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444 Cards in this Set

  • Front
  • Back
amoxicillin
aminopenicillin
methicillin
penicillinase resistant penicillin
ampicillin
aminopenicillin
nafcillin
penicillinase resistant penicillin
dacloxacillin
penicillinase resistant penicillin
Ticarcillin
antipseudomonal
Carbenicillin
antipseudomonal
Piperacillin
antipseudomonal
cefazolin
1st gen cephalosporin
cephalexin
1st gen cephalosporin
cefoxitin
2nd gen ceph
cefaclor
2nd gen ceph
cefuroxime
2nd gen ceph
ceftriaxone
3rd gen ceph
ceftazidime
3rd gen ceph
cefotaxime
3rd gen ceph
cefepime
4th gen ceph
aztreonam
monobactam resistant to beta lactamases
imipenem
carbapenem
cilastatin
used with imipenem
meropenem
carbapenem
vancomycin
binds d-ala d-ala of bacterial cell wall
streptomycin
aminoglycoside
gentamycin
aminoglycoside
tobramycin
aminoglycoside
amikacin
aminoglycoside
neomycin
aminoglycoside
doxycycline
tetracycline
demeclocycline
tetracycline
minocycline
tetracycline
erythromycin
macrolide
azithromycin
macrolide
clarithromycin
macrolide
chloramphenicol
binds 50S
clindamycin
binds 50S
sulfamethoxazole
sulfonamide
sulfisoxazole
sulfonamide
sulfadiazine
sulfonamide
trimethoprim
used with SMX
inhibits dihydrofolate reductase
ciprofloxacin
fluoroquinolone
norfloxacin
fluoroquinolone
ofloxacin
fluoroquinolone
sparfloxacin
fluoroquinolone
moxifloxacin
fluoroquinolone
gatifloxacin
fluoroquinolone
enoxacin
fluoroquinolone
nalidixic acid
fluoroquinolone
metronidazole
antibacterial
antifungal
polymixins
bind bacterial cell membrane
isoniazid
TB
rifampin
TB
pyrazinamide
TB
Ethambutol
TB
dapsone
leprosy
amphotericin B
antifungal, binds ergasterol
nystatin
antifungal, binds ergasterol
azoles
antifungal, inhibit sterol synthesis
fluconazole
azole
ketoconazole
azole
clotrimazole
azole
miconazole
azole
itraconazole
azole
voriconazole
azole
flucytosine
antifungal, used with amph B
caspofungin
antifungal, for asp
terbinafine
antifungal
derm
griseofulvin
antifungal
derm
amantidine
antiviral, prevents uncoating
flu
parkinsons
zanamivir
antiviral
inhibits neuraminidase
flu
oseltamivir
antiviral
blocks neuraminidase
flu
Ribavirin
antiviral
rsv, hep c
acyclovir
antiviral
Herpes viruses
ganciclovir
antiviral
CMV
foscarnet
antiviral
CMV
ritonavir
protease inhibitor
HIV
saquinavir
protease inhibitor
HIV
indinavir
protease inhibitor
HIV
nelfinavir
protease inhibitor
HIV
amprenavir
protease inhibitor
HIV
zidovudine
nucleoside RT inhib
HIV
didanosine
nucleoside RT inhib
HIV
zalcitabine
nucleoside RT inhib
HIV
stavudine
nucleoside RT inhib
HIV
lamivudine
nucleoside RT inhib
HIV
abacavir
nucleoside RT inhib
HIV
nevirapine
non nuc RT inhib
HIV
efavirenz
non nuc RT inhib
HIV
Delavirdine
non nuc RT inhib
HIV
enfuvirtide
fusion inhibitor
HIV
IFN alpha
hep b and c
kaposis
IFN beta
MS
IFN gamma
NADPH oxidase deficiency
cyclosporine
immunosuppressant
organ transplant
tacrolimus FK506
immunosuppressant
organ transplant
azathioprine
immunosuppressant
kidney transplant
autoimmune
Muromonab CD3 (OKT3)
immunosuppressant
kidney transplant
sirolimus (rapamycin)
immunosuppressant
kidney transplant
mycophenolate mofetil
immunosuppressant
wegener's?
