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69 Cards in this Set
- Front
- Back
Name 5 features of the ANS
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1. function is to regulate the many body organ systems during times of physiological war and peace
2. Acts below level of consciousness 3. ANS has EFFERENT/motor and AFFERENT/sensory components 4. perriphal and central components 5. interacts with endocrine and immune system |
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Name 3 internal body functions of ANS
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regulates heart
regulates secretory glands like sweating,saliva,gastric, bronchial regulates smooth muscle ---bronchi/blood vessels/GI/urogenital |
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The nervous sysytem includes 2 main category
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CNS
PNS |
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The periphal nervous system has what under it
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autonomic-not voluntary
somatic- is voluntary |
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Under the ANS are what 2 categories and what do they do
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Parasympathetic- rest /digest
Sympathetic- fight or flight |
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parasympathetic NS _________ sympathetic nervous system
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counterbalnces
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Name 7 regulatory functions of PSNS
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1. decreased heartrate
2. increased gas secretions 3. bladder emptying..relax 4. bowel empting...relax 5. focus on near vision 6. constriction of pupil 7. contraction of bronchial smooth muscle |
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Name 7 regulatory functions of SNS
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1. increased heartrate
2. decreased gas secretions 3. bladder tense 4. bowel tense 5. focus on far way vision 6. dilation of pupil 7. relaxation of bronchial smooth muscle |
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what is the structual arrangement of PNS
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pre gang
post gang rest and digest |
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which two sites do drugs act at PNS
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1. Synapse btw pre and post
2. junction btw post and effector cells |
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what are PNS nuerotransmitters
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preganglion fibers- actrlcholine LONG
postganglion fibers- acetlecholine SHORT CHOLINGERIC FIBERS |
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PNS...ACh release can activate 2 receptor
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Muscarnic
Nicotinic activation ACH causes movement of Na into cell and K out of cell |
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Explain the SNS?
structual arrangemment ? sites where drugs act? |
Fight or flight
pre= short post= long adrenal medulla(at top of kidneys) synapse btw pre post junction btw post and effector cells adrenal medulla releases NT that acts on the effector organs |
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what are the nuerotransmitters for the SNS?
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pre= acetlcholine
post= norephnephrine adrenal medulla= erpinephrine and norepinephrine ALSO CALLED ADRENERGIC FIBERS |
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WHAT IS THE EXCEPTION WITH SWEAT GLANDS IN THE SNS
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THEY USE ACH
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NAME THE MAJOR ADRENERGIC RECEPTORS
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a receptors(1,2)
b receptors (1,2) dopamine |
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PNS IS THE SAME AS_______ AND SNS IS THE SAME AS _________. NICOTINE/MUSCARINIC ARE______ AND ALPHA/BETA/DOPHAMINE ARE ______
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CHOLERGINIC
ADRENERGIC PNS/CHOLERGIN SNS/SYMPATHETIC |
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WHAT IS AN AGONISTS
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A DRUG THAT BINDS AND CHANGES ACTIVITY OF A RECEPTOR
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WHAT IS AN ANTAGONISTS
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A DRUG THAT DOES NOT PROVOKE A BIOLOGICAL RESPONSE ITSELF UPON BINDING TO A RECEPTOR, RATHER BLOCKS AGONIST MEDIATED REPSONSES
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SNS ADRENERGIC AGONISTS, WHAT R THE 3 TYPES
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INOTROPHIC-INCREASE FORCE OF CONTRACTION IN THE HEART
CHRONOTROPIC- INCREASE HEARTRATE DROMOTROPHIC- INCREASE ELECTRICAL CONDUCTION THRU AV NODE |
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WHAT R 3 TYPES OF ALPHA AND BETA AGONISTS? BETA AGONISTS?
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DOPAMINE
EPINEPHRINE NOREPHNIPHRINE DOBUTAMINE ISOPROTONOL |
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WHAT ARE THE INDICATIONS OF ADRENICGIC AGONISTS?
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RESPIRATORY, OPATHALMIC, CARDIOVASCULAR
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WHEN WOULD U NOT WANT TO GIVE ANADRENGIC AGONIST?
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DRUG ALLERGY
HYPERTENSION |
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I JUST TOOK A PILL THAT WORKS ON THE ALPHA RECEPTORS AND IS AN ADRENERGIC AGONISTS WHAT WOULD BE THE ADVERSE SIDE EFFECTS
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HA,RESTLESSNESS,INSOMNIA,HTN, TACHY,DRY MOUTH,LOSS OF APPETITTE
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WHAT ARE THE ADVERSER SIDE EFFECTS OF BETA AGONISTS
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MILD TREMORS,HA,NERVOUS,DIZZY,INCREASED HEART RATE
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A ADRENGINIC DRUG DOES WHAT
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STIMULATES THE SNS
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ANOTHER NAME FOR SNS ADRENGIC DRUG IS
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SYMPOPTHOMIMETICS
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ADREGENIC DRUGS MIMIC THE SNS NUEROTRANMITTERS WHICH ARE WHAT
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NE
EPI DOPAMINE |
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WHERE ARE ADRENCGIC RECEPTORS?
