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72 Cards in this Set

  • Front
  • Back
epinephrine
a + b agonist
norepinephrine
a + b1
isoproterenol
b
clonidine
a2 agonist
a-methyldopa
a2 agonist
phenylephrine
a1 agonist
guanfacine
a2 agonist
guanabenz
a2 agonist
dobutamine
b1 agonist
albuterol
b2 agonist
dopamine
D1 and B1
methoxamine
a agonist
midodrine
a1 agonist
ephedrine
release of NE, CNS stimulant
xylometazoline
a agonist
oxymetazoline
a agonist
amphetamine
NE stimulant
methamphetamine
NE stimulant wiht higher central action
fenoldopam
D1 agonist
bromocriptine
D2 agonist
phenoxybenzamine
a1 and a2 antagonist
phentolamine
a1 and a2 antagonist
prazosin
a1 antagonist
doxazosin
a1 antogonist
terazosin
a1 antagonist
tamsulosin
a2 antagonist
labetalol
B > a1 antagonist
propranolol
b1 and b2 antagonist
nadolol
b1 and b2 antagonist
timolol
b1 and b2 antagonist
metoprolol
b1>b2 antagonist
atenolol
b1>b2 antagonist
pindolol
b1 and b2 antagonist, partial agonist
carvedilol
b>a1 antagonist
esmolol
b1>b2 antagonist
nitroglycerin
releases NO in smooth muscle
propranolol
b antagonist
verapamil
Ca channel blocker
diltiazem
Ca channel blocker
nifedipine (dihydropyridine)
Ca channel blocker
furosemide
loop diuretic
HCTZ
thiazide antidiuretic
spironolactone
aldosterone antagonist (K sparing diuretic)
captopril
ACE inhibitor
losartan
angiotensin receptor blocker
enalaprildigoxin
ACE inhibitor
carvedilol
b1 antagonist
digoxin
Na-K-ATPase inhibitor
isosorbide dinitrate
releases NO, venodilator
hydralazine
arteriolar dilator
nitroprusside
arteriolar and venodilator
inamrinone
phosphodiesterase type 3 inhibitor
milrinone
phosphodiesterase type 3 inhibitor
nesiritide
natriuretic peptide, diuresis
procainamide
class 1a
primary block Na channels
secondary block K channels
quinidine
class 1a
primary block Na channels
secondary block K channels
lidocaine
class 1b
Na channel blocker
flecainide
class 1c
Na channel blocker
propranolol
class 2
adrenoceptor blocker
amiodarone
K, Na, Ca channel, B blocker
dofetilide
class 3
K channel blocker
verapamil
class 4
Ca channel blocker
diltizem
class 4
Ca channel blocker
adenosine
activates K inward current, blocks Ca channel
magnesium
interacts w/Na-K-ATPase channel
Potassium
increases K permeability
Bile acid sequestrants, resins
High LDL, interrupts enter-hepatic circulation of bile acids and prevents their reabsorption
can raise triglycerides
lowers LDL, small rise in HDL
intestinal absorption inhibitors
High LDL, inhibits lipid precursor absoroption and interrupts enterohepatic recirculation of sterols form bile
Niacin, nicotinic acid
High LDL, High tirglyceride, low HDL

lowers triglycerides, lowers LDL, increases HDL
fibric acid derivatives, fibrates
low HDL, high triglycerides, inhibits triglyceride synthesis
sig lowering of triglycerides
modest rise in HDL
marine oils
high triglycerdies
statins
High LDL