daclizumab
immunosuppressant
aldesleukin
recombinant cytokine IL 2
renal cell carcinoma
melanoma
erythropoietin
recombinant cytokine
anemias in renal failure
filgrastim
recombinant cytokine
granulocyte colony stimulating factor
recovery of BM
sargramostim
recombinant cytokine
granulocyte macrophage colongy stimulating factor
recovery of bone marrow
oprelvekin
interleukin 11
thrombocytopenia
thrombopoietin
recombinant cytokine
thrombocytopenia
Methylphenidate
ritalin
increases NE release
amphetomine-like
ADHD
Haloperidol
antispychotic
trifluoperazine
antipsychotic
fluphenazine
antipsychotic
thioridazine
antipsychotic
chlorpromazine
antipsychotic
clozapine
atypical antipsychotic
olanzapine
aytpical antipsychotic
risperidone
atypical antipsychotic
aripiprazole
atypical antipsychotic
quetiapine
atypical antipsychotic
ziprasidone
atypical antipsychotic
lithium
mood stabilizer for bipolar disorder
buspirone
antianxiety
stimulates seratonin receptors
imipramine
TCA
amitriptyline
TCA
desipramine
TCA
nortriptyline
TCA
clomipramine
TCA
Doxepin
TCA
Amoxapine
TCA
Fluoxetine
SSRI
paroxetine
SSRI
Sertraline
SSRI
Citalopram
SSRI
Bupropion
Wellbutrin
antidepressant
Venlafaxine
antidepressant
antianxiety
Duloxetine
antidepressant
Mirtazapine
antidepressant
Maprotiline
antidepressant
Trazadone
insomnia
antidepressant at high doses
Phenelzine
MAO inhibitor
tranylcypromine
MAO inhibitor
mannitol
osmotic diuretic
acetazolamide
carbonic anhydrase inhibitor
diuretic
furosemide
sulfonamide loop diuretic
ethacrynic acid
loop diuretic, not a sulfa
hydrochlorothiazide
thiazide diuretic
spironolactone
K sparing diuretic
Triamterene
K sparing diuretic
Amiloride
K sparing diuretic
eplerenone
K sparing diuretic
captopril
ACE inhibitor
Enalopril
ACE inhibitor
Lisinopril
ACE inhibitor
Losartan
Angio II receptor antagonist
finasteride
propecia
antiandrogen
promotes hair growth, BPH
flutamide
antiandrogen
prostate ca
ketoconazole
antiandrogen
blocks steroid synth
tx: Polycystic ovarian syndrome hirsutism
spironolactone
antiandrogen
blocks steroid binding
tx: Polycystic ovarian syndrome hirsutism
leuprolide
GnRH analogue
infertility, prostate ca, fibroids
Sildenafil
cGMP phosphodiesterase inhib
increases blood flow, smooth muscle relax
ED
Vardenafil
cGMP phosphodiesterase inhib
increases blood flow, smooth muscle relax
ED
Mifepristone RU-486
progestin inhibitor
termination of preg
synthetic progestins, estrogen
oral contr
dinoprostone
PGE2 analogue
induces labor
ritodrine
beta 2 agonist
relaxes uterus, reduce contractions
terbutaline
beta 2 agonist
relaxes uterus, reduce contractions
anastrozole
aromatase inhibitor
post menop. breast ca
exemestane
aromatase inhibitor
post menop breast ca
exemestane
testosterone
treat ER positive breast ca
ethinyl estradiol
estrogen
DES
estrogen
mestranol
estrogen
Selective estrogen receptor modulators
estrogen receptor agonists
infertility
PCOS
diphenhydramine
H1 blocker
allergy, motion sickness, sleep
dimenhydrinate
H1 blocker,
