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519 Cards in this Set
- Front
- Back
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-afil
Used for? |
Erectile dysfunction
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-ane
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inhalational general anesthetic
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-azepam
|
benzodiazepine
All have az in name |
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-azine
(two functions) |
phenothiazine (neuroleptic, antiemetic)
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-conazole
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antifungal
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-barbital
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barbiturate
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-caine
|
local anesthetic
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-cillin
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penicillin
|
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-cycline
(mechanism) |
tetracycline antibiotic, protein synthesis inhibitor
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-etine
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SSRI
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-ipramine
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TCA
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-navir
|
protease inhibitor
|
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-olol
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Beta antagonist
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-operidol
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Butyrophenone (neuroleptic)
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-oxin
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cardiac glycoside (inotropic agent)
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-phylline
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methylxanthine
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-pril
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ACE-I
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-terol
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Beta-2 agonist
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-tidine
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H2 antagonist
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-triptan
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5-HT1a agonists (migraine)
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-triptyline
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TCA
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-tropin
|
pituitary hormone
|
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-zosin
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alpha-1 antagonist
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-dronate
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bisphosphonate
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-sartan
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ARB
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-chol
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cholinergic/muscarinic agonist
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-stigmine
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anti-cholinesterase
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-mustine (and use)
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nitrosurea (cancer drugs)
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-curium/-curonium
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non-depolarizing neuromuscular blocking drug
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-statin
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HMG CoA Reductase Inhibitor
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-glitazone (mechanism)
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increases target cell response to insulin
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-bendazole
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anti-parasitic
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-dipine
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dihydropyridine Calcium channel blocker
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-prost
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PG analog
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-mab
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Ab
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Name some -azole antifungals
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fluconazole, ketoconazole, clotrimazole, miconazole, itraconazole, voriconazole
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Penicillinase-resistant penicillins
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Methicillin, nafcillin, dicloxacillin
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Methicillin
use? |
Penicillinase-resistant penicillins - used on non-MRSA staph
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Nafcillin
use? |
Penicillinase-resistant penicillins - used on non-MRSA staph
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Dicloxacillin
use? |
Penicillinase-resistant penicillins - used on non-MRSA staph
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Ampicillin
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aminopenicillins
(AMPed up penicillin) |
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Amoxicillin
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aminopenicillins
(AMPed up penicillin) |
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Aminopenicillins
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Ampicillin, amoxicillin (AMPed up PCN)
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Antipseudomonals
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Extended spectrum PCN
Ticarcillin, carbenicillin, piperacillin TCP: Takes Care of Pseudomonas |
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Ticarcillin
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Extended spectrum PCN anti-pseudomonals
Ticarcillin, carbenicillin, piperacillin TCP: Takes Care of Pseudomonas |
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Carbenicillin
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Extended spectrum PCN anti-pseudomonals
Ticarcillin, carbenicillin, piperacillin TCP: Takes Care of Pseudomonas |
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Piperacillin
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Extended spectrum PCN anti-pseudomonals
Ticarcillin, carbenicillin, piperacillin TCP: Takes Care of Pseudomonas |
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Cephalosporins
1st generation |
cefazolin, cephalexin
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Cefazolin
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Cephalosporin
1st generation |
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Cephalexin
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Cephalosporin
1st generation |
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Cefoxitin
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Cephalosporin
2nd generation |
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Cefaclor
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Cephalosporin
2nd generation |
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Cefuroxime
|
Cephalosporin
2nd generation |
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Cephalosporins
2nd generation |
Cefoxitin, cefaclor, cefuroxime
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Cephalosporins
3rd generation |
ceftriaxone, cefotaxime, ceftazidime
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Ceftriaxone
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Cephalosporin
3rd generation |
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Cefotaxime
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Cephalosporin
3rd generation |
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Ceftazidime
|
Cephalosporin
3rd generation |
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Cefepime
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Cephalosporin
4th generation |
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Cephalosporin
4th generation |
Cefepime
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Aztreonam
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beta-lactam AB
resistant to beta-lactamases |
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Imipenem/cilastatin
|
imipenem - broad-spectrum, beta-lactamase-resistant carbapenem
Cilastatin - inhibitor of renal dihydropeptidase 1 to decrease inactivation in renal tubules |
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Meropenem
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very strong, broad-spectrum AB
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Cilastatin
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adjunctive always given with imipenem to prevent its deactivation in renal tubules by dihydropeptidase 1
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Vancomycin
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AB - blocks cell wall formation by binding D-ala-D-ala
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Aminoglycoside e.g.s - 5
Hint - mnemonic of annoying bugs - buzz in your ears, making you pee |
GNATS
Gentamicin, Neomycin, Amikacin, Tobramycin, Streptomycin Nephrotoxic, Ototoxic, Teratogenic |
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Gentamicin
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Aminoglycoside
|
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Neomycin
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Aminoglycoside
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Amikacin
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Aminoglycoside
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Tobramycin
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Aminoglycoside
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Streptomycin
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Aminoglycoside
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Lincomycin
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not a macrolide, but similar
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Tetracyclines - Name 4
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Tetracycline, doxycycline, demeclocycline, minocycline
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Doxycycline
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Tetracycline
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Minocycline
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Tetracycline
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Macrolides
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Erythromycin, azithromycin, clarithromycin
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Erythromycin
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Macrolide
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Azithromycin
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Macrolide
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Clarithromycin
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Macrolide
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Chloramphenicol
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AB - 50S protein synthesis inhibitor
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Clindamycin
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AB - 50S protein synthesis inhibitor
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Know your micin/mycins!
