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65 Cards in this Set

  • Front
  • Back
Amitriptyline (Elavil)
Clormipramine (Anafranil)
Desipramine (Norpramine)
Doxepin (Sinequan)
Imapramine (Tofranil)
Maprotiline(Deprilept, Lidiomyl)
Nortriptyline (Aventyl, Pamelor)
Protriptyline (Vivactil)
Trimipramine (Surmontil)
TCA, depression, bipolar, 2nd line drug for OCD
Citalopram (celexa)
Escitalopram (Laxapro)
Fluoxetine (Prozac, Serafem)
Paroxetine (Paxil)
Sertaline (Zoloft)
--oxemine
SSRI, antidepressant, first line drug for OCD, PMD, PTSD (best if started with in 2 weeks of event)
TCA toxicity drug tx
Physostigmine (counteracts anticholinergic actions)
Venlafaxine (Effexor, Effexor XR)
Desvenlafaxine (Pristiq)
Duloxetine (Cymbalta)
S/DRI, major depression, anxiety disorders, fibromyalgia, neuropathic pain
Isocarboxazid (Marplan)
Phenylzine (Nardil)
Tranylecopramine (Parnate)
Selegipine (Emsam)
MAOI, depression, atypical depression, ocd, panic attacks
Welbutrin, Zyban
antidepressants, stimulate, suppresses appetite, inhibits nicotine desire
Diazepam (Valium)
Aprazolam (Xanax)
loprazepam (Ativan)
clonazepam (Klonipin)
Antiolytic- Bensodiazepines
Drug of choice for insomnia and anxiety
Chlordiazepoxide (librium)
for alcohol withdrawal, benzodiazepine
Reveres effects of Benzodiazepines
flumazemil (Romazicon)
Zolpidem (Ambien, Ambien CR)
Zaleplon (Sonata)
Eszopiclone (Lunesta)
Benzo- like
Prolong sleep duration
Ramelteon (Rozerem)
Melatonin Agonists
Triopental
Secobarbital
phenobarbital
Barbiturates
Seizures
Anesthesia
Acute toxicity of Barbiturates
Triad of symptoms
- respiratory depression
- coma
- pinpoint pupils

- often hypotension and hypothermia
Buspirone (Buspar)
Generalized Anxiety disorder
Dextroamphetamine sulfate (Dextrostat, Dexodrine, Dexodrine spanules)
Amphetamine, dextroam phetamine mixture
Adderall
Methamphetamine
Amphetamines
ADHD and Narcolepsy
Methylphenidate (Ritalin, Concerta, Metadate)
Dexmethylphenidate (Focalin)
Amphetamine-like
ADHD
Modafinal (Provigal)
Promote wakfullness
Shiftwork
Narcolepsy
Sleep apnea
Caffeine
Theophylline
Theobromine
Methylxanthines
neonatal apnea
promoting wakfullness
Acute toxicity of methyxanthines
Stimulation of CNS
Tachycardia
Respiratory stimulation
Sensory phenomena
Tamoxifen
- blocks estrogen receptors and inhibit cell growth in the breast
- prevents and treats breast cancer
A/E: hotflashes and increased risk for endometrial cancer and thromboembolism
- protects against osteoporosis and good for LDL and HDL
CRF potassium limit
2-4g/day
CRH protein restriction
.6-.75g/kg/day when creatinine cleatance is less than 25 mL/min
CRF potassium restriction
2-4g/day- see list in med surg book!)
low phosphate diet
dairy, nuts, legumes
Kayexalate
Cation exchange resins
for hyperkalemia
Sevelamar (Renegal, Reneva)
Lowers phosphate
- swallow whole and with meal!
Lanthanium Carbonate (Fosrenal)
lowers phosphate
Oxybutynin (Ditropan, Ditropan XL, Glenique, Oxytrol)
Anticholinergics- preffered for overactive bladder
Antispasmatics
FOR overactive bladder
Darifenacin (Enablex)
Solifenacin (VESIcare)
Overactive bladder
- more M3 receptor selective
Fesoterodine (Toviaz)
Tolterodine (Detrol, Detrol LA)
Muscarinic antagonists
Overactive bladder
Bethanechol (Urecholine)
Urinary retention
Muscarinic agonist (SLUD)
Phenazopyridine (AZO Standard, Pyridium)
UTI pain relief
Sidenafil (Viagra)
ED
Pulmonary hypertension
Verdenafil (Levitra)
ED
60 min for 4 h
Tadalafil (Cialis)
ED
2h for 36h
take daily if sex .2x/wk
hypo and hypertension limits for ED drugs
BP <90/50
BP > 170-110
Finasteride (Proscar)
Propecia
Benign prostate hyperplasia
(propecia used to treat male bladness)
Dutasteride (Avodart)
Benign prostate hyperplasia
** do not touch pill if pregnant!
Terazosin (Hytrin)
Doxazosin (Cardura)
Tamsulosin (Flomax)
Alfuzosin (Uroxatral)
Silodosin (Rapaflo)
Alpha adrenergic antagonists, benign prostate hyperplasia
* contraindicated with ED drugs
Saw palmetto
decreases prostate size
requires 1-2 months
Levodopa (Sinemet, Parcopa)