allergy, motion sickness, sleep
chlorpheniramine
H1 blocker
allergy, motion sickness, sleep
loratidine
H2 blocker
allergy
fexofenadine
H2 blocker
allergy
desloratadine
H2 blocker
allergy
cetirizine
H2 blocker
allergy
isoproterenol
nonspecific beta agonist
asthma
albuterol
beta 2 agonist
asthma
salmeterol
beta 2 agonist
long acting asthma
formoterol
beta 2 agonist
long acting asthma
theophylline
methylxanthine
inhibits phosphodiesterase
asthma
ipratropium bromide
M3 antagonist
asthma
tiotropium
M3 antagonist
asthma
cromolyn
stabilizes mast cells
asthma
beclomethasone
corticosteroid
zileuton
antileukotriene, blocks 5LPO
asthma
zafirlukast
antileukotriene
blocks receptor
asthma
montelukast
antileukotriene
blocks receptor
asthma
guaifenesin
expectorant
removes sputum
Robitussin
N-acetylcysteine
mucolytic
CF
acetaminophen OD
clonidine
sympathoplegic
anti HTN
methyldopa
sympathoplegic
anti HTN
Reserpine
sympatheoplegic
anti HTN
Guanethidine
sympathoplegic
anti HTN
Prazosin
sympathopolegic
anti HTN
hydralazine
vasodilator
anti HTN
CHF
minoxidil
vasodilator
K channel opener
anti HTN
nifedipine
vasodilator
Ca channel blocker
anti HTN
verapamil
vasodilator
Ca channel blocker
Class IV antiarrhythmic
anti HTN
nitroprusside
vasodilator
causes release of NO
anti HTN
diazoxide
vasodilator
K channel opener
anti HTN
diltiazem
vasodilator
ca channel blocker
Class IV antiarrhythmic
anti HTN
nitroglycerin
vasodilator of veins
angina
pulm edema
isosorbide dinitrate
vasodilates veins
angina
pulm edema
Fenoldopam
D1 agonist
relaxes smooth muscle
Pindolol
partial beta antagonist
acebutolol
partial beta blocker
lovastatin
HMG-CoA reductase inhibitor
pravastatin
HMG-CoA reductase inhibitor
simvastatin
HMG-CoA reductase inhibitor
atorvastatin
HMG-CoA reductase inhibitor
rosuvastatin
HMG-CoA reductase inhibitor
Niacin
lowers LDL
cholestyramine
bile acid resin
lipid lowering agent
colestipol
bile acid resin
lipid lowering
colesevelam
bile acid resin
lipid lowering
ezetimibe
cholesterol absorption blocker
gemfibrozil
fibrate
lipid lowering
clofibrate
fibrate
lipid lowering
bezafibrate
fibrate
lipid lowering
fenofibrate
fibrate
lipid lowering
digoxin
cardiac glycoside
inhibits Na/K pump, inc Ca inside cells--> inc contractility
CHF, afib
Quinidine
class 1A Na channel blocker
antiarrhytmic
procainamide
class 1A Na channel blocker
antiarrhytmic
disopyramide
class 1A Na channel blocker
antiarrhythmic
lidocaine
class 1B Na channel blocker
antiarrhythmic
Mexiletine
class 1B Na channel blocker
antiarrhythmic
Tocainide
class 1B Na channel blocker
antiarrhythmic
Flecainide
class 1C Na channel blocker
antiarrhythmic
encainide
class 1C Na channel blocker
antiarrhythmic
Propafenone
class 1C Na channel blocker
antiarrhythmic
sotalol
class III K channel blocker
antiarrhythmic
ibutilide
class III K channel blocker
antiarrhythmic
amiodarone
class III K channel blocker
antiarrhythmic
adenosine
inc k removal from cell
antiarrhythmic
K+
digoxin toxicity
Mg2+
