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109 Cards in this Set

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-azole

Ergosterol synthesis inhibitor

Ketoconazole

-bendazole

Antiparasitic, antihelminitic

Mebendazole

-cillin

Peptidoglycan synthesis inhibitor

Ampicillin

-cycline

Protein synthesis inhibitor

Tetracycline

-ivir

Neuraminidase inhibitor

Osteltamivir

-navir

Protease inhibitor

Ritonavir

-ovir

DNA polymerase inhibitor

Acyclovir

-thromycin

Macrolide abx

Azithromycin

-ane

Inhalation general anaesthetic

Halothane

-azine

Typical antipsychotic

Thioridazine

-barbital

Barbiturate

Phenobarbital

-caine

Local anaesthetic

Lidocaine

-etine

SSRI

Fluoxetine

-ipramine

TCA

Imipramine

-triptan

5-HT 1B/1D agonists

Sumatriptan

-triptyline

TCA

Amitriptyline

-zepam

Benzodiazepine

Diazepam

-zolam

Benzodiazepine

Alprazolam

-chol

Cholinergic agonist

Bethanechol, carbachol

-curium or - curonium

Non-depolarising paralytic

Atracurium, vecuronium

-olol

Beta-blocker

Propranolol

-stigmine

AChE inhibitor

Neostigmine

-terol

Beta2-agonist

Albuterol

-zosin

Alpha1-antagonist

Prazosin

-afil

PDE-5 inhibitor

Sildenafil

-dipine

Dihydropyridine CCB

Amlodipine

-pril

ACE inhibitor

Captopril

-sartan

Angiotensin-2 receptor blocker

Losartan

-statin

HMG-CoA reductase inhibitor

Atorvastatin

-dronate

Bisphosphonate

Aledronate

-glitazone

PPAR-gamma activator

Rosiglitazone

-prazole

PPI

Omeprazole

-prost

Prostaglandin analogue

Latanoprost

-tidine

H2-antagonist

Cimetidine

-tropin

Pituitary hormone

Somatotropin

-ximab

Chimeric monoclonal Ab

Basiliximab

-zumab

Humanised monoclonal Ab

Daclizumab

Sulfa drugs

Probenecid, Furosemide, Acetazolamide, Celecoxib, Thiazides, Sulfonamide abxs, Sulfasalazine, Sulfonylureas

Popular FACTSSS

Sulfa drugs - adverse rxns

Fever, UTI, Steven-Johnson syndrome, hemolytic anemia, thrombocytopenia, agranulocytosis, mild urticaria

Cytochrome P450 Inducers

Chronic alcohol use, Modafinil, St Johns Wort, Phenytoin, Phenobarbital, Nevirapine, Rifampin, Griseofulvin, Carbamazepine

Chronic alcoholic Mona Steals Phen-Phen and Never Refuses Greasy Carbs

Cytochrome P450 Substrates

Anti-epileptics, Antidepressants, Antipsychotics, Anesthetics, Theophylline, Warfarin, Statins, OCPs

Always, Always, Always, Always Think When Starting Others

Cytochrome P450 Inhibitors

Acute alcohol use, Gemfibrozil, Ciprofloxacin, Isoniazid, Grapefruit juice, Quinidine, Amiodarone, Ketoconazole, Macrolides, Sulfonamides, Cimetidine, Ritonavir

A cute Gentleman Cipped Iced Grapefruit juice Quickly And Kept Munching on Soft Cinammon Rolls

Antimuscarinic rxn

Atropine, TCAs, H1-blockers, antipsychotics

Disulfiram-like rxn

Metronidazole, certain Cephalosporins, Griseofulvin, Procarbazine, 1st generation Sulfonylureas

Nephrotoxicity/ototoxicity rxn

Aminoglycosides, vancomycin, loop diuretics, cisplatin

Dry cough rxn

ACE inhibitors

Pulmonary fibrosis rxn

Bleomycin, Amiodarone, Busulfan, MTX

Breathing Air Badly from Medications

SIADH rxn

Carbamazepine, Cyclophosphamide, SSRIs

Can't Concentrate Serum Sodium

Interstitial nephritis rxn

Methicillin, NSAIDs, furosemide

Hemorrhagic cystitis rxn

Cyclophosphamide, ifosfamide

Prevented by coadministering with mesna

Fanconi syndrome rxn

Expired tetracycline

Diabetes insipidus rxn

Lithium, demeclocycline

Tardive dyskinesia rxn

Antipsychotics, metoclopramide

Seizures rxn

INH (vitB12 def), Bupropion, Imipenem/cilastatin, Tramadol, Enflurane, Metoclopramide