Carbadopa
- Parkinson's

** low protein diet
Sinemet 25/100 or 50/200 (carbi, levo)
Parkinson's
most effective
casues Neuroleptic malignant syndrome
Parcopa (levo, carbi)
- Parkinson's
- dissolve under tongue
Pramipexole (Mirapex)
Ropinorole (Requip)
Amantadine (Symmetrel)
Parkinson's
- Impulsive behaviors
Apomorphine (Apokyn/Spontane)
exacerbations of parkinson's

give with antiemetic
Entacarpone (Comtan)
Talcarpone (Tasmar)
Parkinson's
COMT inhibitors
- elevated levadopa levels
Stalevo or Stavelo
Levadop, Carbidopa, Entacarpone
Parkinson's
Rasagiline (Azileft)
Seleglinine (Eldepryl, Carbex)
Parkinson's
MAOB
Adminster before noon
2nd or 3rd line drug
Artane
Cogentin
Centrally acting anticholinergic
Parkinson's- restores balance by reducing available AcH
Neostigmine (Prostigmine)
Pyridostigmine (Mestinon)
Reversible Cholinesterase inhibitor
Myasthenia Gravis
- produces SLUD
Avones
Refib
Betaseron
Interferon beta1a and Betaseron is B1b
MS
Glatiramer Acetate (Copaxone)
long term MS therapy
Matalizumab (Tysabril)
MS and Crohn's
- reactivation of JC Virus
Mitoxantrone (Novatrone)
worsening relapsing remitting MS
Cytotoxic agent
Tizantidine (Zanaflex)
Carsoprodol (Soma)
Chlorzoxazone (Paraflex, Parton Forte)
Cyclobenzaprine (Flexiril)
Metaxalone (Skelaxin)
Methocarbmol (Robaxin)
Orphenadrine (Norflex)
flex or axin
centrally acting muscle relaxants
- muscle spasms from MS, low Ca, epilepsy, trauma, pain
Baclofen (Lioresal)
- for spasticity
** no antidote for oversdose
Phenytoin (Dilantin)
Seizures
levels 10-20 mcg/mL
Carbamezepine (Tegretol)
Seizures
levels 4-12 mcg/mL
Valproid acid (Depakene, Depakote, Depacon)
Seizures
bipolar
migraine
levels 40-100 mcg/mL
oxicarbezipine (Trileptal)
Gabapentin (Neurontin)
Zonisamide (Zonegran)
Topiramate (Topamax)
Levitracetam (Keppra)
Pregabalin (Lyrica)
Lamotigrine (Lamictal)
Epilepsy
(partial and generalized tonic clonic seizures)
new drugs
Donepezil (Aricept)
Galantamine (Razadyne)
Rivastigmine (Excelon)
Reversible cholinesterase inhibitors
- mild to moderate alzheimers disease
- prevents AcH breakdown
Memantine (Namenda)
NMDA class, only one in new class
- moderate to severe Alzeimers disease
Egromar
Ergotamine
Cafergot (Wigraine)
manage migrain headache

give with antiemetic
Simatriptan (Imitrex)

---triptan
Serotonin 1B/1D
**to abort ONGOING migraine
Dihydroergotamine (Migranal)
IM choice drug for terminateing migrain eor cluster HA