digoxin toxicity
Torsades de pointes
lispro
short acting insulin
aspart
short acting insulin
NPH
intermediate insulin
glargine
long acting insulin
detemir
long acting insulin
tolbutamide
1st gen sulfonylurea
triggers insulin release
chlorpropamide
1st gen sulfonylurea
insulin release
glyburide
2nd gen sulfonylurea
insulin release
glimepiride
2nd gen sulfonylurea
insulin release
glipizide
2nd gen sulfonylurea
insulin release
metformin
biguanide
insulin sensitizer
pioglitazone
glitazone
inc cell response to insulin
rosiglitazone
glitazone
inc cell response to insulin
acarbose
alpha glucosidase inhibitor
dec hyperglycemia
miglitol
alpha glucosidase inhibitor
dec hyperglycemia
pramlintide
mimetic
dec glucagon
exenatide
GLP-1 mimetic
inc insulin
orlistat
inhibits pancreatic lipase
obesity
sibutramine
sympathomimetic serotonin and NE reuptake inhibitor

obesity
propylthiouracil
hyperthyroidism
methimazole
hyperthyroidism
Somatostatin (octreotide)
hypothalmic/pituitary drug
oxytocin
hypothalmic/pituitary drug
induces labor
ADH (desmopressin)
pituitary drug
levothyroxine
hypothyroidism
myxedema
triiodothyronine
hypothyroidism
myxedema
hydrocortisone
glucocorticoid
dec leukotrienes and prostaglandins
prednisone
glucocorticoid
dec leukotrienes and prostaglandins
triamcinolone
glucocorticoid
dec leukotrienes and prostaglandins
dexamethosone
glucocorticoid
dec leukotrienes and prostaglandins
demeclocycline
tetracycline
ADH antagonist
diabetes, SIADH
Cimetidine
H2 blocker
ulcers, reflux
Ranitidine
H2 blocker
ulcer, reflux
Famotidine
H2 blocker
ulcer, reflux
Nizatidine
H2 blocker
ulcer, reflux
Omeprazole
Proton pump inhibitor
ulcer, reflux
Lansoprazole
proton pump inhibitor
ulcer, reflux
Bismuth
binds ulcers
H pylori
sucralfate
binds ulcers
Misoprostol
PGE1 analog
maintain PDA
ulcers
X preg!!
Pirenzepine
M1 and M3 blocker
blocks histamine and acid
ulcer
Propantheline
M1 and M3 blocker
blocks histamine and acid
ulcer
aluminum hydroxide
antacid
magnesium hydroxide
antacid
calcium carbonate
antacid
infliximab
immunosuppressant
monoclonal antibody to TNF
Crohns, Rh arthritis
Sulfasalazine (5-ASA)
activated by colonic bacteria
crohns, UC
Ondansetron
Zofran
seretonin antagonist
nausea
Metoclopramide
D2 antagonist
gastroparesis- diabetes and post surgery
heparin
activates antithrombin III
follow PTT
anticoagulant
lepirudin
hirudin derivative
inhibits thrombin
bivalirudin
hirudin derivative
inhibits thrombin
warfarin (coumadin)
blocks vit k dep clotting factor synth
follow PT/INR
anticoagulant
streptokinase
thrombolytic
urokinase
thrombolytic
alteplase
tPA
thrombolytic
anistreplase (APSAC)
thrombolytic
aspirin
irreversibly inhibits COX 1 and 2
Clopidogrel
inhibits platelet aggregation
blocks ADP receptors
inhibits fibrinogen
Ticlopidine
inhibits platelet aggregation
blocks ADP receptors
inhibits fibrinogen
abciximab
monoclonal antibody binds platelets
prevents aggregation
Methotrexate
folic acid analog inhibits dihydrofolate reductase, inh dna synth.
