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51 Cards in this Set

  • Front
  • Back
8 adrenergic agonists
- Epinephrine
- Isoproterenol
- Dopamine
- Dobutamine
- Phenylephrine
- Phenylpropanolamine
- Albuterol
- Clenbuterol
5 adrenergic antagonists
- Phenoxybenzamine HCL
- Propranolol
- Timolol
- Atenolol
- Carvedilol
8 cholinergic agonists
- Bethanechol
- Carbachol
- Pilocarpine
- Physostigmine
- Neostigmine
- Pyridostigmine
- Edrophonium
- Organophosphates
3 cholinergic antagonists
- Atropine
- Glycopyrolate
- N-butylscopalammonium Br
Receptors that Epinephrine works on
- α
- B
α receptor affinity of epinephrine compared to isoproterenol
Epi >>> Iso
B receptor affinity of epinephrine compared to isoproterenol
Iso > Epi
Receptors affected by Isoproterenol
Selective B agonist
Receptors affected by Dopamine
α

B
Receptors affected by Dobutamine
B
Receptors affected by Phenylephrine
α1

B1 (high doses)
Receptors affected by Phenylpropranolamine
α

B
Receptors affected by Albuterol
B2 selective
Receptors affected by Clenbuterol
B2 selective
Receptors affected by Phenoxybenzamine HCL
α blocker
Receptors affected by Propranolol
B blocker
Receptors affected by Timolol
B blocker
Receptors affected by Atenolol
B1 Blocker
Receptors affected by Carvedilol
α1 blocker

β blocker
Receptors affected by Bethanechol
Muscarinic
Receptors affected by Carbachol
Muscarinic

Nicotinic
Receptors affected by Pilocarpine
Muscarinic
Receptors affected by Physostigmine
ACHase inhibitor

Muscarinic

Nicotinic
Receptors affected by Neostigmine
ACHase inhibitor
Receptors affected by Edrophonium
ACHase inhibitor
Receptors affected by Pyridostigmine
ACHase inhibitor
Receptors affected by Organophosphates
ACHase inhibitor

Muscarinic

Nicotinic
MoA of Bethanechol
Direct acting PSNS
MoA of Carbachol
Direct acting PSNS
MoA of Pilocarpine
Cholinomimetic alkaloid
MoA of Physostigmine
Reversible Cholinesterase inhibitor
MoA of Neostigimine
Reversible Cholinesterase inhibitor
MoA of Edrophonium
Reversible Cholinesterase inhibitor
MoA of Pyridostigmine
Reversible Cholinesterase inhibitor
MoA of Organophosphates
Irreversible Cholinesterase inhibitor
Reversible Cholinesterase inhibitors (4)
- Physostigmine
- Neostigmine
- Edrophonium
- Pyridostigmine
Irreverisble cholinesterase inhibitor
Organophosphates
3 muscarinic blockers
- Atropine
- Glycopyrolate
- N-butylscopolammonium Br
MoA of Atropine
Blocks ACH from binding to muscarinic receptors
MoA of Glycopyrolate
Blocks ACH from binding to muscarinic receptors
MoA of N-butylscopolammonium Br
Blocks ACH from binding to muscarinic receptors
Receptors of Atropine
Muscarinic blocker
Receptors of Glycopyrolate
Muscarinic blocker
Receptors of N-butylscopolammonium Br
Muscarinic blocker
3 muscarinic blockers
- Atropine
- Glycopyrolate
- N-butylscopolammonium Br
MoA of Atropine
Blocks ACH from binding to muscarinic receptors
MoA of Glycopyrolate
Blocks ACH from binding to muscarinic receptors
MoA of N-butylscopolammonium Br
Blocks ACH from binding to muscarinic receptors
Receptors of Atropine
Muscarinic blocker
Receptors of Glycopyrolate
Muscarinic blocker
Receptors of N-butylscopolammonium Br
Muscarinic blocker