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120 Cards in this Set

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Oral Rehydration Therapy
N/A
Receptor, Agonist v. Antagonist
Bismuth (Pepto-Bismol)
N/A
Receptor, Agonist v. Antagonist
Fiber, bulk agents ["lignin" (Psyllium, Polycarbophil)]
N/A
Receptor, Agonist v. Antagonist
Saline Laxatives: MgSO4 (Epsom)
N/A
Receptor, Agonist v. Antagonist
Saline Laxatives: NaPO4 (FLEET)
N/A
Receptor, Agonist v. Antagonist
Lubiprostone
ClC2 Agonist
Receptor, Agonist v. Antagonist
Octreotide (Somatostatin mimetic)
ST2 Agonist
Receptor, Agonist v. Antagonist
Bethanechol
M1/2/3 Agonist
Receptor, Agonist v. Antagonist
Neostigmine
AChE Inhibitor
Receptor, Agonist v. Antagonist
Loperamide
Mu Agonist
Receptor, Agonist v. Antagonist
Diphenoxylate
Mu Agonist
Receptor, Agonist v. Antagonist
Clonidine
a2 Agonist
Receptor, Agonist v. Antagonist
Metoclopramide
D2 Antagonist (& 5-HT4 Agonist)
Receptor, Agonist v. Antagonist
Domperidone
D2 Antagonist
Receptor, Agonist v. Antagonist
Alosetron
5-HT3 Antagonist
Receptor, Agonist v. Antagonist
Cisapride
5-HT4 Agonist
Receptor, Agonist v. Antagonist
Tegaserod
5-HT4 Agonist
Receptor, Agonist v. Antagonist
Prucalopride
5-HT4 Agonist
Receptor, Agonist v. Antagonist
Ondansetron
5-HT3 Antagonist
Receptor, Agonist v. Antagonist
Scopolamine
M1(2/3) Antagonist
Receptor, Agonist v. Antagonist
Pirenzipine
M1 Antagonist
Receptor, Agonist v. Antagonist
Promethazine
H1 Antagonist, M1 Antagonist, D2 Agonist
Receptor, Agonist v. Antagonist
Dimenhydrinate
H1 Antagonist, D2 Agonist
Receptor, Agonist v. Antagonist
Metoclopramide
D2 Antagonist, 5-HT4 Agonist
Receptor, Agonist v. Antagonist
Chlorpromazine
D2 Antagonist
Receptor, Agonist v. Antagonist
Aprepritant (EMEND)`
NK1 Antagonists
Receptor, Agonist v. Antagonist
Dronabinol (D9-THC)
CB1 Agonist
Receptor, Agonist v. Antagonist
Ipecac
Mucosal Irritation
Receptor, Agonist v. Antagonist
Apomorphine
D2(/D1) Agonist
Receptor, Agonist v. Antagonist
Prednisone
N/A (Immune Antagonist)
Receptor, Agonist v. Antagonist
Sulfalazine
COX Inhibitor
Receptor, Agonist v. Antagonist
Azathioprine -> 5-MP
N/A
Receptor, Agonist v. Antagonist
MTX
Folate Inhibitor
Receptor, Agonist v. Antagonist
Infliximab
TNFa Inhibitor
Receptor, Agonist v. Antagonist
CaCO3
N/A
Receptor, Agonist v. Antagonist
NaHCO3
N/A
Receptor, Agonist v. Antagonist
Al(OH)3
N/A
Receptor, Agonist v. Antagonist
Mg(OH)2
N/A
Receptor, Agonist v. Antagonist
Cimetidine
H2 Antagonist
Receptor, Agonist v. Antagonist
Ranitidine
H2 Antagonist
Receptor, Agonist v. Antagonist
Pirenzipine
M1 Antagonist
Receptor, Agonist v. Antagonist
Atropine/Scopolamine
M1/2/3 Antagonist
Receptor, Agonist v. Antagonist
Omeprazole
H+/K+ ATPase
Receptor, Agonist v. Antagonist
Misoprostol
PGE1 Agonist
Receptor, Agonist v. Antagonist
Sucralfate
N/A
Receptor, Agonist v. Antagonist
Bismuth (Pepto-Bismol)
N/A
Receptor, Agonist v. Antagonist
Oral Rehydration Therapy
Acute Diarrhea
Main Indication
Bismuth (Pepto-Bismol)
Acute Diarrhea, Ulcer Healing
Main Indication
Fiber, bulk agents ["lignin" (Psyllium, Polycarbophil)]
Chronic Diarrhea
Main Indication
Saline Laxatives: MgSO4 (Epsom)
Chronic Diarrhea
Main Indication
Saline Laxatives: NaPO4 (FLEET)
Chronic Diarrhea
Main Indication
PEG
Bowel Prep (*Cathartic*)
Main Indication
Lubiprostone
IBS-C (women), CIC
Main Indication
Octreotide (Somatostatin mimetic)
*Gastrinoma*, Diarrhea[…]
Main Indication
Bethanechol
Post-op ileus: 2nd line (vs. Domperidone)
Main Indication
Neostigmine
Acute colonic (pseudo-)obstruction
Main Indication
Loperamide
Diarrhea: First Line! (Known Etiology)
Main Indication
Diphenoxylate
Diarrhea: First Line! (Known Etiology)
Main Indication
Clonidine
Diarrhea: Diabetic Neuropathy, Opiate Withdrawal
Main Indication
Metoclopramide
Post-op ileus: 1st-line
Main Indication
Domperidone
Post-op ileus: 2nd-line
Main Indication
Alosetron
IBS-D
Main Indication
Cisapride
IBS-C
Main Indication
Tegaserod
IBS-C
Main Indication
Prucalopride
IBS-C
Main Indication
Ondansetron
Chemo-Induced N/V
Main Indication
Scopolamine
PROPHYLACTIC Motion Sickness
Main Indication
Pirenzipine
(Only one…)
Main Indication
Promethazine
ACUTE Motion Sickness, Acute N/V
Main Indication
Dimenhydrinate
ACUTE Motion Sickness, Acute N/V
Main Indication
Metoclopramide
Diabetic neuropathy w/ n/v; Post-op N/V
Main Indication
Chlorpromazine
Diabetic neuropathy w/ n/v; Post-op N/V
Main Indication
Aprepritant (EMEND)`
??