leukemia, lymphoma, etc
5 fluorouracil
antimetabolite
colon cancer
bcc
6 Mercaptopurine
blocks purine synth
leuk, lymphoma
Cytarabine (ara-C)
inhibits DNA pol
AML, ALL, non Hodgkins lymph
cyclophosphamide
alkylating agent
NHL, breast, ovca
Ifosfamide
alkylating agent
NHL, breast, ovca
carmustine
nitrosourea
alkylating agent
brain tumors
lomustine
nitrosourea
alkylating agent
brain tumors
semustine
nitrosourea
alkylating agent
brain tumors
streptozocin
nitrosourea
alkylating agent
brain tumors
cisplatin
cross links dna
test, bladder, lung, ovca
carboplatin
cross links dna
test, bladder, lung, ovca
Busulfan
alkylates dna
CML
doxorubicin
adriamycin
DNA breaks
Hodgkins, myelomas, sarcomas,
solid-br/ov/lung
daunorubicin
DNA breaks
Hodgkins, myelomas, sarcomas,
solid-br/ov/lung
dactinomycin
actinomycin D
intercalates in DNA
wilms, ewings, rhabdo
bleomycin
DNA breaks
test, ovca, HL
hydroxyurea
inhibits dna synth
melanoma, CML, sickle cell
etoposide (VP 16)
inhibits topo
lung, prostate, testicular ca
tamoxifen
SERMs- receptor ant in breast
breast cancer
raloxifene
SERMs- receptor ant in breast
breast cancer
Trastuzumab
herceptin
HER-2 antibody
breast cancer
Imatinib
gleevec
bcr-abl tyrosine kinase inhibitor
CML, GI tumors
Vincristine
blocks microtubules
HL, wilms, choriocarcinoma
vinblastine
blocks microtubules
HL, wilms, choriocarcinoma
paclitaxel
binds microtubules
breast and ovca
ibuprofen
NSAID
COX 1 and 2
naproxen
NSAID
COX 1 and 2
indomethacin
NSAID
COX 1 and 2
ketorolac
NSAID
COX 1 and 2
celecoxib
COX 2 inhibitor
arthritis
acetaminophen
reversibly inhibits COX
etidronate
bisphosphonate
inhibits osteoclasts
hypercalcemia, Paget's, osteoporosis
pamidronate
bisphosphonate
inhibits osteoclasts
hypercalcemia, Paget's, osteoporosis
alendronate
bisphosphonate
inhibits osteoclasts
hypercalcemia, Paget's, osteoporosis
risedronate
bisphosphonate
inhibits osteoclasts
hypercalcemia, Paget's, osteoporosis
colchicine
blocks microtubules
gout
probenecid
inhibits uric acid resorption
gout
allopurinol
inhibits Xanthine Oxidase
gout
etanercept
binds TNF
rh arthritis, ankylosing spondylitis
infliximab
anti TNF
crohns, rh arthritis, ank spond.
pilocarpine
cholinomemetic
glaucoma
carbachol
cholinomemetic
glaucoma
physostigmine
cholinomemetic
glaucoma
echothiophate
cholinomemetic
glaucoma
latanoprost
prostaglandin
glaucoma
morphine
opioid analgesic
mu receptor
fentanyl
opioid analgesic
codeine
opioid analgesic
heroin
opioid analgesic
methadone
opioid analgesic
addiction programs
meperidine
opioid analgesic
dextromethorphan
opioid analgesic
pain, cough
loperamide
opioid analgesic
diarrhea
diphenoxylate
opioid analgesic
diarrhea
butorphanol
partial opioid analgesic
mu
tramadol
weak opioid agonist
phenytoin
block Na channel
epilepsy
simple, complex, general T-C
carbamazepine
blocks Na channel
epilepsy
simple, complex, general T-C
trigeminal neuralgia
lamotrigine
blocks Na channels
epilepsy
simple, complex, general T-C
gabapentin
increases GABA
epilepsy
simple, complex, general T-C
topiramate
blocks Na, inc GABA
epilepsy
simple, complex, general T-C
phenobarbital
inc GABA
epilepsy
simple, complex, general T-C
valproic acid
blocks Na, Inc GABA
epilepsy
