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69 Cards in this Set

  • Front
  • Back
Name 5 features of the ANS
1. function is to regulate the many body organ systems during times of physiological war and peace
2. Acts below level of consciousness
3. ANS has EFFERENT/motor and AFFERENT/sensory components
4. perriphal and central components
5. interacts with endocrine and immune system
Name 3 internal body functions of ANS
regulates heart
regulates secretory glands like sweating,saliva,gastric, bronchial
regulates smooth muscle ---bronchi/blood vessels/GI/urogenital
The nervous sysytem includes 2 main category
CNS
PNS
The periphal nervous system has what under it
autonomic-not voluntary
somatic- is voluntary
Under the ANS are what 2 categories and what do they do
Parasympathetic- rest /digest
Sympathetic- fight or flight
parasympathetic NS _________ sympathetic nervous system
counterbalnces
Name 7 regulatory functions of PSNS
1. decreased heartrate
2. increased gas secretions
3. bladder emptying..relax
4. bowel empting...relax
5. focus on near vision
6. constriction of pupil
7. contraction of bronchial smooth muscle
Name 7 regulatory functions of SNS
1. increased heartrate
2. decreased gas secretions
3. bladder tense
4. bowel tense
5. focus on far way vision
6. dilation of pupil
7. relaxation of bronchial smooth muscle
what is the structual arrangement of PNS
pre gang
post gang
rest and digest
which two sites do drugs act at PNS
1. Synapse btw pre and post
2. junction btw post and effector cells
what are PNS nuerotransmitters
preganglion fibers- actrlcholine LONG
postganglion fibers- acetlecholine SHORT
CHOLINGERIC FIBERS
PNS...ACh release can activate 2 receptor
Muscarnic
Nicotinic
activation ACH causes movement of Na into cell and K out of cell
Explain the SNS?
structual arrangemment ?
sites where drugs act?
Fight or flight
pre= short post= long adrenal medulla(at top of kidneys)
synapse btw pre post
junction btw post and effector cells
adrenal medulla releases NT that acts on the effector organs
what are the nuerotransmitters for the SNS?
pre= acetlcholine
post= norephnephrine
adrenal medulla= erpinephrine and norepinephrine
ALSO CALLED ADRENERGIC FIBERS
WHAT IS THE EXCEPTION WITH SWEAT GLANDS IN THE SNS
THEY USE ACH
NAME THE MAJOR ADRENERGIC RECEPTORS
a receptors(1,2)
b receptors (1,2)
dopamine
PNS IS THE SAME AS_______ AND SNS IS THE SAME AS _________. NICOTINE/MUSCARINIC ARE______ AND ALPHA/BETA/DOPHAMINE ARE ______
CHOLERGINIC
ADRENERGIC
PNS/CHOLERGIN
SNS/SYMPATHETIC
WHAT IS AN AGONISTS
A DRUG THAT BINDS AND CHANGES ACTIVITY OF A RECEPTOR
WHAT IS AN ANTAGONISTS
A DRUG THAT DOES NOT PROVOKE A BIOLOGICAL RESPONSE ITSELF UPON BINDING TO A RECEPTOR, RATHER BLOCKS AGONIST MEDIATED REPSONSES
SNS ADRENERGIC AGONISTS, WHAT R THE 3 TYPES
INOTROPHIC-INCREASE FORCE OF CONTRACTION IN THE HEART
CHRONOTROPIC- INCREASE HEARTRATE
DROMOTROPHIC- INCREASE ELECTRICAL CONDUCTION THRU AV NODE
WHAT R 3 TYPES OF ALPHA AND BETA AGONISTS? BETA AGONISTS?
DOPAMINE
EPINEPHRINE
NOREPHNIPHRINE

DOBUTAMINE
ISOPROTONOL
WHAT ARE THE INDICATIONS OF ADRENICGIC AGONISTS?
RESPIRATORY, OPATHALMIC, CARDIOVASCULAR
WHEN WOULD U NOT WANT TO GIVE ANADRENGIC AGONIST?
DRUG ALLERGY
HYPERTENSION
I JUST TOOK A PILL THAT WORKS ON THE ALPHA RECEPTORS AND IS AN ADRENERGIC AGONISTS WHAT WOULD BE THE ADVERSE SIDE EFFECTS
HA,RESTLESSNESS,INSOMNIA,HTN, TACHY,DRY MOUTH,LOSS OF APPETITTE
WHAT ARE THE ADVERSER SIDE EFFECTS OF BETA AGONISTS
MILD TREMORS,HA,NERVOUS,DIZZY,INCREASED HEART RATE
A ADRENGINIC DRUG DOES WHAT
STIMULATES THE SNS
ANOTHER NAME FOR SNS ADRENGIC DRUG IS
SYMPOPTHOMIMETICS
ADREGENIC DRUGS MIMIC THE SNS NUEROTRANMITTERS WHICH ARE WHAT
NE
EPI
DOPAMINE
WHERE ARE ADRENCGIC RECEPTORS?
