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62 Cards in this Set
- Front
- Back
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Inhibit Choline transporter into presynapticnerve neuron
Drug? |
Hemicholinium
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Inhibit ACh storage
drug? |
Vesamicol
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Inhibit ACh release
Drug? |
Botulinum
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blocks accumulation of noradrenaline and dopamine into synaptic vesicles
drug? |
reserpine
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Blocks NE release
Drug? |
Guanethidine
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stimulates NE release
drug? |
amphetamine
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inhibits NE reuptake
drug? |
cocaine
TCA |
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Activates bowel and bladder smooth muscle; resistant to AChE
drug? |
bethanechol
*B*ethanacol=Bowel and Bladder |
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Bethanechol type of agonist
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direct cholinergic agonist
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Activates ciliary muscle of eye
& pupillary sphincter resists AchE treats glaucoma drug? |
Carbachol, pilocarpine
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Treats postoperative and neurogenic ileus and urinary retention
myasthenia gravis reversal of neuromuscular blockade increases endogenous ACh drug? |
Neostigmine
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treatment of myasthenia gravis
increase endogenous ACh drug? |
pyridostigmine
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Diagnosis of myasthenia gravis
increase endogenous ACh |
Edrophonium
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Treats glaucoma (crosses blood brain barrier into CNS
atropine overdose increase endogenous ACh |
Physostigmine
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Echothiophate
treatment for? |
glaucoma
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Pyridostigmine treatment for?
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Myasthenia gravis
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Edrophonium use?
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diagnosis of myasthenia gravis
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phyiostigmine use?
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tx glaucoma
tx atropine overdose |
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Bethanechol mechanism
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cholinergic direct agonist
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carbachol mechanism
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cholinergic direct agonist
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pilocarpine mechanism
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cholinergic direct agonist
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neostgmine mechanism
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anticholinesterase
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pyridostigmine mechanism
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anticholinesterase
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edrophonium mechanism
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anticholinesterase
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physostigmine mechanism
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anticholinesterase
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mechanism of echothiophate
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anticholinesterase
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antidote to cholinesterase inhibitor poisoning
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atropine and pralidoxime
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atropine use in Eye
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poruduce mydriasis and cyclopplegia
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homatropine use in eye
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produce mydriasis and cycloplegia
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tropicamide use in eye?
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Produce mydreiasis and cyloplegia
(cholinoreceptor blocker) |
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benzotropine use in CNS
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tx of parkinson's
(cholinoreceptor blocker) |
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scopolamine use in CNS?
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tx of motion sickness
(cholinoreceptor blocker) |
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Methscopolamine use in genitourinary system
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reduce urgency in mild cystiti and reduce bladder spasms
(cholinoreceptor blocker) |
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oxybutin use in genitourinary system
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reduce urgency in mild cystiti and reduce bladder spasms
(cholinoreceptor blocker) |
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glycopyrrolate use in genitourinary system
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reduce urgency in mild cystiti and reduce bladder spasms
(cholinoreceptor blocker) |
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effect of atropine on eye
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increased pupil dilation, cycloplegia
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effect of atropine on airway
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decreased secretion
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effect of atropine on stomach
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decreeased acid
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effect of atropine on gut
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decreased motility
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effect of atroine on bladder
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decreased urgency in cystitis
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hechanism of mexamethonium
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nicotinic ACh receptor Antagonist
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drug which prevents vagal reflex response to changes in blood pressure
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hexamethonium
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direct general agonist
alpha1 alpha2 beta1 beta2 Drug? |
Epinephrine
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Tx of anaphylaxis, glaucoma (open angle), asthma, hypotension
Drug? |
Epinephrine
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selective for alpha1, alpha2, beta1
drug? |
Norepinephrine
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Tx of hypotension (but decreases renal perfusion)
Drug? |
Norepinephrine
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Selectivity: beta1 = beta2 sympathomimetic
Drug? |
Isoproterenol
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Tx of AV block
Drug? |
Isoproterenol
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amphetamine mechanism
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releases stored catecholamines
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tx of nasal congestion, urinary incontinence, hypotension
drug? |
ephedrine
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ephedrine mechanism
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releases stored catecholamines
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centrally acting alpha agonist, decreased adrenergic outflow
drug? |
clonidine
alpha-methyldopa |
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tx of hypertension, especially with renal disease (no decreased renal blood flow)
drug? |
clonidine
alpha-methyldopa |
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clonidine mechanism
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decreased central adrenergic outflow
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alpha-methyldopa mechanism
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decreased central adrenergic outflow
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clinical use of clonidine
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tx of hypertension w/ renal disease
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clinical use of alpha methyldopa
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tx of hypertensino w/ renal disease
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mechanism of prazosin
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alpha 1 blocker
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mechanism of doxazosin
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alpha 1 blocker
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mirtazapine mechanism
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alpha 2 blocker
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clinical application of mirtazapine
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depression
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mirtazapine side effects
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sedation
increased cholesterol increased appetite |