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ALL THRU BODY
THE RECEPTORS FOR THE SYMPATHETIC NEUROTRANSMITTERS= ALPHA,BETA,DOPAMINERGINICS(ONLY RESPOND TO DOPAMINE) |
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HOW ARE A1 AND A2 DIFFERENTATED
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BY LOCATION ON THE NERVES
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ON POST SYNAPTIC EFFECTOR CELLS
CELL/MUSCLE/ORGAN THAT CELLS STIMULATES |
WHERE ARE A1 RECEPTORS AT
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WHERE ARE A2 RECEPTORS AT
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ON PRESYNAPTIC NERVE TERMINAL , NERVE THAT STIMULATES EFFECTOR CELL
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_____ ______ CONTOL THE RELEASE OF NUUROTRANSMITTER
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A2 ADRENERGIC RECEPTORS
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NAME THE 2 PREDOMINANT RESPONSES OF ADRENERGIC AGONIST
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VASOCONSCRITON(INCREASED BLOOD FLOW)
CNS STIMULATION |
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WHERE ARE BETA ADRENERGIC RECEPTORS AT
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POSTSYNAPTIC CELLS
B1- HEART B2-SMOOTH MUSCLE OF BRONCHIOLES,ARTERIOLES,VISCERAL ORGANS |
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WHAT WOULD BE THE RESPONSE IF I GAVE U BETA ADREN AGONIST
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RELAXED BRONCHIALS,GI,UTERINE,GLYCOGNOLYSIS= BREAKS DOWN SUGAR QUICKER WHICH ALLOWS U HAVE MORE ENERGY TO RUN
CARDIAC STIMULATION |
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DOPANMINERGIC RECEPTORS
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- AN EXTRA ADREN RECEPTO
- STIMULA BY DOPAMINE - CAUSES DILATION OF FOLLOWING VESSELS RENAL,MESNTRIC , CORONARY,CERREBRAL |
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what is a catecholamine
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substance that can make a sympathiticmimetic response
endogenous(body make)e,n,dop synthetic- dobutamine phenylephrine |
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what is a direct sympathomimetic
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binds directly to receptor and causes a physiologic response
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explain a indirect acting sympathmimetic
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causes a release of catecolamine from the vesicles, then binds to receptors and causes physiolic response
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i just gave joe a drug and is working on the alpha adrenergic receptor what are the effects
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-vasoconstriction of blood vessels=high BP
- RELAX OF GI - CONTRACTION OF UTERUS /BLADDER - MALE EJACULATION - DECREASED INSULIN RELEASED - DILATION OF PUPILS |
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I AM TAKING A DRUG THAT IS ACTING ON THE B1 ADRENGENC RECEPTORS ON MYOCARDIUM,AV,SA NODES= CARDIAC STIMULATION
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INCREASED HEART RATE,FORCE OF CONTRACTION,CONDUCTION THRU AV NODE
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B2 HAS WHAT SIDE EFFECTS
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BRONCHODILATION, UTERINE RELAXATION,GLYCOGGENOLYSIS IN LIVER, INCREASED RENIN(RAISES BP??)
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I HAVE ASTHMA, WHAT WOULD U GIVE AND WHERE WOULD IT ACT AT
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BRONCHODILATOR
B2 ADREN RECEPTORS OF BRONCHIAL SMOOTH MUSCLE WHICH WOULD CAUSE RELAXATION SO MORE AIR CAN GET THRU |
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EXPLAIN VASOCONSTRICITON
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FLOW OF BLOOD IS SLOWED=HIGHER BP AND INCREASED VASCULAR RESISTENCE
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VASODILATION
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VESSEL IS WIDENED AND BLOOD FLOW IS INCREASED, LOWER BLOOD PRESSURE, DECREASE IN VASCULAR RESISTENCE
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TERBUTILINE IS WHAT
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B2 ADRENERGIC,SNS,CAUSES RELAXATION OF UTERINE SMOOTH MUSCLE , STOPS PRETERM LABOR
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I HAVE OPEN GLAUCOMA WHAT WOULD U GIVE AND WHRE WOULD IT ACT
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A OR B2 RECEPTORS, CAUSES PUPIL DILATION, EX: EPINEPHRINE
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I HAVE CONJUCTIVE CONGESTION WHAT WOULD U GIVE ME
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WORK ON A-ADRENGERIC RECEPTORS, DECREASE SECRETIONS
EX: EPINEPHRINE, TETRHYROZOLINE(VISINE) |
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EX OF NASAL DECONGESTANT
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EPHEDRINE
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VASOACTIVE SYMPATHOMIMETICS ALSO CALLED_____ ________. ALSO A PRESSOR/INOTROPE. WHAT IS THIS USED TO SUPPORT THE HEART IN?