|
Clindamycin - lincosamide AB
Lincomycin - not a macrolide but similar Azithromycin, Clarithromycin, Erythromycin - MACROLIDES (ACE) Gentamicin, Neomycin, Amikacin, Tobramycin, Streptomycin - AMINOGLYCOSIDES (GNATS) Vancomycin |
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Sulfonamides - name three
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Sulfamethoxazole (SMX), sulfisoxazole, sulfadiazine (silvadine is silver sulfadiazine)
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Sulfamethoxazole (SMX)
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Sulfonamide
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Sulfisoxazole
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Sulfonamide
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Sulfadiazine
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Sulfonamide
Found in "silvadene" - silver sulfadiazine |
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Trimethoprim (TMP)
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Bacteriostatic AB
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Fluoroquinolones
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Ciprofloxacin, Norfloxacin, ofloxacin, sparfloxacin, moxifloxacin, gatifloxacin, enoxacin
Nalidixic acid (quinolone) |
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Ciprofloxacin
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Fluoroquinolone
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Norfloxacin
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Fluoroquinolone
|
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Ofloxacin
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Fluoroquinolone
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Sparfloxacin
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Fluoroquinolone
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Moxifloxacin
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Fluoroquinolone
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Gatifloxacin
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Fluoroquinolone
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Enoxacin
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Fluoroquinolone
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Nalidixic acid
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Quinolone
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Metronidazole
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Antimicrobial/parasite
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Polymyxins
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topical AB (neosporin)
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Quinupristin/dalfopristin
Used for? |
Streptogramins
AB used for VRSA/VRE |
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Streptogramins
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quinupristin/dalfopristin
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Protease inhibitors
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All END in vir
Saquinavir, ritonavir, indinavir, nelfinavir, amprenavir |
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Saquinavir
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Protease inhibitor
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Ritonavir
|
Protease inhibitor
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Indinavir
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Protease inhibitor
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Nelfinavir
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Protease inhibitor
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Amprenavir
Hint: ends in -vir |
Protease inhibitor
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Ziduvodine
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ZDV, formerly AZT
Nucleoside Reverse Transcriptase Inhibitor |
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Didanosine
|
ddI
Nucleoside Reverse Transcriptase Inhibitor |
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Zalcitabine
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ddC
Nucleoside Reverse Transcriptase Inhibitor |
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Stavudine
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d4T
Nucleoside Reverse Transcriptase Inhibitor |
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Lamivudine
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3TC
Nucleoside Reverse Transcriptase Inhibitor |
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Abacavir
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Nucleoside Reverse Transcriptase Inhibitor
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Nucleoside Reverse Transcriptase Inhibitors
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NRTIs
Zidovudine (ZDV, formerly AZT), didanosine (ddI), zalcitabine (ddC), stavudine (d4T), lamivudine (3TC), abacavir |
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Non-nucleoside Reverse Transcriptase Inhibitors (NNRTIs)
All have what root in their names? Name three |
Nevirapine, Efavirenz, Delavirdine
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Nevirapine
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Non-nucleoside Reverse Transcriptase Inhibitor (NNRTI)
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Efavirenz
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Non-nucleoside Reverse Transcriptase Inhibitor (NNRTI)
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Delavirdine
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Non-nucleoside Reverse Transcriptase Inhibitor (NNRTI)
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Enfuvirtide
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Fusion inhibitor (HIV Tx)
|
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Fusion inhibitor
|
Enfuvirtide
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5-FU
Inhibits what? |
5-fluorouracil
Nucleotide synthesis inhibitor Inhibits thymidylate synthase |
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Hydroxyurea
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Nucleotide synthesis inhibitor
|
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6-MP
|
6-mercaptopurine
Nucleotide synthesis inhibitor |
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Methotrexate (MTX)
|
Nucleotide synthesis inhibitor
Antimetabolite anti-cancer drug |
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Cyclosporine
|
Immunosuppressant
|
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Tacrolimus (FK506)
|
Immunosuppressant
|
