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11 Cards in this Set
- Front
- Back
- 3rd side (hint)
Sildenafil
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phosphodiesterase 5 antagonist
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PDE5 antagonist=>prevents conversion of cGMP=>prolonged relaxation
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Alprostadil
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PGE1
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Vasodilator
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Oxybutynin
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non-selective M antagonist
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Blocks M receptors=>inhibits ACh=>detrusor relaxation
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Mirabegron
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B2 adrenergic agonist
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Activates B2 receptor on detrusor=>relaxes
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Darifenacin
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M3 antagonist
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BLocks M3=>bladder relaxes
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Solifenacin
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M3 antagonist
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BLocks M3=>bladder relaxes
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Tolterodine
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M3 antagonist
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BLocks M3=>bladder relaxes
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Desmopression
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ADH analogue
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Binds V2 receptors=>increases water resorption=>decreases urine
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Phenylephrine
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a1 agonist
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Binds a1 receptors=>vasoconstricts=>detumescence
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Tamsulosin
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a1 antagonist
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BLocks a1 receptors=>relaxation=>less resistance to flow in BPH
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Alfuzosin
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a1 antagonist
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BLocks a1 receptors=>relaxation=>less resistance to flow in BPH
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