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CARDIOSELECTIVE SYMPATHOMIMETICS
SHOCK OR CARDIAC FAILURE A AND B RECEPTORS |
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WHAT WOULD INTERACT WITH SNS ADRENERIC DRUGS
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ANESTHESTICS, TRICYL ANTIDEPRESS, MAOIS, ANTIHISTMINES, THYROID PREPARATIONS, ANTIHYPERTENSIVES,
THESE WILL DIRECTLY ANTAGONIZE ANOTHER ADRENGIC DRUG RESULTING IN REDUCED EFFECT |
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WHEN GIVING ADRENNIC DRUGS WHAT WILL U ASSESS
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HYPERTENSION, CARDIAC,RENAL,LIVER,CARDIAC TREATMENT
GET BASELINE VITALS,PERIPHAL PULSES, SKIN COLOR, TEMP, CAP REFILL,POSTURAL BP, |
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WHEN GIVING A ADRENCIC AGONIST IV MAKE SURE TO
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USE PUMP, INFUSE SLOWLY TO AVOID DANGER HEART PROBLEMS, MOITOR CARDIAC RYTHM
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WHEN GIVING ADRENGIC AGOANIST AND THEY HAVE CHRONIC LUNG DISEASE MAKE SURE TO
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TELL CLIENT TO AVOID THINGS THAT EXACERBTE SYMPTOMS
ENCOURAGE FLUID INTAKE EDUCATE ABOUT PROPER DOSING |
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WARNING ABOUT ADRENERGIC DRUGS
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GIVING 2 TOGETHER MAY BRING ON SEVERE CARDIO EFFECTS LIKE TACHY AND HYTENSION
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WHAT ARE THERPUETIC EFFECTS ON THE HEART WHEN GIVING ADRENGERIC AGONISTS
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INCREASED LOC,IMPROVED SKIN COLOR AND TEMP,NORMAL VITALS,INCR OUTPUT, DECREASED EDEMA
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i have asthma what are the therpuetic effects of adrenagonists
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normal rr, few crackles, increasd air exchange, improved blood gases, incre activity tolerance
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what does aadrengeric blocker do ?
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bind to adrenergic receptors but BLOCK STIMULATION OF THE SNS
THERE ARE ALPHA AND BETA BLOCKERS |
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ADRENERGIC BLOCKERS HAVE THE ______ ______ OF ADRENERGIC DRUGS
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OPPOSITE EFFECT
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NAME 3 SYNONYMS 4 ADREN BLOCKERS
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- ADREN ANTAGONISTS
- SYMPATHOLYTICS - A,B,AB BLOCKERS |
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ERGOT ALKOIDS A BLOCKERS
Alpha blocking |
- CONSTRICT DILATED ARTERIOLES IN THE BRAIN
- USED TO TREAT VASCULAR HA - STIMULATES UTERINE CONTRACTIONS AND INDUCE LOCAL VASOCONSTRICTION - CONTROLS POSTPARTUM BLEEDING |
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PRAZOSIN, MINIPRESS
Alpha blocking |
USED FOR HYPERTENSION, URINARY OBSTRUCTION IN MEN WITH BPH, DILATES VESSELS, ORAL, WATCH ORTHOSTATIC HPTENSION
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REGITINE PHENTOLAMINE
Alpha blocking |
REDUCES PERIPHAL VASCULAR RESISTANCE , TREAT HYPTENSION,
ACUTE PROLONGED HYPOTENSION IS ADVERSE EFECT |
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ERGOSTAT
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VASOCONSTRICTION OF DILATED BLOOD VESSELS BY ALPHA RECEPTORS
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ATENOLOL-TENORMIN
Beta blocking |
B BLOCKER, DECREASES BP BY LOWERING, BRADY, ERECTLYE DSYFUNCTION,PREVENTS MI,TREAT ANGINA
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METOPROLOL
Beta blocking |
HYPERTENSION , LATE EARLY MI, CARDIAC FAILURE, ACT- SLOWS SA NODE
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PROPRANOLOL
Beta blocking |
DECREASES BP AND HEART RATE, CAN PASS BLOOD BRAIN BARRIER, DONT GIVE WITH BRONCHIAL ASTHMA, CAN CAUSE MENTAL DEPRESSION
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ESMOLOL B BLOCKER
Beta blocking |
TREAT HPT, BEST ROUTE IV, NON ALCOHOL INTOLERANCE
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