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Azathioprine
|
Immunosuppressant
|
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Muromonab-CD3 (OKT3)
(Class/purpose) |
Immunosuppressant
|
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OKT3
|
Muromonab-CD3 (OKT3)
Immunosuppressant |
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Sirolimus (rapamycin)
|
Immunosuppressant
|
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Mycophenolate mofetil
|
Immunosuppressant
|
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Daclizumab
|
Immunosuppressant
|
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FK506
|
Immunosuppressant
AKA: Tacrolimus |
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Thalidomide
|
Immunosuppressant
|
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Bethanechol
|
Direct cholinomimetic agonist
|
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Carbachol
|
Direct cholinomimetic agonist
|
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Pilocarpine
|
Direct cholinomimetic agonist
|
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Methacholine
|
Direct cholinomimetic agonist
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Direct cholinomimetic agonists
|
Bethanechol, Carbachol, Pilocarpine, Methacholine
|
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Neostigmine
|
Cholinomimetic agent: Indirect agonist (anti-AchE)
|
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Cholinomimetic agents: Indirect agonists (anti-AchE)
|
Neostigmine, Pyridostigmine, Edrophonium, Physostigmine, Echothiophate
|
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Pyridostigmine
|
Cholinomimetic agent: Indirect agonist (anti-AchE)
|
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Edrophonium
|
Cholinomimetic agent: Indirect agonist (anti-AchE)
|
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Physostigmine
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Cholinomimetic agent: Indirect agonist (anti-AchE)
|
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Echothiophate
|
Cholinomimetic agent: Indirect agonist (anti-AchE)
|
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Muscarinic antagonists
|
Atropine, Homatropine, Tropicamide, Benztropine, Scopolamine, Ipratropium, Oxybutynin, Glycopyrrolate, Methscopolamine, Propantheline
|
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Atropine
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Muscarinic antagonist
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Homatropine
|
Muscarinic antagonist
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Tropicamide
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Muscarinic antagonist
|
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Benztropine
|
Muscarinic antagonist
|
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Scopolamine
|
Muscarinic antagonist
|
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Ipratropium
|
Muscarinic antagonist
|
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Oxybutynin
|
Muscarinic antagonist
|
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Glycopyrrolate
|
Muscarinic antagonist
|
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Methscopolamine
|
Muscarinic antagonist
|
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Propantheline
|
Muscarinic antagonist
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Hexamethonium
|
Nicotinic antagonist
|
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Nicotinic antagonist
|
Hexamethonium
|
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Isoproteronol
|
Non-selective Beta agonist
|
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Dopamine
Effects on receptors? Effects on heart? |
Sympathomimetic
D1=D2 > beta > alpha Inotropic and chronotropic |
|
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Dobutamine
Hint: used in cardiogenic shock and heart failure |
Beta1 > Beta2 agonist
|
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Phenylephrine
|
alpha1 > alpha2 agonist
|
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Sympathomimetics – Indirect
|
Amphetamine, Ephedrine, Cocaine
|
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Amphetamine
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Sympathomimetic – Indirect
Indirect general agonist |
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Ephedrine
|
Sympathomimetic – Indirect
Indirect general agonist |
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Cocaine (non-anesthetic use)
|
Sympathomimetic – Indirect
Indirect general agonist reuptake inhibitor |
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Sympathoplegics - name 2
|
Clonidine, alpha-methyldopa
|
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Clonidine
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Sympathoplegic (decreases sympathetic discharge or its effect on the CNS, specifically via alpha2 agonistic effect)
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Alpha-methyldopa
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Sympathoplegic (decreases sympathetic discharge or its effect on the CNS)
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Selective beta2 agonists:
|
MAST – metaproteronol, albuterol, salmeterol, terbutaline
|
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Metaproteronol
|
Selective beta2 agonist
MAST – metaproteronol, albuterol, salmeterol, terbutaline |
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Albuterol
|
Selective beta2 agonist
MAST – metaproteronol, albuterol, salmeterol, terbutaline |
|
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Salmeterol
|
Selective beta2 agonist
MAST – metaproteronol, albuterol, salmeterol, terbutaline |
|
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Terbutaline
|
Selective beta2 agonist
MAST – metaproteronol, albuterol, salmeterol, terbutaline |
|
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Alpha blockers – nonselective
|
Phenoxybenzamine, phentolamine
|
|
|
Phenoxybenzamine
Reversible/irreversible? |
Nonselective alpha blocker – irreversible (vs. phentolamine)
|
|
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Phentolamine
Reversible/irreversible? |
Nonselective alpha blocker – reversible (vs. phenoxybenzamine)
|
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Alpha1 blockers
|
-azosins
Prazosin, terazosin, doxazosin |
|
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Prazosin
|
Alpha1 blocker
-osins |
|
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Terazosin
|
Alpha1 blocker
-osins |
|
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Doxazosin
