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14 Cards in this Set
- Front
- Back
Aspirin (acetylsalicylic acid)
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irreversible inactivation of cyclooxygenase.
action- anti-inflammatory, inhibit platelet aggregation, MI. SidEf- normal dos- GI bleeding. large dose- dizziness, deaf, tinnitus, comp respiratory alkalosis. toxic dos- uncomp respiratory & metabolic acidosis. t1\2- 3-5h |
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Diflunisal
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indication- pain, arthritis, inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). less GIT irritation then aspirin. long acting (then aspirin). t1\2- 8-13h |
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Ibuprofen
AKA Nurofen & Advil |
indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). first choice drug, lowest SidEf. t1\2- 2h |
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Naproxen
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indication- pain, fever, inflammation, stiffness, primary dysmenorrhea.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). same as Ibuprofen but stronger and higher chance of SidEf. t1\2- 14h |
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Paracetamol
AKA Acamol, Tylenol |
indication- analgesic, antipyretic, weak anti-inflammatory.
SidEf- in toxic amount stomach bleeding, nausea & vomiting and fatal liver damage. t1\2- 2-4h |
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Diclofenac
AKA Voltaren |
indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). moderate potency and GIT effect. t1\2- 1-2h |
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Indometacin
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). high incidence of headache & dizziness. t1\2- 2h |
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Tolmetin
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). efficacy as ibuprofen, moderate risk of SidEf. t1\2- 5h |
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Piroxicam
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, tinnitus, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). t1\2- 45h |
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Tenoxicam
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). steady state plasma C after 2 weeks. t1\2- 72h |
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Etodolac
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). possibly fewer GIT effects then other. t1\2- 7h |
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Meloxicam
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indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation.
SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). possibly fewer GIT effects then other. t1\2- 20h |
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Celecoxib
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specific COX-2 inhibitor
indication- arthritis, primary dysmenorrhea, fever, analgesic in inflammation. SidEf- Dyspepsia (indigestion), nausea, vomiting, GI damage (for chronic), skin reaction, hemorrhage, reversible renal insufficiency, nephropathy, liver & bone disorder (less common), bronchospasm (if aspirin sensitive asthma). new compound, markedly less GIT toxicity. t1\2- 11h |
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name all the types of NSAIDs
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Aspirin Diclofenac
Diflunisal Indometacin Ibuprofen Tolmetin Naproxen Piroxicam Paracetamol Tenoxicam Etodolac Meloxicam Celecoxib |