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75 Cards in this Set

  • Front
  • Back
physostigmine
CLASS: indirect acting cholinomimetric (parasympathomimetic)

MOA: reversible AChE inhibitor

USE: glaucoma; reduce IOP, short acting
neostigmine
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: increase urinary tension & decrease GI motility
edrophonium
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: distinguish between myasthenic & cholinergic crisis
ambenonium
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: management of myasthenia gravis
pilocarpine
CLASS: direct acting cholinomimetric

MOA: muscarinic agonist

USE: glaucoma, short acting
carbachol
CLASS: direct acting cholinomimetric

MOA: muscarinic agonist

USE: glaucoma, short acting
ecothiophate
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: glaucoma long acting
isoflurophate
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: glaucoma long acting
parathion
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: insecticide
malathion
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: insecticide
sarin
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: nerve gas
soman
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: nerve gas
tabun
CLASS: indirect acting cholinomimetric

MOA: irreversible AChE inhibitor

USE: nerve gas
bethanecol
CLASS: direct acting cholionomimetric

MOA: muscarinic agonist

USE: increase urinary tension, decrease GI motility, symptoms xerostoma
cevimeline
CLASS: direct acting cholinomimetric

MOA: muscarinic agonist

USE: increase urinary tension, decrease GI motility, symptoms of xerostoma
tacrine
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: dementia
donepezil
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: dementia
rivastigmine
CLASS: indirect acting cholinomimetric

MOA: reversible AChE inhibitor

USE: dementia
galantamine
CLASS: indirect acting cholino

MOA: reversible AChE inhibitor

USE: dementia
atropine
CLASS: para-sympathetic Belladona Alkaloid

MOA: muscarinic antagonist

USE: antidote; nerve gas, poisonous mushrooms
scopolamine (Transderm Scop)
CLASS: parasympatholitic Belladonna Alkaloid

MOA: muscarinic antagonist

USE: motion sickness, inhibits vestibular stimulation in inner ear
tropicaine (Mydriacyl)
CLASS: parasympatholytic

MOA: muscarinic antagonist

USE: eye exams, possibly for early detection of dementia
homatropine (Isopto Homatropine)
CLASS: parasympatholitic

MOA: muscarinic antagonist

USE: eye exams
ipratropium bromide (Atrovent)
CLASS: parasympatholitic

MOA: muscarinic antagonist

USE: COPD, bronchodilator
tiotropium bromide (Spiriva)
CLASS: parasympatholitic

MOA: M1/M3 selective antagonist

USE: COPD
flavoxate HCl (Urispas)
CLASS: parasympatholitic

MOA: muscarinic antagonist

USE: antispasmotic for GI/urinary tract
dicyclomine HCl (Bentyl)
CLASS: parasympatholitic

MOA: muscarinic antagonist

USE: antispasmotic for GI/urinary tract
tolterodine tartrate (Detrol LA)
CLASS: parasympatholitic

MOA: muscarinic antagonist

USE: antispasmotic for overactive bladder, bladder specific
pirenzepine
CLASS: parasympatholitic

MOA: M1/M4 selective antagonist

USE: peptic ulcer
telenzepine
CLASS: parasympatholitic

MOA: M1 selective

USE: peptic ulcer
tripitamine
CLASS: parasympatholitic

MOA: M2 selective antagonist

USE: block cholinergic bradycardia
darifenacin
CLASS: parasympatholitic

MOA: M3 selective antagonist

USE: block cholinergic smooth muscle spasms, secretions
biperiden (Akineton)
CLASS: parasympatholitic

MOA: muscarinic/nicotinic antagonist

USE: blocks Parkinsonism and SE of antipsychotic drugs
dextroamphetamine (Dexedrine)
CLASS: indirect acting sympathomimetic

MOA:

USE: ADD/ADHD
methylphenidate (Ritalin)
CLASS: indirect acting sympathomimetic

MOA:

USE: ADD/ADHD
pemoline (Cylert)
CLASS: indirect acting sympathomimetic

MOA:

USE: ADD/ADHD
epinephrine
CLASS: direct acting sympathomimetic

MOA: non-selective agonist

USE: allergic rxn, vasoconstriction
isoproterenol (Isuprel)
CLASS: direct acting sympathomimetic

MOA: non-selective Beta agonist

USE: shock treatment
dobutamine (Dobutrex)
CLASS: direct acting sympathomimetic

MOA: Beta agonist

USE: shock treatment
phenylephrine (Neosynephrine)
CLASS: direct acting sympathomimetic

MOA: alpha-1 selective agonist

USE: nasal congestion
apraclonidine (Iopidine)
CLASS: direct acting sympathomimetic

