Wvsom Pharm 2013

Front 1

Norepinephrine

Back 1

Direct Acting Adrenal Mimetics
parenteral
low oral bioavailablility
Anaphylaxis

Front 2

Dopamine

Back 2

Direct Acting Adrenal Mimetics
activates β1 and α receptors

Front 3

Xylometazoline

Back 3

α1 selective agonists
long duration of action
nasal decongestant

Front 4

Oxymetazoline

Back 4

α1 selective agonists
long duration of action, also activates α2
nasal decongestant

Front 5

Brimonidine

Back 5

α2 selective agonists
opthalmic

Front 6

Apraclonidine

Back 6

α2 selective agonists
opthalmic

Front 7

Metaproterenol

Back 7

β2 selective agonists
lungs

Front 8

Pirbuterol

Back 8

β2 selective agonists
lungs

Front 9

Terbutaline

Back 9

β2 selective agonists
stop premature labor

Front 10

Formoterol

Back 10

β2 selective agonists
lungs

Front 11

Arformoterol

Back 11

β2 selective agonists
lungs

Front 12

Tyramine

Back 12

Indirect Acting Adrenomimetics
Not a drug, from gut bacteria
release of NE

Front 13

Ephedrine

Back 13

Mixed Acting Adrenomimetics
acts on α and β, releases NE, crosses BBB
Asthma, COPD, Nasal Congestion

Front 14

Prazosin

Back 14

α Antagonists, selective reversible
hypertension, Raynauds

Front 15

Doxazosin

Back 15

α Antagonists, selective reversible
hypertension

Front 16

Nadolol

Back 16

β Antagonists, nonselective, competitive, reversible
Migraine

Front 17

Timolol

Back 17

β Antagonists, nonselective, competitive, reversible
Migraine

Front 18

Pindolol

Back 18

β Antagonists, nonselective, competitive, reversible

Front 19

Carteolol

Back 19

β Antagonists, nonselective, competitive, reversible

Front 20

Levobunolol

Back 20

β Antagonists, nonselective, competitive, reversible

Front 21

Metoprolol

Back 21

β1 Antagonists, selective, competitive, reversible
migraine

Front 22

Acebutolol

Back 22

β1 Antagonists, selective, competitive, reversible

Front 23

Betaxolol

Back 23

β1 Antagonists, selective, competitive, reversible

Front 24

Bisoprolol

Back 24

β1 Antagonists, selective, competitive, reversible

Front 25

Acetylcholine

Back 25

Direct Acting Muscarinic Agonists

Front 26

Bethanechol

Back 26

Direct Acting Muscarinic Agonists
most effect on M of urinary bladder and GI
Post-Op abdominal distention, urinary retention

Front 27

Muscarine

Back 27

Direct Acting Muscarinic Agonists
mushroom poisoning

Front 28

Physostigmine

Back 28

Reversible AChE Inhibitors
acts on all cholinergic synapses, passes BBB
Miotic, glaucoma
reverse antimuscarinic

Front 29

Neostigmine

Back 29

Reversible AChE Inhibitors
Post op urinary retention, abd distension, myasthenia gravis

Front 30

Echothiophate

Back 30

Irreversible AChE Inhibitors
Miosis, glaucoma

Front 31

Parathion

Back 31

Irreversible AChE Inhibitors
Insecticide

Front 32

Malathion

Back 32

Irreversible AChE Inhibitors
Insecticide, lice

Front 33

Sarin

Back 33

Irreversible AChE Inhibitors
P-O bond not hydrolysable, highly lethal
Nerve gas, kills via resp. failure (need 2-PAM and Atropine)

Front 34

Tubocurarine

Back 34

Neuromuscular Blockers (non-depolarizing)

Front 35

Atracurium

Back 35

Neuromuscular Blockers (non-depolarizing)

Front 36

Cisatracurium

Back 36

Neuromuscular Blockers (non-depolarizing)

Front 37

Mivacurium

Back 37

Neuromuscular Blockers (non-depolarizing)

Front 38

Pancuronium

Back 38

Neuromuscular Blockers (non-depolarizing)

Front 39

Vecuronium

Back 39

Neuromuscular Blockers (non-depolarizing)

Front 40

Scopolamine

Back 40

Cholinolytics
Miosis, pre-op

Front 41

Tropicamide

Back 41

Cholinolytics
Mydriasis, cycloplegia

Front 42

Tiotropium bromide

Back 42

Cholinolytics
Inhalation

Front 43

Tolterodine

Back 43

Cholinolytics

Front 44

Oxybutynin chloride

Back 44

Cholinolytics

Front 45

Darifenacin HBr

Back 45

Cholinolytics