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57 Cards in this Set
- Front
- Back
Labetalol
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Nonselective alpha and beta antagonist
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Carvedilol
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Nonselective alpha and beta antagonist
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Phenoxybenzamine
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Nonselective alpha antagonist
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Phentolamine
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Nonselective alpha antagonist
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Prazosin
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Alpha1 antagonist
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Terazosin
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Alpha1 antagonist
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Doxazosin
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Alpha1 antagonist
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Indoramin
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Alpha1 antagonist
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Rauwolscine
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Alpha2 antagonist
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Yohimbine
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Alpha2 antagonist
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Tolazoline
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Alpha2 antagonist
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Propranolol
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Nonselective beta antagonist
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Pindolol
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Nonselective beta antagonist
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Timolol
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Nonselective beta antagonist
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Penbutolol
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Nonselective beta antagonist
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Nadolol
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Nonselective beta antagonist
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Carteolol
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Nonselecive beta antagonist
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Sotalol
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Nonselective beta antagonist
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Acebutolol
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Beta1 antagonist
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Betaxolol
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Beta1 antagonist
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Esmolol
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Beta1 antagonist
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Atenolol
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Beta1 antagonist
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Celiprolol
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Beta1 antagonist
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Metoprolol
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Beta1 antagonist
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Butoxamine
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Beta2 antagonist
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Isoproterenol
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Nonselective beta agonist
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Xamoterol
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Beta1 agonist
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Metaproterenol
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Beta2 agonist
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Fenoterol
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Beta2 agonist
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Terbutaline
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Beta2 agonist
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Salbutamol
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Beta2 agonist
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Ritodrine
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Beta2 agonist
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Salmeterol
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Beta2 agonist
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Formoterol
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Beta2 agonist
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Pirbuterol
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Beta2 agonist
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Bitolterol
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Beta2 agonist
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BRL 37344
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Beta3 agonist
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Oxymetazoline
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Nonselective alpha agonist
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Xylometazoline
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Nonselective alpha agonist
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Tetrahydrozoline
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Nonselective alpha agonist
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Phenylephrine
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Alpha1 agonist
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Metaraminol
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Alpha1 agonist
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Methoxamine
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Alpha1 agonist
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Clonidine
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Alpha2 agonist
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Guanabenz
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Alpha2 agonist
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Guanfacine
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Alpha2 agonist
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Rilmenidine
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Alpha2 agonist
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Moxonidine
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Alpha2 agonist
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Alpha-methyldopa
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Alpha2 agonist
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Propanolol
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Nonselective B1 and B2 blocker
Large first pass effect T 1/2 = 3-5 hr Some CNS effects First used as antiarrhythmic agent |
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Metoprolol
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B1 50-100 > B2
T1/2 = 3-5 hr Fewer side effects Decreases renin release |
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Nadolol
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Nonselective B1 and B2 blocker
Not readily metabolized T1/2 = 14-24 hr Once daily dosing is possible No significant CNS effect |
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Timolol
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Nonselective B1 and B2 blocker
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Pindolol
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Nonselective B1 and B2 blocker with intrinsic sympathomimetic activity (ISA) (partial agonist) Leads to less beta receptor up-regulation and less supersensitivity
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Labetolol
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Nonselective B1 and B2 plus a1 blocker
Beta:alpha block is 3:1 Beta blockade occurs at lower doses Alpha plus beta blockade is good for treatment of pheochromocytoma |
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Carvediolol
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S(-) isomer or racemic mixture exhibits non-selective beta blockade while the R(+) exhibits alpha blockade.
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Bisoprolol
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Selective B1 blocker
B1 selectivity is not absolute so that B2 activity occurs at doses above 20 mg. |