MOA: alpha-2 selective agonist

USE: lower IOP, glaucoma
mephentermine (Wyamine Sulfate)
CLASS: direct acting sympathomimetic

MOA: alpha-1 selective agonist

USE: anti-hypotension
metaraminol (Aramine)
CLASS: direct acting sympathomimetic

MOA: alpha-1 selective agonist

USE: anti-hypotension
methoxamine (Vasoxyl)
CLASS: direct acting sympathomimetic

MOA: alpha-1 selective agonist

USE: anti-hypotension
clonidine (Catapres)
CLASS: direct acting sympathomimetic

MOA: alpha-2 selective agonist (pre-synaptic actions)

USE: anti-hypertensive; diarrhea; drug withdrawal; migraine; Tourette's syndrome
metaproterenol (Alupent)
CLASS: direct acting sympathomimetic

MOA: beta-2 selective agonist

USE: bronchospasms
terbutaline (Brethine)
CLASS: direct acting sympathomimetic

MOA: beta-2 selective agonist

USE: bronchospasms
albuterol (Proventil, Ventolin)
CLASS: direct acting sympathomimetic

MOA: beta-2 selective agonist

USE: bronchospasms
ritodrine (Yutopar)
CLASS: direct acting sympathomimetic

MOA: beta-2 selective agonist

USE: uterine relaxant
BRL 37344
CLASS: direct acting sympathomimetic

MOA: beta-3 selective agonist

USE: lipolysis
guanadrel (Hylorel)
CLASS: indirect acting sympatholytic

MOA: NE release inhibitor

USE: anti-hypertension
alpha-methyldopa
CLASS: indirect acting sympatholytic

MOA: neurotransmitter synthesis inhibitor

USE: inhibits L-aromatic amino acid decarboxylase
carbidopa
CLASS: indirect acting sympatholytic

MOA: neurotransmitter synthesis inhibitor

USE: inhibits L-aromatic amino acid decarboxylase; combo w/levodopa to treat Parkinson's
alpha-methyltyrosine
CLASS: indirect acting sympatholytic

MOA: neurotransmitter synthesis inhibitor

USE: inhibits tyrosine hydroxylase; Pheochromocytoma
fusaric acid
CLASS: indirect acting sympatholytic

MOA: neurotransmitter synthesis inhibitor

USE: inhibits DA beta-hydroxylase
phentolamine (Regitine)
CLASS: direct acting sympatholytic

MOA: non-selective alpha-antagonist

USE: male sexual dysfunction
prazosin (Minipress)
CLASS: direct acting sympatholytic

MOA: alpha-1 selective antagonist

USE: anti-hypertensive; BPH
terazosin (Hytrin)
CLASS: direct acting sympatholytic

MOA: alpha-1 selective antagonist

USE: anti-hypertensive; BPH
tamsulosin HCl (Flomax)
CLASS: direct acting sympatholytic

MOA: alpha-1 selective antagonist

USE: BPH
doxazosin (Cardura)
CLASS: direct acting sympatholytic

MOA: alpha-1 selective antagonist

USE: BPH
yohimbine (Yocon)
CLASS: direct acting sympatholytic

MOA: alpha-2 selective antagonist

USE: male sexual dysfunction
propranolol (Inderal)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: anti-hypertension; panic symptoms
nadolol (Corgard)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: anti-hypertension; panic symptoms
timolol (Blocadren)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: anti-hypertension; panic
pindolol (Visken)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: anti-hypertension; panic
timolol (Timoptic)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: glaucoma
levobunolol (Betagan)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: glaucoma
carteolol (Ocupress)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: glaucoma
metipranolol (Optipranolol)
CLASS: direct acting sympatholytic

MOA: non-selective beta antagonist

USE: glaucoma
acebutolol (Sectral)
CLASS: direct acting sympatholytic

MOA: beta-1 selective antagonist

USE: HTN; angina; sinus; tachycardia; atrial fib/flutter
atenolol (Tenormin)
CLASS: direct acting sympatholytic

MOA: beta-1 selective antagonist

USE: HTN; angina; sinus; tachycardia; atrial fig/flutter
metoprolol tartrate (Lopressor)
CLASS: direct acting sympatholytic

MOA: beta-1 selective antagonist

USE: HTN; angina; sinus; tachycardia; atrial fig/flutter
esmolol (Brevibloc)
CLASS: direct acting sympatholytic

MOA: beta-1 selective antagonist

USE: HTN; angina; sinus; tachycardia; atrial fig/flutter
ICI 118551
CLASS: direct acting sympatholytic

MOA: beta-2,3 selective antagonist

USE: unknown
CGP 20712A
CLASS: direct acting sympatholytic

MOA: beta-2,3 selective antagonist

USE: unknown