Main Indication
Dronabinol (D9-THC)
Last-Line: Chemo n/v, chronic dz; Decreased Appetite
Main Indication
Ipecac
Emergency emesis
Main Indication
Apomorphine
NONCOMPLIANT Emergency Emesis
Main Indication
Prednisone
UC/CD
Main Indication
Sulfalazine
UC
Main Indication
Azathioprine -> 5-MP
UC/CD
Main Indication
MTX
UC
Main Indication
Infliximab
UC/CD
Main Indication
CaCO3
GERD: 1st Line
Main Indication
NaHCO3
GERD: 1st Line
Main Indication
Al(OH)3
GERD: 1st Line
Main Indication
Mg(OH)2
GERD: 1st Line
Main Indication
Cimetidine
GERD: 1st/2nd Line
Main Indication
Ranitidine
GERD: 1st/2nd Line
Main Indication
Pirenzipine
Never used, only M1 drug
Main Indication
Atropine/Scopolamine
Never used for acid mgmt, only M1 drug
Main Indication
Omeprazole
GERD: 3rd-Line, Z-E/Gastrinoma
Main Indication
Misoprostol
GERD: NSAID-induced Peptic Ulcer PREVENTION/Healing
Main Indication
Sucralfate
GERD: Binds @ ulcer base (Protective)
Main Indication
Bismuth (Pepto-Bismol)
GERD: Ulcer Healing; *Traveler's Diarrhea*
Main Indication
Octreotide (Somatostatin mimetic)
"Diarrhea": Dumping syndrome, AIDS, acute variceal bleeds, vagotomy
Notes
Bismuth (Pepto-Bismol)
"Traveler's"
Notes
PEG
Can be used as laxative (low-dose w H2O)
Notes
Tegaserod
Caution v. Lubiprostone
Notes
Oral Rehydration Therapy
Cholera
Notes
Alosetron
Females, Tx-Unresponsive
Notes
Lubiprostone
IBS-C: v. Cisapride/Tegaserod
Notes
Omeprazole
Irreversible Inhibition
Notes
Dimenhydrinate
Less Muscarinic SE's, Less D2 SE's (EPS)
Notes
Fiber, bulk agents ["lignin" (Psyllium, Polycarbophil)]
Mild, "Old People"
Notes
Saline Laxatives: MgSO4 (Epsom)
Mild, "Old People"
Notes
Saline Laxatives: NaPO4 (FLEET)
Mild, "Old People"
Notes
Cisapride
Not available (FDA)
Notes
Prucalopride
Not yet FDA Approved
Notes
Bethanechol
Post-op ileus: 1. Metoclopramide, 2. Bethanechol v. Domperidone
Notes
Metoclopramide
Post-op ileus: 1. Metoclopramide, 2. Bethanechol v. Domperidone
Notes
Domperidone
Post-op ileus: 1. Metoclopramide, 2. Bethanechol v. Domperidone
Notes
Cimetidine
Promotes Ulcer healing, Good Long Term Maintenance
Notes
Ranitidine
Promotes Ulcer healing, Good Long Term Maintenance
Notes
Azathioprine -> 5-MP
Remission
Notes
Prednisone
REMISSION (UC/CD)
Notes
Clonidine
Safe w/ buprenorphine/naloxone, NOT CI w preg
Notes
Scopolamine
Some use in post-op n/v
Notes
Infliximab
Symptomatic Management (Not Remission)
Notes
Sulfalazine
UC- First-Line (Mild/Moderate); CD- only if SI-limited
Notes
MTX
UC: "Last-Line"
Notes
Neostigmine
usu used IH IV
Notes