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13 Cards in this Set
- Front
- Back
Sulfonylureas
|
Glyburide
Glipizide Glimepiride Chlorpropamide (1st gen- not used) |
|
Thiazolidinediones (TZDs)
|
Pioglitazone
|
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Biguanide
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Metformin
|
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Dipeptidyl peptidase (DPP- 4 Inhibitor)
|
Sitagliptin
Saxagliptin Linagliptin |
|
Glucagon-Like Peptide (GLP-1 Agonist)
|
Exenatide
Exenatide ER Liraglutide |
|
Metformin
|
Glucophage, Glucophage XR, Fortamet, Glumetza
|
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Biguanide Class Effect
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BBW: Lactic Acidosis
CI: SCr >1.5mg/dL in males, >1.4 in females or CrCl <60 SE: vitamin B12 deficiency long term Weight neutral and NO hypoglycemia! |
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Chlorpropamide (1st gen- not used)
|
Diabinese
|
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Glipizide
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Glucotrol, Glucotrol XR
|
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Glimepiride
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Amaryl
|
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Glyburide
|
DiaBeta
|
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Sulfonylurea Class Effect
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SE: Hypoglycemia, weight gain
Decrease A1C 1-2% Decreased efficacy after long term use |
|
Sulfonylurea Drug Interactions
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Do not use with meglitinides due to similar MOA (nateglinide)
Avoid with insulin because both can cause hypoglycemia |