MAO-i and thioridazine, antidepressants inc suicidal thoughts in kids
Ae's: nausea, insomnia, anorexia, headache, nervousness, drowsy, tremor, diarrhea, sweating, asthenia, dec libido
PxCx: observe changes in mood, may inc suicidal thoughts, drowsy/machinery/alertness, avoid alcohol, takes up to 2 weeks to see therapeutic effects, dont d/c suddenly, call doc if rash or hives appear