ALL THRU BODY
THE RECEPTORS FOR THE SYMPATHETIC NEUROTRANSMITTERS= ALPHA,BETA,DOPAMINERGINICS(ONLY RESPOND TO DOPAMINE)
HOW ARE A1 AND A2 DIFFERENTATED
BY LOCATION ON THE NERVES
ON POST SYNAPTIC EFFECTOR CELLS
CELL/MUSCLE/ORGAN THAT CELLS STIMULATES
WHERE ARE A1 RECEPTORS AT
WHERE ARE A2 RECEPTORS AT
ON PRESYNAPTIC NERVE TERMINAL , NERVE THAT STIMULATES EFFECTOR CELL
_____ ______ CONTOL THE RELEASE OF NUUROTRANSMITTER
A2 ADRENERGIC RECEPTORS
NAME THE 2 PREDOMINANT RESPONSES OF ADRENERGIC AGONIST
VASOCONSCRITON(INCREASED BLOOD FLOW)
CNS STIMULATION
WHERE ARE BETA ADRENERGIC RECEPTORS AT
POSTSYNAPTIC CELLS
B1- HEART
B2-SMOOTH MUSCLE OF BRONCHIOLES,ARTERIOLES,VISCERAL ORGANS
WHAT WOULD BE THE RESPONSE IF I GAVE U BETA ADREN AGONIST
RELAXED BRONCHIALS,GI,UTERINE,GLYCOGNOLYSIS= BREAKS DOWN SUGAR QUICKER WHICH ALLOWS U HAVE MORE ENERGY TO RUN
CARDIAC STIMULATION
DOPANMINERGIC RECEPTORS
- AN EXTRA ADREN RECEPTO
- STIMULA BY DOPAMINE
- CAUSES DILATION OF FOLLOWING VESSELS
RENAL,MESNTRIC , CORONARY,CERREBRAL
what is a catecholamine
substance that can make a sympathiticmimetic response
endogenous(body make)e,n,dop
synthetic- dobutamine phenylephrine
what is a direct sympathomimetic
binds directly to receptor and causes a physiologic response
explain a indirect acting sympathmimetic
causes a release of catecolamine from the vesicles, then binds to receptors and causes physiolic response
i just gave joe a drug and is working on the alpha adrenergic receptor what are the effects
-vasoconstriction of blood vessels=high BP
- RELAX OF GI
- CONTRACTION OF UTERUS /BLADDER
- MALE EJACULATION
- DECREASED INSULIN RELEASED
- DILATION OF PUPILS
I AM TAKING A DRUG THAT IS ACTING ON THE B1 ADRENGENC RECEPTORS ON MYOCARDIUM,AV,SA NODES= CARDIAC STIMULATION
INCREASED HEART RATE,FORCE OF CONTRACTION,CONDUCTION THRU AV NODE
B2 HAS WHAT SIDE EFFECTS
BRONCHODILATION, UTERINE RELAXATION,GLYCOGGENOLYSIS IN LIVER, INCREASED RENIN(RAISES BP??)
I HAVE ASTHMA, WHAT WOULD U GIVE AND WHERE WOULD IT ACT AT
BRONCHODILATOR
B2 ADREN RECEPTORS OF BRONCHIAL SMOOTH MUSCLE
WHICH WOULD CAUSE RELAXATION SO MORE AIR CAN GET THRU
EXPLAIN VASOCONSTRICITON
FLOW OF BLOOD IS SLOWED=HIGHER BP AND INCREASED VASCULAR RESISTENCE
VASODILATION
VESSEL IS WIDENED AND BLOOD FLOW IS INCREASED, LOWER BLOOD PRESSURE, DECREASE IN VASCULAR RESISTENCE
TERBUTILINE IS WHAT
B2 ADRENERGIC,SNS,CAUSES RELAXATION OF UTERINE SMOOTH MUSCLE , STOPS PRETERM LABOR
I HAVE OPEN GLAUCOMA WHAT WOULD U GIVE AND WHRE WOULD IT ACT
A OR B2 RECEPTORS, CAUSES PUPIL DILATION, EX: EPINEPHRINE
I HAVE CONJUCTIVE CONGESTION WHAT WOULD U GIVE ME
WORK ON A-ADRENGERIC RECEPTORS, DECREASE SECRETIONS
EX: EPINEPHRINE, TETRHYROZOLINE(VISINE)
EX OF NASAL DECONGESTANT
EPHEDRINE
VASOACTIVE SYMPATHOMIMETICS ALSO CALLED_____ ________. ALSO A PRESSOR/INOTROPE. WHAT IS THIS USED TO SUPPORT THE HEART IN?
