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76 Cards in this Set
- Front
- Back
Endrophonium
|
Rev ACE-I
*Myasthenia Gravis |
|
Physostigmine
|
Rev ACE-I
*glaucoma |
|
Neostigmine
|
Rev ACE-I
*ileus, urinary ret, myasthenia gravis |
|
Pyridostigmine
|
Rev ACE-I
*ileus, urinary ret, myasthenia gravis |
|
Echothiophate
|
Irrev ACE-I
|
|
Malathion
|
Irrev ACE-I
|
|
Parathion
|
Irrev ACE-I
|
|
Rx for Malathion/Parathion OD
|
Atropine + 2PAM
|
|
Acetylcholine
|
Dir Cholinomimetic
|
|
Bethanechol
|
Dir Cholinomimetic
|
|
Metacholine
|
Dir Cholinomimetic
|
|
Pilocarpine
|
Dir Cholinomimetic
|
|
Donezepil
|
Rev ACE-I
|
|
Tacrine
|
Rev ACE-I
|
|
Atropine
|
M-blocker
|
|
Scopolamine
|
M-blocker
|
|
Glycopyrolate
|
M-blocker
|
|
Benztropine
|
M-blocker
|
|
Trihexylphenidyl
|
M-blocker
|
|
Ipratropium
|
M-blocker
|
|
Tropicamide
|
M-blocker
*topical ophthalmic use |
|
Hexamethonium
|
Ganglionic blocker
|
|
Mecamylamine
|
Ganglionic blocker
|
|
Succinylcholine
|
Depolarizing NMJ blocker
*Nm agonist |
|
Tubocurarine
|
Non-depolarizing NMJ blocker
*Nm competitive antagonist |
|
Atracurium
|
Non-depolarizing NMJ blocker
*Nm competitive antagonist |
|
Pancuronium
|
Non-depolarizing NMJ blocker
*Nm competitive antagonist |
|
Phenylephrine
|
α1 Agonist
*decongestant |
|
Methoxamine
|
α1 Agonist
*paroxysmal atrial tachycardia |
|
Clonidine
|
α2
*mild/mod htn |
|
α-Methyldopa
|
α2 Agonist
*mild-mod htn |
|
Isoproterenol
|
Nonselective β Agonist
*β1=β2, acute CHF |
|
Dobutamine
|
Nonselective β Agonist
*β1>β2, acute CHF |
|
Salmetelol
|
β2 Agonist
*asthma |
|
Albuterol
|
β2 Agonist
*asthma |
|
Metaproterenol
|
β2 Agonist
*asthma |
|
Terbulatine
|
β2 Agonist
*asthma |
|
Ritrodine
|
β2 Agonist
*premature labor |
|
Norepinephrine
|
α1, α2, β1 Agonist
|
|
Epinephrine
|
α1, α2, β1,
β2 Agonist |
|
Dopamine
|
α1, β1, D1 Agonist
|
|
Tyramine
|
Indirect Sympathomimetic
*displace Ne, inc pressor activity |
|
Amphetamine
|
Indirect Sympathomimetic
*rel Ne, DA, ADHD, wt loss, narcolepsy |
|
Methylphenidate
|
Indirect Sympathomimetic
*rel Ne, DA, ADHD, wt loss, narcolepsy |
|
Ephedrine
|
Indirect Sympathomimetic
*rel NE, decongestant |
|
Cocaine
|
Indirect Sympathomimetic
*loc anesthesia |
|
Phentolamine
|
α1α2 blocker
|
|
Phenoxybenzamine
|
α1α2 blocker
|
|
Prazosin
|
α1 blocker
|
|
Yohimbe
|
α2 blocker
|
|
Mirtazapine
|
α2 blocker
|
|
Acebutolol
|
β1 blocker
|
|
Atenolol
|
β1 blocker
|
|
Esmolol
|
β1 blocker
|
|
Metoprolol
|
β1 blocker
|
|
Pindolol
|
Nonselective β blocker
|
|
Propanolol
|
Nonselective β blocker
|
|
Timolol
|
Nonselective β blocker
|
|
Labetalol
|
Cardio-selective α, β blocker
|
|
Carvedilol
|
Cardio-selective α, β blocker
|
|
Sotalol
|
Cardio-selective β, K+ blocker
|
|
Hemicholinium
|
Block choline uptake
|
|
Botox
|
Block Ach rel
|
|
Methyl-P-tyrosine
|
Inhibit tyrosine hydroxylase so tyrosine can't convert to DOPA
|
|
Phenelzine
|
MAO-I
* inc prejunctional NE |
|
Tranylcypromine
|
MAO-I
* inc prejunctional NE |
|
Reserpine
|
Block granular NE uptake
|
|
Guanethidine
|
Block granular NE release
|
|
Tyosine Hydroxylase
|
Convert tyrosine to DOPA
RLS of catecholamine synthesis |
|
Carbachol
|
GLAUCOMA: Cholinomimetic
*! M = contrxn ciliary muscles = inc fluid outflow |
|
Pilocarpine
|
GLAUCOMA: Cholinomimetic
*! M = contrxn ciliary muscles = inc fluid outflow |
|
Echothiophate
|
GLAUCOMA: Cholinomimetic
*! M = contrxn ciliary muscles = inc fluid outflow |
|
Apraclonidine, Epi
|
GLAUCOMA: Sympathomimetic
*dec NE rel= dec AH syn; inc outflow |
|
Betaxolol, Timolol
|
GLAUCOMA:β blockers
*inh NE = dec AH syn |
|
Acetazolamide
|
GLAUCOMA:carbonic anhydrase inhbiitor
* dec HCO3 = dec AH syn |
|
Latanoprost
|
PGF2α analog
* inc fluid outflow |