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75 Cards in this Set
- Front
- Back
physostigmine
|
CLASS: indirect acting cholinomimetric (parasympathomimetic)
MOA: reversible AChE inhibitor USE: glaucoma; reduce IOP, short acting |
|
neostigmine
|
CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: increase urinary tension & decrease GI motility |
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edrophonium
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CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: distinguish between myasthenic & cholinergic crisis |
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ambenonium
|
CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: management of myasthenia gravis |
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pilocarpine
|
CLASS: direct acting cholinomimetric
MOA: muscarinic agonist USE: glaucoma, short acting |
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carbachol
|
CLASS: direct acting cholinomimetric
MOA: muscarinic agonist USE: glaucoma, short acting |
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ecothiophate
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: glaucoma long acting |
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isoflurophate
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: glaucoma long acting |
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parathion
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: insecticide |
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malathion
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: insecticide |
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sarin
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: nerve gas |
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soman
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: nerve gas |
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tabun
|
CLASS: indirect acting cholinomimetric
MOA: irreversible AChE inhibitor USE: nerve gas |
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bethanecol
|
CLASS: direct acting cholionomimetric
MOA: muscarinic agonist USE: increase urinary tension, decrease GI motility, symptoms xerostoma |
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cevimeline
|
CLASS: direct acting cholinomimetric
MOA: muscarinic agonist USE: increase urinary tension, decrease GI motility, symptoms of xerostoma |
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tacrine
|
CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: dementia |
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donepezil
|
CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: dementia |
|
rivastigmine
|
CLASS: indirect acting cholinomimetric
MOA: reversible AChE inhibitor USE: dementia |
|
galantamine
|
CLASS: indirect acting cholino
MOA: reversible AChE inhibitor USE: dementia |
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atropine
|
CLASS: para-sympathetic Belladona Alkaloid
MOA: muscarinic antagonist USE: antidote; nerve gas, poisonous mushrooms |
|
scopolamine (Transderm Scop)
|
CLASS: parasympatholitic Belladonna Alkaloid
MOA: muscarinic antagonist USE: motion sickness, inhibits vestibular stimulation in inner ear |
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tropicaine (Mydriacyl)
|
CLASS: parasympatholytic
MOA: muscarinic antagonist USE: eye exams, possibly for early detection of dementia |
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homatropine (Isopto Homatropine)
|
CLASS: parasympatholitic
MOA: muscarinic antagonist USE: eye exams |
|
ipratropium bromide (Atrovent)
|
CLASS: parasympatholitic
MOA: muscarinic antagonist USE: COPD, bronchodilator |
|
tiotropium bromide (Spiriva)
|
CLASS: parasympatholitic
MOA: M1/M3 selective antagonist USE: COPD |
|
flavoxate HCl (Urispas)
|
CLASS: parasympatholitic
MOA: muscarinic antagonist USE: antispasmotic for GI/urinary tract |
|
dicyclomine HCl (Bentyl)
|
CLASS: parasympatholitic
MOA: muscarinic antagonist USE: antispasmotic for GI/urinary tract |
|
tolterodine tartrate (Detrol LA)
|
CLASS: parasympatholitic
MOA: muscarinic antagonist USE: antispasmotic for overactive bladder, bladder specific |
|
pirenzepine
|
CLASS: parasympatholitic
MOA: M1/M4 selective antagonist USE: peptic ulcer |
|
telenzepine
|
CLASS: parasympatholitic
MOA: M1 selective USE: peptic ulcer |
|
tripitamine
|
CLASS: parasympatholitic
MOA: M2 selective antagonist USE: block cholinergic bradycardia |
|
darifenacin
|
CLASS: parasympatholitic
MOA: M3 selective antagonist USE: block cholinergic smooth muscle spasms, secretions |
|
biperiden (Akineton)
|
CLASS: parasympatholitic
MOA: muscarinic/nicotinic antagonist USE: blocks Parkinsonism and SE of antipsychotic drugs |
|
dextroamphetamine (Dexedrine)
|
CLASS: indirect acting sympathomimetic
MOA: USE: ADD/ADHD |
|
methylphenidate (Ritalin)
|
CLASS: indirect acting sympathomimetic