|
Alpha1 blocker
-osins |
|
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Beta blockers
|
Acebutolol, betaxolol, Esmolol, Atenolol, Metoprolol, Propranolol, Timolol, Pindolol
|
|
|
Beta1 blockers
|
Start with A-M
Atenolol, Acebutalol (partial agonist) Betaxolol, Esmalol, Metoprolol |
|
|
Nonselective Beta Blockers
|
N-Z
Nadolol, Pindolol, Propranolol, Timolol |
|
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Nonselective alpha/beta blockers
|
Carvedilol, labetalol
|
|
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Acebutalol
|
Beta1 blocker (partial agonist): Beta1 > Beta2
|
|
|
Atenolol
|
Beta1 blockers Beta1 > Beta2
Start with A-M |
|
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Betaxolol
|
Beta1 blockers Beta1 > Beta2
Start with A-M |
|
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Esmolol
|
Beta1 blockers Beta1 > Beta2
Start with A-M |
|
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Metoprolol
|
Beta1 blockers Beta1 > Beta2
Start with A-M |
|
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Nadolol
|
Nonselective Beta Blockers (beta1=beta2)
N-Z |
|
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Pindolol
Selective/Nonselective? Action? |
Nonselective Beta Blockers (beta1=beta2). partial agonist
N-Z |
|
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Propranolol
|
Nonselective Beta Blockers (beta1=beta2)
N-Z |
|
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Timolol
|
Nonselective Beta Blockers (beta1=beta2)
N-Z |
|
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Labetalol
|
Nonselective alpha/beta blocker – alpha1/beta1
|
|
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Carvedilol
|
Nonselective alpha/beta blocker
|
|
|
Partial beta-agonists
|
Partial Agonists = Pindolol, Acebutolol
|
|
|
Ca Channel Blockers
|
Nifedipine, Amlodipine, Verapamil, Diltiazem
|
|
|
Nifedipine, amlodipine
|
Ca Channel Blocker – dihydropyridine
|
|
|
Verapamil
|
Ca Channel Blocker – non-dihydropyridine – affects heart, not really vascular smooth muscle
|
|
|
Diltiazem
|
Ca Channel Blocker – in between dihydropyridine/non
|
|
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Nitroglycerin
|
Vasodilator via NO
|
|
|
Isosorbide dinitrate
|
Vasodilator via NO
|
|
|
Fenoldopam
Use? |
Dopamine D1 receptor agonist used in Malignant HTN Tx
|
|
|
Statins
Mechanism, purpose, eg.s. |
HMG-CoA reductase inhibitors – Lipid lowering agents
Lovastatin, pravastatin, simvastatin, atorvastatin, rosuvastatin |
|
|
Lovastatin
|
HMG-CoA reductase inhibitor – Lipid lowering agents
|
|
|
Pravastatin
|
HMG-CoA reductase inhibitor – Lipid lowering agents
AKA Pravachol |
|
|
Simvastatin
|
HMG-CoA reductase inhibitor – Lipid lowering agents
|
|
|
Atorvastatin
|
HMG-CoA reductase inhibitor – Lipid lowering agents
|
|
|
Rosuvastatin
|
HMG-CoA reductase inhibitor – Lipid lowering agents
|
|
|
Bile Acid Resins
|
Cholestyramine, Colestipol, Colesevelam
|
|
|
Cholestyramine
|
Bile Acid Resin Lipid Lowering Agent
|
|
|
Colestipol
|
Bile Acid Resin Lipid Lowering Agent
|
|
|
Colesevelam
|
Bile Acid Resin Lipid Lowering Agent
|
|
|
Ezetimibe
|
Cholesterol absorption blocker – Lipid lowering agent
|
|
|
Fibrates
e.g.s |
Lipid lowering agents
Gemfibrozil, clofibrate, bezafibrate, fenofibrate |
|
|
Gemfibrozil
|
Fibrate Lipid lowering agent
|
|
|
Clofibrate
|
Fibrate Lipid lowering agent
|
|
|
Bezafibrate
|
Fibrate Lipid lowering agent
PPAR-alpha agonist |
|
|
Fenofibrate
|
Fibrate Lipid lowering agent
|
|
|
Cardiac Glycoside (name one)
|
Digoxin
|
|
|
Digoxin
|
Cardiac Glycoside
|
|
|
Antiarrhythmics – classes
|
No Bad Boy Keeps Clean
Class I – Na channel blockers Class II – Beta Blockers Class III – K channel blockers Class IV – Ca channel blockers |
|
|
Class I Antiarrhythmic drugs
|
Police Department Questioned - IA
The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Procainamide
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Disopyramide
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Quinidine
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Tocainide
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Lidocaine - 2 uses
|
Amide local anesthetic AND
Class I Antiarrhythmic drugs Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC (also amide local anesthetic) |
|
|
Mexiletine
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Flecainide
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Propafenone
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
|
|
Encainide
|
Class I Antiarrhythmic drugs
Police Department Questioned - IA The Little Man - IB For Pushing Ecstasy – IC Procainamide, Disopyramide, Quinidine – IA Tocainide, Lidocaine, Mexiletine – IB Flecainide Propafenone, Encainide – IC |
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Class II Antiarrhythmics
|
Beta blockers
TAP ME Timolol, Atenolol, Propranolol, Metoprolol, Esmolol |
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Class III Antiarrhythmics
|
K channel blockers
Sotalol, Ibutilide, Amiodarone, Bretylium |
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Sotalol
|
Class III Antiarrhythmic
K channel blocker |
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Ibutilide
|
Class III Antiarrhythmic
K channel blocker |
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Amiodarone
|
Class III Antiarrhythmic
K channel blocker |
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Bretylium
|
Class III Antiarrhythmic
K channel blocker Sotalol, Ibutilide, Amiodarone, Bretylium |
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Class IV Antiarrhythmics
|
Ca channel blockers (non-dihydropyridines)
Verapamil, diltiazem |
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Verapamil
use? |
Class IV Antiarrhythmic
Ca channel blocker (non-dihydropyridine) |
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Diltiazem
|
Class IV Antiarrhythmic
Ca channel blocker (non-dihydropyridine) |
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Desmopressin
|
ADH analog
|
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Lispro
|
Short-acting Insulin
|
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Aspart
|
Short-acting Insulin
|
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Regular Insulin - duration?
|
Short-acting Insulin
|
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NPH
|
Intermediate-acting insulin
|
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Glargine
|
Long-acting insulin
|
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Detemir
|
Long-acting Insulin
|
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Sulfonylureas
