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5 Cards in this Set
- Front
- Back
Penicillins
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Mechanism:Bind PBPs; inhibit formation of bridges in peptidoglycan.
Antimicrobial Action: Bactericidal. Spectrum: Gram positive. Inhibition:Beta-lactamases; Efflux of drug; Porin size (Gm -). Notes: PenG=IV, IM PenV=PO 1st gen.; effective vs. growing bacteria. |
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Methicillin
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Mechanism: Bind PBP's, Antimicrobial Action: Bacteriocidal
Inhibition: Same as Penicillin.Spectrum:Gram Positive Notes: Beta Lactamases, Resistant to inactivation by penicillinase of CA-MRSA. |
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Ampicillin
Amoxicillin |
Mechanism: Bind PBP's, Microbial Action: Bacteriocidal
Spectrum: Gm+; growing E. coli, Proteus. Inhibition: Same as Penicillin.Notes: PO 2nd Generation. |
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Carbenicillin
Ticarcillin |
Mechanism: Bind PBP's, Microbial Action: Bacteriocidal
Spectrum: Gm+ & Gm-, incl. Pseudomonas. Inhibition: Resistant to B-lactamases. Notes:Narrow spectrum given to those allergic to penicillin. |
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Monobactams
(Aztreonam) |
Microbial Action: Bacteriocidal
Spectrum: Aerobic Gm-; Enterobac-teriaceae. Inhibition: Same as Penicillin. Notes: PO 3rd Generation. |