simple, complex, general T-C
ethosuximide
blocks Ca T channels
epilepsy
general absence seizures
benzodiazepines
inc GABA
epilepsy
phenobarbital
barbiturate
inc GABA
pentobarbital
barbiturate
inc GABA
thiopental
barbiturate
inc GABA
secobarbital
barbiturate
inc GABA
diazepam
benzo
inc GABA
lorazepam
benzo
inc GABA
triazolam
benzo
inc GABA
temazepam
benzo
inc GABA
oxazepam
benzo
inc GABA
midazolam
benzo
inc GABA
chlordiazepoxide
benzo
inc GABA
alprazolam
benzo
inc GABA
halothane
inhaled anesthetic
enflurane
inhaled anesthetic
isoflurane
inhaled anesthetic
sevoflurane
inhaled anesthetic
methoxyflurane
inhaled anesthetic
nitrous oxide
inhaled anesthetic
thiopental
barbituate
IV anesthetic
midazolam
benzo
IV anesthetic for endoscopy
arylcyclohexylamine
ketamine
PCP analogue
IV anesthetic
propofol
rapid IV anesthetic
procaine
local anesthetic
ester
blocks Na channels
tetracaine
local anesthetic
ester
blocks Na channels
lidocaine
local anesthetic
amide
blocks Na channels
mepivacaine
local anesthetic
amide
blocks Na channels
bupivacaine
local anesthetic
amide
blocks Na channels
succinylcholine
neuromuscular blocking
depolarizing
tubocurarine
neuromuscular blocking
nondepolarizing
binds ACh receptor
atracurium
neuromuscular blocking
nondepolarizing
binds ACh receptor
mivacurium
neuromuscular blocking
nondepolarizing
binds ACh receptor
pancuronium
neuromuscular blocking
nondepolarizing
binds ACh receptor
vecuronium
neuromuscular blocking
nondepolarizing
binds ACh receptor
rocuronium
neuromuscular blocking
nondepolarizing
binds ACh receptor
neostigmine
cholinesterase inhibitor
edrophonium
cholinesterase inhibitor
dantrolene
treats malignant hypothermia
bromocriptine
Dopamine receptor agonist
parkinsons
amantadine
inc dopamine
parkinsons
flu
rubella
levodopa
with carbidopa
converted to Dopa in CNS
parkinsons
selegiline
MAO B inhibitor
antimuscarinic
parkinsons
entacapone
COMT inhibitor
antimuscarinic
parkinsons
tolcapone
COMT inhibitor
antimuscarinic
parkinsons
benztropine
antimuscarinic
parkinsons
sumatriptan
seretonin agonist
migraines
memantine
NMDA receptor antagonist
alzheimers
donepezil
Ach-esterase inhibitor
alzheimers
propranolol
nonselective beta blocker
timolol
nonselective beta blocker
nadolol
nonselective beta blocker
pindolol
partial beta agonist
acebutolol
partial beta antagonist
labetalol
nonselective beta blocker
alpha blocker
betaxolol
beta 1 blocker
esmolol
b1 blocker
atenolol
b1 blocker
metoprolol
b1 blocker
carvedilol
nonselective a and b blocker
NaHCO3
salicylate OD
TCA OD
NH4Cl
amphetamine OD
pralidoxime
anticholinesterases or organophosphate OD
physostigmine salicylate
antimuscarinic or anticholinergic OD
glucagon
Beta blocker OD
deferoxamine
Iron OD
CaEDTA
lead OD
demercaprol
lead OD
mercury OD
arsenic OD
gold OD
penicillamine
lead
copper
arsenic
gold
nitrite
cyanide OD
hydroxycobalamin
cyanide OD
thiosulfate
cyanide OD
methylene blue
methemoglobin OD
fomepizole
methanol
ethylene glycol OD
naloxone
opioid OD
naltrexone
opioid OD
flumazenil
benzo OD
protamine
heparin OD
aminocaproic acid
tPA OD
theophylline OD
beta blocker
Most potent anti-dopamine drugs
metoclopramide
phenothiazines (haloperidol, antispychotics)

causes-- hyperprolactinemia