|
First generation: Tolbutamide, Chlorpropamide
Second generation: Glyburide, Glimepiride, Glipizide |
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Tolbutamide
|
First generation sulfonylurea – DM drug
|
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Chlorpropamide
|
First generation sulfonylurea – DM drug
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Glyburide
|
Second generation sulfonylurea – DM drug
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Glimepiride
|
Second generation sulfonylurea – DM drug
|
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Glipizide
|
Second generation sulfonylurea – DM drug
|
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Biguanide
|
Metformin
|
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Metformin
|
Biguanide – DM drug
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Glitazones (aka thiazolidinediones, aka TZDs)
|
DM Drug
Pioglitazone, Rosiglitazone |
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Pioglitazone
|
Glitazone (aka thiazolidinedione, aka TZD)
DM Drug |
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Rosiglitazone
|
Glitazone (aka thiazolidinedione, aka TZD)
DM Drug |
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Name a mimetic
What is it? |
Pramlintide – DM drug
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Pramlintide
|
Amylinomimetic – DM drug
Works by mimicking amylin. Blocks inappropriate glucagon release during postprandial hyperglycemic state, but not in response to hypoglycemic states. |
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GLP-1 (an incretin) mimetic
|
Exenatide – DM Drug
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Exenatide
|
GLP-1 (an incretin) mimetic – DM Drug
|
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Sitagliptin
|
Dipeptidyl-Peptidase-4 (DPP-4) inhibitor used for DM
|
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Dipeptidyl-Peptidase-4 (DPP-4) inhibitor
|
Sitagliptin (DM drug)
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Orlistat
|
Obesity drug – pancreatic lipase inhibitor
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Obesity drug – pancreatic lipase inhibitor
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Orlistat
|
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SNRI used for obesity
|
Sibutramine
|
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Propylthiouracil
|
Hyperthyroidism Drug
|
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Methimazole
|
Hyperthyroidism Drug
|
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Hyperthyroidism drugs
|
Propylthiouracil, Methimazole
|
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Levothyroxine, triiodothyronine
|
Hypothyroidism/myxedema drugs
|
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Hypothyroidism/myxedema drugs
|
Levothyroxine, triiodothyronine
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Glucocorticoids
|
Hydrocortisone, prednisone, triamcinolone, dexamethasone, beclomethasone
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Hydrocortisone
|
Glucocorticoid
|
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Prednisone
Bioavailability? |
Glucocorticoid (needs to be converted to prednisolone in liver)
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Triamcinolone
|
Glucocorticoid
|
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Dexamethasone
duration? |
Glucocorticoid (long-acting)
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Beclomethasone
duration? |
Glucocorticoid (long-acting)
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Demeclocycline
Two functions |
ADH antagonist, tetracycline
|
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Name an ADH antagonist that’s in the tetracycline family
|
Demeclocycline
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H2 Blockers
|
Cimetidine, Ranitidine, Famotidine, Nizatidine
Take H2 blockers before you DINE. Table for “2” |
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Cimetidine
|
H2 Blocker
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Ranitidine
|
H2 Blocker
|
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Famotidine
|
H2 Blocker
|
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Nizatidine
|
H2 blocker
|
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Proton pump inhibitors
|
Omeprazole, Lansoprazole
|
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Omeprazole
|
Proton pump inhibitor
|
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Lansoprazole
|
Proton pump inhibitor
|
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Misoprostol
|
Prostaglandin (PGE1) analog
|
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Pirenzepine
|
Muscarinic Antagonist
|
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Infliximab
|
Monoclonal TNF Ab
|
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Monoclonal TNF Ab
|
Infliximab, adalimumab, etanercept
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Adalimumab
|
Monoclonal TNF Ab used in autoimmune disorders
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Etanercept
|
Monoclonal TNF Ab
|
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Sulfasalazine
|
(5-aminosalycilic acid) – COX blocker
|
|
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Ondansetron
|
5-HT3 antagonist antiemetic
|
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Granisetron
|
5-HT3 antagonist
|
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5-HT3 antagonists
|
Ondansetron, Granisetron
antiemetics |
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Metoclopramide
|
5HT receptor agonist, D2 receptor antagonist. antiemetic, gastroprokinetic drug used to treat nausea and facilitate gastric emptying in gastric paresis. Also migraine drug
|
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5HT receptor agonist that’s also a D2 receptor antagonist?
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Metoclopramide
antiemetic, promotes gastric emptying, migraine drug |
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Lepirudin
|
Hirudin derivative – anticoagulant
|
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Bivalirudin
|
Hirudin derivative - anticoagulant
|
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Argatrovan
|
Non-hirudin-derived antithrombin
|
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Non-hirudin-derived anti-thrombin
|
Argatrovan
|
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Anti-platelet aggregators (via ADP receptors)
|
Clopidogrel, Ticlopidine
|
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Clopidogrel