MOA: USE: ADD/ADHD |
|
pemoline (Cylert)
|
CLASS: indirect acting sympathomimetic
MOA: USE: ADD/ADHD |
|
epinephrine
|
CLASS: direct acting sympathomimetic
MOA: non-selective agonist USE: allergic rxn, vasoconstriction |
|
isoproterenol (Isuprel)
|
CLASS: direct acting sympathomimetic
MOA: non-selective Beta agonist USE: shock treatment |
|
dobutamine (Dobutrex)
|
CLASS: direct acting sympathomimetic
MOA: Beta agonist USE: shock treatment |
|
phenylephrine (Neosynephrine)
|
CLASS: direct acting sympathomimetic
MOA: alpha-1 selective agonist USE: nasal congestion |
|
apraclonidine (Iopidine)
|
CLASS: direct acting sympathomimetic
MOA: alpha-2 selective agonist USE: lower IOP, glaucoma |
|
mephentermine (Wyamine Sulfate)
|
CLASS: direct acting sympathomimetic
MOA: alpha-1 selective agonist USE: anti-hypotension |
|
metaraminol (Aramine)
|
CLASS: direct acting sympathomimetic
MOA: alpha-1 selective agonist USE: anti-hypotension |
|
methoxamine (Vasoxyl)
|
CLASS: direct acting sympathomimetic
MOA: alpha-1 selective agonist USE: anti-hypotension |
|
clonidine (Catapres)
|
CLASS: direct acting sympathomimetic
MOA: alpha-2 selective agonist (pre-synaptic actions) USE: anti-hypertensive; diarrhea; drug withdrawal; migraine; Tourette's syndrome |
|
metaproterenol (Alupent)
|
CLASS: direct acting sympathomimetic
MOA: beta-2 selective agonist USE: bronchospasms |
|
terbutaline (Brethine)
|
CLASS: direct acting sympathomimetic
MOA: beta-2 selective agonist USE: bronchospasms |
|
albuterol (Proventil, Ventolin)
|
CLASS: direct acting sympathomimetic
MOA: beta-2 selective agonist USE: bronchospasms |
|
ritodrine (Yutopar)
|
CLASS: direct acting sympathomimetic
MOA: beta-2 selective agonist USE: uterine relaxant |
|
BRL 37344
|
CLASS: direct acting sympathomimetic
MOA: beta-3 selective agonist USE: lipolysis |
|
guanadrel (Hylorel)
|
CLASS: indirect acting sympatholytic
MOA: NE release inhibitor USE: anti-hypertension |
|
alpha-methyldopa
|
CLASS: indirect acting sympatholytic
MOA: neurotransmitter synthesis inhibitor USE: inhibits L-aromatic amino acid decarboxylase |
|
carbidopa
|
CLASS: indirect acting sympatholytic
MOA: neurotransmitter synthesis inhibitor USE: inhibits L-aromatic amino acid decarboxylase; combo w/levodopa to treat Parkinson's |
|
alpha-methyltyrosine
|
CLASS: indirect acting sympatholytic
MOA: neurotransmitter synthesis inhibitor USE: inhibits tyrosine hydroxylase; Pheochromocytoma |
|
fusaric acid
|
CLASS: indirect acting sympatholytic
MOA: neurotransmitter synthesis inhibitor USE: inhibits DA beta-hydroxylase |
|
phentolamine (Regitine)
|
CLASS: direct acting sympatholytic
MOA: non-selective alpha-antagonist USE: male sexual dysfunction |
|
prazosin (Minipress)
|
CLASS: direct acting sympatholytic
MOA: alpha-1 selective antagonist USE: anti-hypertensive; BPH |
|
terazosin (Hytrin)
|
CLASS: direct acting sympatholytic
MOA: alpha-1 selective antagonist USE: anti-hypertensive; BPH |
|
tamsulosin HCl (Flomax)
|
CLASS: direct acting sympatholytic
MOA: alpha-1 selective antagonist USE: BPH |
|
doxazosin (Cardura)
|
CLASS: direct acting sympatholytic
MOA: alpha-1 selective antagonist USE: BPH |
|
yohimbine (Yocon)
|
CLASS: direct acting sympatholytic
MOA: alpha-2 selective antagonist USE: male sexual dysfunction |
|
propranolol (Inderal)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: anti-hypertension; panic symptoms |
|
nadolol (Corgard)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: anti-hypertension; panic symptoms |
|
timolol (Blocadren)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: anti-hypertension; panic |
|
pindolol (Visken)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: anti-hypertension; panic |
|
timolol (Timoptic)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: glaucoma |
|
levobunolol (Betagan)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: glaucoma |
|
carteolol (Ocupress)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: glaucoma |
|
metipranolol (Optipranolol)
|
CLASS: direct acting sympatholytic
MOA: non-selective beta antagonist USE: glaucoma |
|
acebutolol (Sectral)
|
CLASS: direct acting sympatholytic
MOA: beta-1 selective antagonist USE: HTN; angina; sinus; tachycardia; atrial fib/flutter |
|
atenolol (Tenormin)
|
CLASS: direct acting sympatholytic
MOA: beta-1 selective antagonist USE: HTN; angina; sinus; tachycardia; atrial fig/flutter |
|
metoprolol tartrate (Lopressor)
|
CLASS: direct acting sympatholytic
MOA: beta-1 selective antagonist USE: HTN; angina; sinus; tachycardia; atrial fig/flutter |
|
esmolol (Brevibloc)
|
CLASS: direct acting sympatholytic
MOA: beta-1 selective antagonist USE: HTN; angina; sinus; tachycardia; atrial fig/flutter |
|
ICI 118551
|
CLASS: direct acting sympatholytic
MOA: beta-2,3 selective antagonist USE: unknown |
|
CGP 20712A
|
CLASS: direct acting sympatholytic
MOA: beta-2,3 selective antagonist USE: unknown |