CARDIOSELECTIVE SYMPATHOMIMETICS
SHOCK OR CARDIAC FAILURE
A AND B RECEPTORS
WHAT WOULD INTERACT WITH SNS ADRENERIC DRUGS
ANESTHESTICS, TRICYL ANTIDEPRESS, MAOIS, ANTIHISTMINES, THYROID PREPARATIONS, ANTIHYPERTENSIVES,
THESE WILL DIRECTLY ANTAGONIZE ANOTHER ADRENGIC DRUG RESULTING IN REDUCED EFFECT
WHEN GIVING ADRENNIC DRUGS WHAT WILL U ASSESS
HYPERTENSION, CARDIAC,RENAL,LIVER,CARDIAC TREATMENT
GET BASELINE VITALS,PERIPHAL PULSES, SKIN COLOR, TEMP, CAP REFILL,POSTURAL BP,
WHEN GIVING A ADRENCIC AGONIST IV MAKE SURE TO
USE PUMP, INFUSE SLOWLY TO AVOID DANGER HEART PROBLEMS, MOITOR CARDIAC RYTHM
WHEN GIVING ADRENGIC AGOANIST AND THEY HAVE CHRONIC LUNG DISEASE MAKE SURE TO
TELL CLIENT TO AVOID THINGS THAT EXACERBTE SYMPTOMS
ENCOURAGE FLUID INTAKE
EDUCATE ABOUT PROPER DOSING
WARNING ABOUT ADRENERGIC DRUGS
GIVING 2 TOGETHER MAY BRING ON SEVERE CARDIO EFFECTS LIKE TACHY AND HYTENSION
WHAT ARE THERPUETIC EFFECTS ON THE HEART WHEN GIVING ADRENGERIC AGONISTS
INCREASED LOC,IMPROVED SKIN COLOR AND TEMP,NORMAL VITALS,INCR OUTPUT, DECREASED EDEMA
i have asthma what are the therpuetic effects of adrenagonists
normal rr, few crackles, increasd air exchange, improved blood gases, incre activity tolerance
what does aadrengeric blocker do ?
bind to adrenergic receptors but BLOCK STIMULATION OF THE SNS
THERE ARE ALPHA AND BETA BLOCKERS
ADRENERGIC BLOCKERS HAVE THE ______ ______ OF ADRENERGIC DRUGS
OPPOSITE EFFECT
NAME 3 SYNONYMS 4 ADREN BLOCKERS
- ADREN ANTAGONISTS
- SYMPATHOLYTICS
- A,B,AB BLOCKERS
ERGOT ALKOIDS A BLOCKERS
Alpha blocking
- CONSTRICT DILATED ARTERIOLES IN THE BRAIN
- USED TO TREAT VASCULAR HA
- STIMULATES UTERINE CONTRACTIONS AND INDUCE LOCAL VASOCONSTRICTION
- CONTROLS POSTPARTUM BLEEDING
PRAZOSIN, MINIPRESS
Alpha blocking
USED FOR HYPERTENSION, URINARY OBSTRUCTION IN MEN WITH BPH, DILATES VESSELS, ORAL, WATCH ORTHOSTATIC HPTENSION
REGITINE PHENTOLAMINE
Alpha blocking
REDUCES PERIPHAL VASCULAR RESISTANCE , TREAT HYPTENSION,
ACUTE PROLONGED HYPOTENSION IS ADVERSE EFECT
ERGOSTAT
VASOCONSTRICTION OF DILATED BLOOD VESSELS BY ALPHA RECEPTORS
ATENOLOL-TENORMIN
Beta blocking
B BLOCKER, DECREASES BP BY LOWERING, BRADY, ERECTLYE DSYFUNCTION,PREVENTS MI,TREAT ANGINA
METOPROLOL
Beta blocking
HYPERTENSION , LATE EARLY MI, CARDIAC FAILURE, ACT- SLOWS SA NODE
PROPRANOLOL
Beta blocking
DECREASES BP AND HEART RATE, CAN PASS BLOOD BRAIN BARRIER, DONT GIVE WITH BRONCHIAL ASTHMA, CAN CAUSE MENTAL DEPRESSION
ESMOLOL B BLOCKER
Beta blocking
TREAT HPT, BEST ROUTE IV, NON ALCOHOL INTOLERANCE