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44 Cards in this Set

  • Front
  • Back
Norepinephrine
Alpha-1, Beta-1 Agonist
vasoconstrictive increase in blood pressure
Epinephrine
Alpha 1, Beta 1, Beta 2 agonist
vasoconstrictive benefit to retail local anesthetics in the injection site.
Pseudoephedrine
Alpha 1, Beta 1 agonist
vasoconstrictive decongestant
Phenylephrine
Alpha 1 agonist
vasoconstrictive decongestant
vasoconstrictor in cases of hypotension due to anesthesia in surgery raise BP
Methoxamine
Alpha 1 agonist
vasoconstrictor in cases of hypotension due to anesthesia in surgery. Raise BP
Prazosin, Doxazosin
Alpha 1 Antagonist
Antihypertensive
Terazosin
Alpha 1 Antagonist
antihypertensive, BPH
Tamsulosin, Alfuzosin, Silodosin
Alpha 1 Antagonist
BPH
Phentolamine
Alpha 1 and Alpha 2 short acting antagonist
antihypertensive, diagnostic pheochromocytoma, management of pheochromocytoma, Alpha 2 block increases reflexive tachycardia when BP too low
Phenoxybenzamine
Alpha 1 and Alpha 2 long acting antagonist
Antihypertensive, management of pheochromcytoma, alpha 2 block for reflexive tachycardia
Clonidine, Guanfacine, Guanabenz
Alpha 2 Agonist
antihypertensive
Methyldopa
Alpha 2 Agonist
Antihypertensive
Drug of choice for pregnancy hypertension
ephedrine
alpha 1, beta 1, beta 2 agonist
long acting bronchodilator
not usually used anymore
Isoproternol
beta 1, beta 2 agonist
Bronchodilator with strong cardiac side effect (arrhythmia)
Dobutamine
beta 1 agonist
cardiotonic, improves ventricular contractility in heart failure
Dopamine
beta 1, D1, D2 agonist
improves cardiac performance in shock state and improves renal blood flow
Metaproterenol
beta 2 agonist (inhalation)
bronchodilator
albuterol, terbutaline, pirbuterol
Beta 2 agonist inhalation short acting
bronchodilator
Salmeterol, Formotorol
Beta 2 agonist inhalation long acting
bronchodilator
Propanolol
Beta 1 and beta 2 antagonist
antihypertensive, antianginal, antiarrhythmic
Timolol
Beta 1 and Beta 2 antagonist
Glaucoma, Hypertension
Nadolol
Beta 1 and Beta 2 antagonist
hypertension, antianginal, antiarrhthmic, migraine headache
Carvedilol
Alpha 1 and Beta 1 and Beta 2 antagonist
pheochromocytoma, CHF
Atenolol
Beta 1 antagonist
antihypertensive, antianginal
Metoprolol
Beta 1
Antihypertensive, antianginal, CHF
Acebutolol
Beta 1 (ISA) funtional beta 1 antagonist (partial agonist)
antihypertensive, antiarrhythmic
Bisoprolol
Beta 1 antagonist
antihypertensive, antianginal, CHF
Pindolol
Beta 1 and beta 2 partial agonist (functional antagonist)
antihypertensive
Nicotine and Acetylcoline
Nicotinic agonist
physostigmine
anticholinesterase
antimuscarinic poisoning
neostigmine, pyridostigmine
anticholinesterase
myasthenia gravis
Sarin
Anticholinesterase, irreversible
toxin
Mecamylamine
Ganglionic blocker
antihypertensive, loss of predominant function
Curare
NM, nondepolarizing blocker, competitive antagonist
skeletal muscle relaxation
Succinycholine
NM, depolarizing blocker, persistent depolarization
skeletal muscle relaxation
Bethanacol
M3 agonist
GI and urinary stasis, minimal toxicity
Pilocarpine (topical)
M3 agonist
Glaucoma (relieves congestion, toxicity = near vision)
Echothiophate
Indirect agonist via anticholinesterase, long lasting
Glaucoma
Acetylcholine
M2, M3, Nn and Nm agonists
neurotransmitter
Anticholinesterases
M2, M3, Nn, Nm, reversible indirect agonists
Atropine
M2 and M3 antagonists
opthalmic: mydriasis and cycloplegia
GI and Bladder relation
counteracts anticholinesterase
Tropicamide, Cyclopentolate
M3 antagonist
Opthalmic: mydriasis and cycloplegia
Scopolamine
M3 antagonist
motion sickness, bronchodilation, reverse bradycardia, dry airway in anesthesia
Ipratropium
M3 antagonists
bronchodilator in asthma and COPD