With seizures I BITE My tongue

Parkinson-like syndrome rxn

Antipsychotics, Reserpine, Metoclopramide

Cogwheel rigidity of ARM

Cinchonism

Quinidine, quinine

Tendonitis/tendon rupture/cartilage damage

Fluoroquinolones

Teeth discolouration rxn

Tetracyclines

SLE-Like syndrome rxn

Sulfa drugs, Hydralazine, INH, Procainamide, Phenytoin, Etanercept

Having lupus is SHIPP-E

Steven-Johnson syndrome rxn

Anti-epileptics, Allopurinol, Sulfa drugs, Penicillin

Steven Johnson has epileptic Allergy to Sulfa drugs and Penicillin

Photosensitivity rxn

Sulfonamides, Amiodarone, Tetracyclines, 5-FU

SAT for photo

Osteoporosis rxn

Corticosteroids, heparin

Myopathy rxn

Fibrates, niacin, colchicine, hydroxychloroquine, interferon-alpha, penicillamine, statins, glucocorticoids

Hyperuricemia rxn

Pyrazinamide, Thiazides, Furosemide, Niacin, Cyclosporine

Painful Tophi and Feet Need Care

Gingival hyperplasia rxn

Phenytoin, verapamil, cyclosporine, nifedipine

Fat redistribution rxn

Protease inhibitors, glucocorticoids

Fat PiG

Thrombotic complications rxn

OCPs - estrogen

Thrombocytopenia rxn

Heparin, cimetidine

Megaloblastic anemia rxn

Phenytoin, MTX, Sulfa drugs

Having a blast with PMS

Hemolysis in G6PD deficiency

INH, Sulfonamides, Dapsone, Primaquine, Aspirin, Ibuprofen, Nitrofurantoin

Hemolysis IS D PAIN

Gray baby syndrome rxn

Chloramphenicol

Direct Coombs+ hemolytic anaemia rxn

Methyldopa, penicillin

Aplastic anemia rxn

Carbamazepine, Methimazole, NSAIDs, Benzene, Chloramphenicol, Propylthiouracil

Can't Make New Blood Cells Properly

Agranulocytosis rxn

Dapsone, Clozapine, Carbamazepine, Colchicine, Methimazole, Propylthiouracil

Drugs CCCrush Myeloblasts and Promyelocytes

Pseudomembranous colitis rxn

Clindamycin, ampicillin, cephalosporins

Abx predispose to superinfection by resistant C Diff

Pancreatitis rxn

Didanosine, Corticosteroids, Alcohol, Valproic acid, Azathioprine, Diuretics

Drugs Causing A Violent Abdominal Distress

Hepatitis rxn

INH

Focal -> Massive hepatic necrosis rxn

Halothane, Amanita phalloides (death cap mushroom), Valproic acid, Acetaminophen

Liver HAVAc

Diarrhoea rxn

Metformin, Erythromycin, Colchicine, Orlistat, Acarbose

Might Excite Colon On Accident

Acute cholestatic hepatitis, jaundice rxn

Erythromycin

Hypothyroidism rxn

Lithium, Amiodarone, Sulfonamides

Hyperglycaemia rxn

Tacrolimus, Protease inhibitors, Niacin, HCTZ, Beta-blockers, Corticosteroids

Taking Pills Necessitates Having Blood Checked

Hot flashes rxn

Tamoxifen, clomiphene

Adrenocortical insufficiency rxn

HPA suppression secondary to glucocorticoid withdrawal

Torsades de pointed rxn

Class 3 (sotalol) and class 1A (quinidine) antiarrhythmics, Macrolides, Abx, antipsychotics, TCAs

Dilated cardiomyopathy rxn

Doxorubicin, Daunorubicin

Cutaneous flushing rxn

Vancomycin, Adenosine, Niacin, Ca channel blockers

VANC

Coronary vasospasm rxn

Cocaine, sumatriptan, ergot alkaloids

Acetaminophen AtD

N-acetylcysteine

Replenishes glutathione

AChE inhibitors, organophosphates AtD

Atropine, followed by pralidoxine

Amphetamines AtD

NH4Cl

Antimuscarinics, anticholinergic agents AtD

Physostigmine salicylate, control hyperthermia

Benzodiazepine AtD

Flumazenil

Beta-blockers AtD

Glucagon

CO AtD

100% O2, hyperbaric O2

Cu, arsenic, gold AtD

Penicillamine

Cyanide AtD

Nitrite + thiosulfate, hydroxocobalamin

Digitalis AtD

Anti-dig Fab fragments

Heparin AtD

Protamine sulfate

Iron AtD

Deferoxamine, deferasirox

Lead AtD

EDTA, dimercaprol, penicillamine, succimer for children

Mercury, arsenic, gold AtD

Dimercaprol, succimer

Methanol, ethylene glycol AtD

Fomepizole, ethanol, dialysis

Methemoglobin AtD

Methylene blue, vitamin C

Opioids AtD

Naloxone

Salicylates AtD

NaHCO3, dialysis

TCAs AtD

NaHCO3

tPA, streptokinase, urokinase AtD

Aminocaproic acid

Warfarin AtD

Vitamin K, plasma if active bleeding