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49 Cards in this Set

  • Front
  • Back
NE
α agonist
Phenlephrine
Methoxamine
Metaraminol
Tetrahydrozoline
α1 agonist
Clonidine
α-Methyldopa
α2 agonist

(↓ NE release)
Phenoxybenzamine
Prazosin
α antagonists
Albuterol
Terbutaline
Metaproterenol
β2 agonist

(activate adenylyl cyclase → ↑ cAMP → bronchodilation)
Isoproterenol
β agonist
Propranolol
(and others ending in -olol)
β antagonist

(Class II anti-arrhythmic)
(anti-angina)
Epi
α & β agonist
Ephedrine
Amphetamine
α & β agonist

(ephedrine - β)
(amphetamine - α)
Cocaine
prevent re-uptake of NE
Reserpine
prevent SYNTHESIS of NE
Guanethidine
prevent RELEASE of NE
Pilocarpine
Bethanecol
Carbachol
muscarinic cholinergic AGONIST

(↓ HR, vasodilation, bronchoconstriction, mydriasis)
Atropine
Scopolamine
muscarinic cholinergic ANTAGONIST

(↑ HR, vasoconstriction, bronchodilation, myosis)
Physostigmine
Neostigmine
Anti-AchE

(prevent degradation of Ach)
(↑ [Ach])
Pralidoxime
antidote to Anti-AchE
Turbocurarine
NON-DEPOLARAIZING Anti-nicotinic cholinergic acting at NMJ (Neuromuscular Blockade)

(Produce paralysis)
Succinylcholine
DEPOLARAIZING Anti-nicotinic cholinergic acting at NMJ
(Neuromuscular Blockade)

(Produce paralysis)
Mannitol
Osmotic diuretic
Acetazolamide
CA-Inhibitor diuretic

(Inhibits carbonate reabsorption = ↓ Na⁺ reabsorption & H⁺ excretion)
Furosemide
Ethacrynic Acid
Loop diuretic

(Furosemide = sulfonamide)
(Ethacrynic Acid = non-sulfonamide)

(Inhibit Na⁺-K⁺-2Cl⁻ symport)
Spironolactone
K⁺ Sparing diuretic

(aldosterone antagonist)
(inhibits Na⁺ reabsorption)
Amiloride
K⁺ Sparing diuretic

(Na⁺ channel inhibitor)
(inhibits Na⁺ reabsorption)
Verapamil
Ca²⁺ channel blocker

(Class IV anti-arrhythmic)
(anti-angina)
Lisinopril
Benazepril
(and other drugs that end in -pril)
ACE Inhibitors
Hydrochlorothiazide
Thiazide diuretic

(inhibit Na⁺-Cl⁻ symport)
Digoxin
Digitoxin
Glycoside (inotrope)

(for CHF)
Milrinone
Phosphodiesterase III inhibitor (inotrope)

(for CHF)
Hydralazine
Minoxidil
Sodium nitroprusside
Direct vasodilators
Nifedipine
Ca²⁺ channel blocker

(Class IV anti-arrhythmic)
(anti-angina)
Losartan
Angiotensin-II Receptor Antagonist
Quinidien
Procainamide
Lidocaine
Phenytoin
Na⁺ channel blockers
(Class I anti-arrhythmic)
Nitroglycerin
Nitrate/Nitrite

(anti-angina)
Aspirin
NSAID

(salicylate)
Ibuprofin
NSAID

(propionic acid)
Naproxen
NSAID

(propionic acid)
Acetaminophen
NSAID?

(aminophenol)

(NOT anti-inflammatory)
Sulfasalazine
penicillamine
hydroxychloroquine
methotrexate
DMARD

(anti-rheumatoid)
cyclosporin tacrolimus
azathioprine
glucocorticoids
Immunosuppressant

(anti-rheumatoid)
Infliximab
adalimumab
etanercept
anakinra
Anti-cytokine / Biopharmaceuticals

(anti-rheumatoid)
Cromolyn
Epinephrine
INDIRECT anti-histamine

(Cromolyn - prevents mast cell degranulation)
(Epi - counteracts histamine activity)
Diphenhydramine
Chlorpheniramine
Promethazine
H1 antagonists (1st gen)
Loratadine
Fexofenadine
H1 antagonists (2nd gen)
Promethazine
Meclizine
Dimenhydrinate
H1 antagonists (1st gen)
(anti-emetic & motion sickness)
Cimetidine
Famotidine
Ranitidine
H2 antagonists
Beclomethasone
Flunisolide
Inhaled corticosteroids

(anti-asthma)
Montelukast
Zafirlukast
Leukotriene antagonists

(anti-asthma)
Theophyline
Methylxanthine

(anti-asthma)

(inhibits PDE → ↑ cAMP → bronchodilation)
Dobutamine
β1 agonist