|
Anti-platelet aggregator
|
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Ticlopidine
|
Anti-platelet aggregator
|
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GPIIb/IIIa blockers
|
Abciximab, Tirofiban, Eptifibatide
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Abciximab
|
GPIIb/IIIa blocker
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Tirofiban
|
GPIIb/IIIa blocker
|
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Eptifibatide
|
GPIIb/IIIa blocker
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Antineoplastics – Nucleotide synthesis
|
Decrease Thymidine synthesis – MTX, 5-FU
Decrease purine synthesis – 6-MP |
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Antineoplastics – DNA
Cross-link DNA (2) Intercalate DNA (2) TopoII inhibitor (1) |
Cross-link DNA – Alkylating agents, cisplatin
Intercalate DNA – Dactinomycin, Doxorubicin Topo-II inhibition - Etoposide |
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Antineoplastics – Cellular division
|
MT formation inhibition – Vinca alkaloids
MT disassembly – Paclitaxel |
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Cancer Drugs – Cell Cycle – S, G2, M, G1
|
S – Antimetabolites (e.g. MTX, 5-FU, Etoposide)
G2 – Etoposide, Bleomycin M – Vinca alkaloids and taxols |
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5-FU
|
S-phase-specific antimetabolite cancer drug
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6-MP
|
antimetabolite cancer drug
|
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|
Cytarabine (ara-C)
|
DNA polymerase inhibitor – cancer drug
|
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Alkylating agents
|
Cyclophosphamide, ifosfamide
|
|
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Cyclophosphamide
|
Alkylating agent
|
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Ifosfamide
|
Alkylating agent
|
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|
Nitrosureas
|
Carmustine, lomustine, semustine, streptozocin
“Nitros on my Mustang” - -stine endings for most |
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Carmustine
|
Nitrosurea
Carmustine, lomustine, semustine, streptozocin “Nitros on my Mustang” - -stine endings for most |
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Lomustine
|
Nitrosurea
Carmustine, lomustine, semustine, streptozocin “Nitros on my Mustang” - -stine endings for most |
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Semustine
|
Nitrosurea
Carmustine, lomustine, semustine, streptozocin “Nitros on my Mustang” - -stine endings for most |
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Streptozocin
|
Nitrosurea
Carmustine, lomustine, semustine, streptozocin “Nitros on my Mustang.” -stine endings for all but streptozocin |
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SERMs
|
Tamoxifen, Raloxifene, Clomiphene
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Tamoxifen
|
SERM
|
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Raloxifene
|
SERM
|
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Clomiphene
|
SERM
|
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Trastuzumab (Herceptin)
|
Monoclonal Ab against HER-2 (erb-B2), cancer drug
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Imatinib (Gleevac)
|
Cancer drug – tyrosine kinase inhibitor
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Vincristine
use? |
MT polymerization blocker – cancer drug
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Vinblastine
|
MT polymerization blocker – cancer drug
|
|
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MT Polymerization blockers
|
Vincristine, Vinblastine
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Paclitaxel
|
Taxol – prevents MT depolymerization, cancer drug
|
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Taxols - name one
MOA Use |
Include paclitaxel – prevents MT depolymerization. cancer drug
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NSAIDs
|
Ibuprofen, Naproxen, indomethacin, ketorolac
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|
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Ketorolac
|
NSAID
|
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Naproxen
|
NSAID
|
|
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COX-2 inhibitor
|
Celecoxib
|
|
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Celecoxib
|
Cox-2 inhibitor
|
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Bisphosphanates
|
Etidronate, Pamidronate, Alendronate, Risedronate
|
|
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Etidronate
|
Bisphosphanate – all –dronate
Etidronate, Pamidronate, Alendronate, Risedronate |
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Pamidronate
|
Bisphosphanate – all –dronate
Etidronate, Pamidronate, Alendronate, Risedronate |
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Alendronate
|
Bisphosphanate – all –dronate
Etidronate, Pamidronate, Alendronate, Risedronate |
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Risedronate
|
Bisphosphanate – all –dronate
Etidronate, Pamidronate, Alendronate, Risedronate |
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Glaucoma drugs
|
ABCDP
Alpha-agonists – epinephrine, Brimonidine Beta blockers – timolol, betaxolol, carteolol Cholinomimetics – pilocarpine, carbachol, physostigmine, echothiophate Diuretics – acetazolamide, mannitol Prostanglandin – Latanoprost (PGF-2alpha) |
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Mannitol
|
Osmotic diuretic
|
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Opioid analgesics
|
Morphine, fentanyl, codeine, heroin, methadone, meperidine, dextromethorphan
|
|
|
Morphine
|
Opioid analgesic
|
|
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Fentanyl
|
Opioid analgesic
|
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Codeine
|
Opioid analgesic
|
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Heroin
|
Opioid analgesic
|
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Methadone
|
Opioid analgesic
|
|
|
Meperidine
|
Opioid analgesic
|
|
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Dextromethorphan
|
Opioid analgesic
|
|
|
Butorphanol
|
Weak/partial opioid agonist
|
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|
Tramadol
|
Weak opioid agonist. Also SNRI
|
|
|
Phenytoin
|
Anti-epileptic, also considered Class IB antiarrhythmic (along with Tocainide, Lidocaine, Mexiletine)
|
|
|
Barbiturates
|
Phenobarbital, pentobarbital, thiopental, secobarbital
|
|
|
Phenobarbital
|
Barbiturate
|
|
|
Pentobarbital
|
Barbiturate
|
|
|
Thiopental
|
Barbiturate
|
|
|
Secobarbital
|
