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25 Cards in this Set

  • Front
  • Back
WHAT IS A MUSCARINIC AGONIST?
CHOLINERGIC DRUG. STIMULATES MUSCARINE RECEPTOR, SO IT STIMULATES LOWER BP AND VASODILATION
NAME A MUSCARINIC AGONIST DRUG
BETHANECHOL
BETHANECHOL USED FOR
URINARY RETENTION
BETHANECHOL IS A ____DRUG
CHOLINERGIC
BETHANECHOL CONTRAINDICATIONS
GI LESIONS, HYPERTENSION, ASTHMA
BETHANECHOL SIDE EFFECTS
OVERSTIM OF PNS
NEVER EVER EVER EVER GIVE BETHANECHOL
IM OR IV
BETHANECHOL DANGER
CHOLINERGIC CRISIS
-RESP FAILURE
-INCREASE SALIVATION
-FLACCID PARALYSIS
-CARDIAC FAILURE
WHAT DOES A NICOTINIC STIMULATING DRUG DO?
STIMLUATES NICOTINIC RECEPTOR = EPI RELEASE, SKELETAL MUSCLE CONTRACTIONS INCREASE
NICOTINE PT EDUCATIO
AVOID OTHER STIMULANTS
CORRECT ADM ROUTE
NICOTINE USE
SMOKING REPLACEMENT THERAPY
NICOTINE CONTRAINDICATED
MI, ANGINA, HYPERSENSITIVITY TO NIC, NON SMOKERS,
NICOTINE ADVERSE EFFECTS
VASOCONSTRICTION, INSOMNIA, TACHYCARDIA, HA, FATIGUE
NICOTINE STIM. NICOTINIC RECEPTOR, WHICH MEANS ___RELEASE AND ____
EPI, AND THINK CAFFIENE SIDE EFFECTS. DOES NOT RELAX YOU!!!
NAME THE CHOLINESTERASE INHIBITOR DRUG
NEOSTIGMINE (PROSTIGMIN)
NEOSTIGMINE/PROSTIGMIN USED FOR
MYASTHENIA GRAVIS, ILEO PARALYSIS (POST OP)
URINARY RETENTION
NEOSTIGMINE/PROSTIGMIN CONTRAINDICATED
GI BLOCK, UT BLOCK, ILEO BLOCK
NEOSTIGMINE/PROSTIGMIN SIDE EFFECTS
VASODILATION (LOW BP), CHOLINERGIC CRISIS, RESP ARREST, BRONCHIAL CONSTRICTION, salivation increase, SWEATING
ATROPINE OVERDOSE
MAD AS A HATTER (CNS PSYCHOSIS) DRY AS A BONE (DECREASED SALIVARY) RED AS A BEET (VASODILATION) BLIND AS A BAT (MYDRIASIS)
ATROPINE CONTRAINDICATIONS
TACHYCARDIA, GLAUCOMA, HYPERSENSITIVITY, MYASTHENIA GRAVIS
ATROPINE SIDE EFFECTS
DECREASED : SALIVARY, GI MOTILITY, SWEAT

CONSTIPATION, BLURRED VISION, URINARY RETENTION, CHANGE HR, SMOOTH MUSCLE AND BLADDER CONTRACTION, TACHYCARDIA, HA, DIZZY, DRY MOUTH
ATROPINE =
RAPID ONSET
ATROPINE CAUSES ?
VASOCONSTRICTION =INCREASED HR AND BP

USED FOR 911 BRADYCARDIA
NAME THE CHOLINERGIC ANTAGONIST DRUG:
ATROPINE SULFATE
ATROPINE DOES WHAT?
BLOCKS ACh AT MUSCARINE RECEPTOR SITE. BLOCKS PNS RECEPTOR SITE MUSCARINE.

MUSCARIINE CAUSES VASODILATION AND LOW BP