Barbiturate
|
|
|
Benzodiazepines
|
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them)
|
|
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Diazepam
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Lorazepam
Can you name other examples? |
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Triazolam
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Temazepam
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Oxazepam
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Midazolam
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Chlordiazepoxide
|
Benzodiazepine
Diazepam, lorazepam, triazolam, temazepam, oxazepam, midazolam, chlordiazepoxide (all have “az” in them) |
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Short acting Benzos
(TOM) |
TOM
Triazolam, Oxazepam, Midazolam Highest addictive potential |
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Carbamazepine
(think use, not class) |
Antiepileptic
|
|
|
Lamotrigine
|
Antiepileptic
"Lamictal" |
|
|
Gabapentin (2 uses)
|
Adjuvant Antiepileptic, neuropathy med
|
|
|
Topiramate
|
Antiepileptic
|
|
|
Valproic acid
|
Antiepileptic
|
|
|
Ethosuximide
|
Antiepileptic
|
|
|
Inhaled anesthetics
|
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide
|
|
|
Halothane
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
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Enflurane
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
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Isoflurane
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
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Sevoflurane
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
|
|
Methoxyflurane
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
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Nitrous oxide
|
Inhaled anesthetic
Halothane, Enflurane, Isoflurane, Sevoflurane, Methoxyflurane, Nitrous oxide |
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Name 5 types/eg.s of Intravenous anesthetics
|
Barbiturates, benzodiazepines, arylcyclohexylamines (ketamine), opiates, propofol
|
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Arylcyclohexylamine
|
Ketamine – PCP analog that acts as dissociative anesthetic
|
|
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Ketamine
|
Arylcyclohexylamine - PCP analog that acts as dissociative anesthetic
|
|
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Propofol
|
IV anesthetic
|
|
|
Local anesthetics
|
Esters end in –aine: procaine, cocaine, tetracaine
Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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Lidocaine
|
Local anesthetic - amide (also Class IB antiarrhythmic)
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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Mepivacaine
|
Local anesthetic - amide
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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Bupivacaine
|
Local anesthetic - amide
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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Procaine
Type? |
Local anesthetic - ester
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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Cocaine
|
Local anesthetic - ester
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
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|
Tetracaine
|
Local anesthetic - ester
Esters end in –aine: procaine, cocaine, tetracaine Amides do too, but have two Is in name: lIdocaIne, mepIvacaIne, bupIvacaIne |
|
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Depolarizing Neuromuscular blocking drug
|
Succinylcholine
|
|
|
Nondepolarizing Neuromuscular blocking drugs
All have what root in their name? Name six |
All have “cur” in the name
Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
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|
Succinylcholine
|
Depolarizing Neuromuscular blocking drug
|
|
|
Tubocurarine
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
|
Atracurium
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
|
Mivacurium
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
|
Pancuronium
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
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Vecuronium
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
|
Rocuronium
|
Nondepolarizing Neuromuscular blocking drug
All have “cur” in the name Tubocurarine, atracurium, mivacurium, pancuronium, vecuronium, rocuronium |
|
|
Parkinson’s disease drugs
|
BALSA
Bromocriptine Amantadine Levodopa (with carbidopa) Selegiline (and COMT inhibitors) Antimuscarinics |
|
|
Bromocriptine
What kind of parkinson"s drug is it? |
Parkinson’s disease drug, Pituitary adenoma suppression
Ergot alkaloid, partial dopamine agonist |
|
|
Pramipexole
|
Non-ergot dopamine agonist used in Parkinson’s disease
|
|
|
Ropinirole
|
Non-ergot dopamine agonist used in Parkinson’s disease
|
|
|
Amantadine
name two uses |
Parkinson’s disease drug, antiviral
|
|
|
Levodopa+carbidopa/Tolcapone
|
Parkinson’s disease drug and adjuvant
|
|
|
Selegiline
use and class |
Parkinson’s disease drug
MAO-B inhibitor |
|
|
Antimuscarinics (one use)
|
Parkinson’s disease drug
e.g. atropine, scopolamine |
|
|
MAO-B Inhibitor
|
Selegiline
|
|
|
Sumatriptan
|
5HT agonist
|
|
|
Alzheimer’s drugs
|
Memantine - NMDA Glutamate Receptor blocker
Donepezil "Aricept" - AchE-I Rivastigmine "Exelon" - AchE-I Galantamine - alkaloid |
|
|
Memantine
(opposes effects of?) |
Alzheimer drug – NMDA receptor antagonist (opposes glutamate"s effects)
|
|
|
Antipsychotics (neuroleptics)
|
Haloperidol, Thiothixene , Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine
(Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Haloperidol
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Trifloperazine
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Fluphenazine
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Thioridazine
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Thiothixene
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Chlorpromazine
|
Antipsychotic (neuroleptic)
Haloperidol, Thiothixene, Trifluoperazine, Fluphenazine, Thioridazine, Chlorpromazine (Haloperidol, Thiothixene and a bunch of –azines) |
|
|
Atypical Antipsychotics
|
Pras/z, pines and dones:
Clozapine, Olanzapine, Quetiapine, Risperidone, Ziprasidone, Aripiprazole |
|
|
Clozapine
|
Atypical Antipsychotic
Pras/z, pines and dones: Clozapine, Olanzapine, Risperidone, Aripiprazole, Quetiapine, Ziprasidone |
|
|
Olanzapine
|
Atypical Antipsychotic
Pras/z, pines and dones: Clozapine, Olanzapine, Risperidone, Aripiprazole, Quetiapine, Ziprasidone |
|
|
Risperidone
|
Atypical Antipsychotic
Pras/z, pines and dones: Clozapine, Olanzapine, Risperidone, Aripiprazole, Quetiapine, Ziprasidone |
|
|
Aripiprazole
|
Atypical Antipsychotic
Pras/z, pines and dones: Pines: Quetiapine, Clozapine, Olanzapine Dones: Risperidone, Ziprasidone Praz/Pras: Aripiprazole, Ziprasidone |
|
|
Quetiapine
|
Atypical Antipsychotic
Pras/z, pines and dones: Clozapine, Olanzapine, Risperidone, Aripiprazole, Quetiapine, Ziprasidone |
|
|
Ziprasidone
|
Atypical Antipsychotic
Pras/z, pines and dones: Clozapine, Olanzapine, Risperidone, Aripiprazole, Quetiapine, Ziprasidone |
|
|
TCAs
|
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine
(End in –pin(e), -pramine, -triptyline) |
|
|
Imipramine
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Amitriptyline
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Desipramine
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Nortriptyline
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Chlomipramine
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Doxepin
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
Amoxapine
|
TCA
Imipramine, Amitriptyline, Desipramine, Nortriptyline, Chlomipramine, Doxepin, Amoxapine (End in –pin(e), -pramine, -triptyline) |
|
|
SSRIs
|
Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine
|
|
|
Fluoxetine
|
SSRI
Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine |
|
|
Paroxetine
|
AKA Paxil
SSRI Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine |
|
|
Sertraline
|
SSRI
Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine |
|
|
Citalopram
|
SSRI
Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine |
|
|
Fluvoxemine
Hint: rhymes with? |
SSRI
Fluoxetine, paroxetine, sertraline, citalopram, fluvoxemine |
|
|
Venlafaxine
|
SNRI antidepressant/antianxiety
|
|
|
Nefazodone
|
SNRI
|
|
|
Milnacipran
|
SNRI used for fibromyalgia
|
|
|
SNRIs
|
Venlafaxine, Desvenlafaxine, Duloxetine, nefazodone, sibutramine, milnacipran
|
|
|
Sibutramine
|
SNRI used in weight loss
|
|
|
Duloxetine
|
SNRI
Cymbalta |
|
|
Tetracyclic Antidepressants
|
Mirtazapine, Maprotiline
|
|
|
Mirtazapine
|
Tetracyclic Antidepressant
Mirtazapine, Maprotiline |
|
|
Maprotiline
|
Tetracyclic Antidepressant
Mirtazapine, Maprotiline |
|
|
MAOIs
|
Phenelzine, tranylcypromine
|
|
|
Phenelzine
|
MAOI
|
|
|
Tranylcypromine
|
MAOI
|
|
|
Acetazolamide
|
Carbonic anhydrase inhibitor – diuretic
|
|
|
Furosemide
|
Loop diuretic
Furosemide, Bumetanide, Torasemide |
|
|
Bumetanide
|
Loop diuretic
Furosemide, Torasemide, Bumetanide |
|
|
Torasemide
|
Loop diuretic
Furosemide, Bumetanide, Torasemide |
|
|
Loops (e.g.s)
|
Furosemide, Torasemide, Bumetanide, Ethacrynic Acid
|
|
|
Ethacrynic acid
|
Loop Diuretic
|
|
|
Hydrochlorothiazide
|
Thiazide diuretic
|
|
|
K-sparing diuretics
|
Spironolactone, Triamterine, Amiloride, Eplerenone
|
|
|
Spironolactone
2 uses Name other examples |
K-sparing diuretic (as well as anti-androgen)
Spironolactone, Triamterine, Amiloride, Eplerenone |
|
|
Triamterine
|
K-sparing diuretics
Spironolactone, Triamterine, Amiloride, Eplerenone |
|
|
Amiloride
|
K-sparing diuretics
Spironolactone, Triamterine, Amiloride, Eplerenone |
|
|
Eplerenone
|
K-sparing diuretics
Spironolactone, Triamterine, Amiloride, Eplerenone |
|
|
ACE inhibitors
|
Captopril, Enalapril, Lisinopril
|
|
|
Captopril
|
ACE inhibitor
Captopril, Enalapril, Lisinopril |
|
|
Enalapril
|
ACE inhibitor
Captopril, Enalapril, Lisinopril |
|
|
Lisinopril
|
ACE inhibitor
Captopril, Enalapril, Lisinopril |
|
|
Leuprolide
|
GnRH analog
|
|
|
Clomiphene
|
SERM
|
|
|
Antiandrogens
|
Finasteride, Flutamide, Ketoconazole, Spironolactone
|
|
|
Finasteride
|
Antiandrogen, BPH drug
AKA Proscar, Propecia |
|
|
Flutamide
|
Antiandrogen, prostate carcinoma drug
|
|
|
Ketocanazole
Name two functions |
Antifungal, antiandrogen
|
|
|
cGMP phosphodiesterase inhibitors
|
Sildenafil, Vardenafil, Tadalafil
cGMP phosphodiesterase inhibitors |
|
|
Sildenafil
|
cGMP phosphodiesterase inhibitor
|
|
|
Vardenafil
|
cGMP phosphodiesterase inhibitor
|
|
|
Tadalafil
|
cGMP phosphodiesterase inhibitor
|
|
|
Mifepristone (RU-486)
|
Progestin antagonist
Abortant |
|
|
Dinoprostone
|
PGE2 analog
|
|
|
B2 agonist tocolytics
|
Ritodrine, terbutaline
|
|
|
Ritodrine
|
B2 agonist tocolytic
|
|
|
Terbutaline
|
B2 agonist tocolytic
|
|
|
Aromatase inhibitors
|
Anastrozole, Exemestane
|
|
|
Anastrozole
|
Aromatase inhibitor
|
|
|
Exemestane
|
Aromatase inhibitor
|
|
|
H1-Blockers
|
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine
2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Diphenydramine
|
H1-blocker – 1st generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Dimenhydrinate
|
H1-blocker – 1st generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Chlorpheniramine
|
H1-blocker – 1st generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Hydroxazine
|
Sounds like a typical neuroleptic but isn"t
H1-blocker – 1st generation 1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Loratadine
|
H1-blocker – 2nd generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Fexofenadine
|
H1-blocker – 2nd generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Destoratadine
|
H1-blocker – 2nd generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Ceterizine
|
H1-blocker – 2nd generation
1st generation – Diphenhydramine, Dimenhydrinate, Chlorpheniramine, Hydroxazine 2nd Generation – Loratadine, fexofenadine, Destoratadine, Ceterizine |
|
|
Methylxanthines
|
Theophylline, Aminophylline
(asthma meds) |
|
|
Theophylline
|
Methylxanthine Asthma med
|
|
|
Aminophylline
|
Methylxanthine asthma med
|
|
|
Zileuton
|
Antileukotriene – asthma prophylactic
|
|
|
Leukotriene receptor blockers
|
ZafirLUKast, monteLUKast
|
|
|
Zafirlukast
|
Leukotriene receptor blocker used in asthma - think leuko - ZafirLUKast. Like monteLUKast
|
|
|
Montelukast
|
Leukotriene receptor blocker used in asthma - monteLUKast
|
|
|
Expectorants
|
Guaifenesin, N-acetylcysteine
|
|
|
Guaifenesin
|
Expectorant
|
|
|
Alpha glucosidase inhibitors
|
acarbose, miglitol
|
|
|
Acarbose
|
alpha glucosidase inhibitor
|
|
|
Miglitol
|
alpha glucosidase inhibitor
|
|
|
Tadalafil
|
cGMP phosphodiesterase inhibitor
|
|
|
Zolpidem
Works similarly to? How do they compare? |
GABAa receptor agonist (similar mechanism but different structure from benzos), rapid onset, short term insomnia drug
|
|
|
Epinephrine
|
nonselective sympathomimetic
Low doses selective for Beta1 |
|
|
Norepinephrine
|
Sympathomimetic
alpha1 > alpha2 > Beta1 |
