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42 Cards in this Set
- Front
- Back
CHOLOMIMETICS:
direct-acting (receptor agonists) choline esters: |
Ach (Miochol)
bethanechol (Urecholin) carbachol (Miostat) methacholine |
|
CHOLOMIMETICS:
direct-acting (receptor agonists) alkaloids |
muscarine (M)
pilocarpine (M, Pilocar) nicotine (N) |
|
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases) - reversible - carbamates |
edrophonium (Tensilon)
demecarium (Humorsol) neostigine (Prostigmin) physostigmine (generic) pyridostigmine (Mestinon) |
|
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases) - reversible - for Alzheimers disease |
donepezil (Aricept)
galntamine (Reminyl) |
|
CHOLOMIMETICS:
indirect-acting (anti-cholinesterases) - irreversible - organophosphates |
echothiophate (phosholine)
malathion parathion soman |
|
CHOLOMIMETICS:
acute narrow angle glaucoma - muscarinic agonist |
pilocarpine (Pilocar) drops
carbachol (Isopto-carbachol) drops |
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CHOLOMIMETICS:
acute narrow angle glaucoma anticholinesterase |
- physostigmine ophth. ointment
- echothiophate (Phospholine) drops - demecarium (Humorsol) drops |
|
CHOLOMIMETICS:
chronic open angle glaucoma anticholinesterase |
- physostigmine
|
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CHOLOMIMETICS:
chronic open angle glaucoma muscarinic agonist |
- pilocarpine
- carbachol |
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Non-CHOLOMIMETICS:
chronic open angle glaucoma carbonic anhydrase inhibitors |
- acetazolamide (Diamox)
- brinzolamide (Azopt) |
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Non-CHOLOMIMETICS:
chronic open angle glaucoma prostaglandins |
- bimatoprost (lumigan)
- unoprostone (Rescula) |
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Non-CHOLOMIMETICS:
chronic open angle glaucoma alpha agonists - non-selective |
- epinephrine
- dipivefrin (Propine) |
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Non-CHOLOMIMETICS:
chronic open angle glaucoma alpha-2 agonists |
- aproclonidine (Iopidine)
- brimonidine (Alphagan) |
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Non-CHOLOMIMETICS:
chronic open angle glaucoma beta blockers |
- betaxolol ( Betoptic )
- timolol ( Timoptic, Betimol) |
|
CHOLOMIMETICS:
GI and urinary tract anticholinesterase |
neostigmine (Prostigmin)
|
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CHOLOMIMETICS:
GI and urinary tract muscarinic agonist |
bethanechol (Urecholine)
|
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CHOLOMIMETICS:
GI and urinary tract for GERD |
H2 blockers
|
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CHOLOMIMETICS:
dry mouth muscarinic agonist |
cevimiline (Evoxac)
|
|
CHOLOMIMETICS:
Myasthenia Gravis (MG) anticholinesterase for diagnosis |
- edrophonium (Tensilon )
|
|
CHOLOMIMETICS:
Myasthenia Gravis (MG) anticholinesterase to assess level of long term treatment |
- edrophonium (Tensilon )
|
|
CHOLOMIMETICS:
Myasthenia Gravis (MG) anticholinesterase long term treatment |
- pyridostigmine ( Mestinon )
- neostigmine (Prostigmin ) - ambenonium (Mytelase ) - demercarium ( Humorsol ) |
|
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade anticholinesterase |
- neostigmine (Prostigmin )
- pyridostigmine ( Mestinon ) - edrophonium (Tensilon ) |
|
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade depolarizing drugs |
- succinylcholine
|
|
CHOLOMIMETICS:
reversal of surgical neuromuscular blockade non-polarizing drugs |
- curare
- atracurium - pipecuronium - pancuronium - vecuronium |
|
CHOLOMIMETICS:
antidote for insecticides and humanocides |
- atropine (Protopam, 2-PAM)
|
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) prototype |
- atropine (Protopam, 2-PAM)
|
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) synthetic tertiary ammonium analogues of atropine |
- dicyclomine (Bentyl)
- tropicamide (Mydriacil) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) synthetic tertiary ammonium analogues of atropine antihistamines |
- dimenhydrinate (Dramamine)
- diphenhydramine (Benadryl) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) synthetic tertiary ammonium analogues of atropine tricyclic antidepressants |
- amitriptyline (Elavil)
|
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) synthetic tertiary ammonium analogues of atropine antipsychotics |
- haloperidol (Haldol)
- chlorpromazine (Thorazine) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for fundoscopic exam |
- tropicamide (Mydriacil)
- cyclopentolate (Cyclogil) - Atropine sulfate (Isopto Atropine) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for IBS and peptic ulcer |
- glycopyrrolate (Robinul) 4o
- dicyclomine (Bentyl) 3o - hyoscyamine (Levsin) 3o - hyoscyamine + phenobarbital (Donnatal) 3o - clidinium + chlordiazepoxide (Librax) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for traveler's diarrhea & other mild GI tract hypomotility |
atropine + diphenoxylate (Lomotil)
|
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) NO antimuscarinic agents, just opioid for traveler's diarrhea & other mild GI tract hypomotility |
- loperamide (Imodium A-D) OTC
- loperamide (Imodium) Rx |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for overactive bladder and urge incontinence |
- oxybutynin (Ditropan)
- tolterodine (Detrol LA) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) as adjunct to surgical anesthesia |
- no longer used
- replaced by halothane, enflurane or isoflurane |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for asthma & COPD |
- ipratropium (Atrovent)
- tiotropium (Spiriva) - ipratropium + albuterol (Combivent) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) adjunct for Parkinson's Disease |
- benztropine (Cogentin)
- trihexyphenidyl (Artane) - diphenhydramine (Benadryl inj.) |
|
CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) antimuscarinic agents (Muscarinic Receptor Blockers) for motion sickness |
scopolamine (Transderm Scop)- a dermal patch
|
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CHOLINOCEPTOR-BLOCKING AGENTS
(Anticholinergics) Non - antimuscarinic agent (Muscarinic Receptor Blockers) antihistamines for motion sickness with antimuscarinic effects |
- dimenhydrinate (Dramamine)
- meclizine (Antivert) |
|
for poisoning from cholinomimetic agent
|
- atropine
|
|
Antidotes for insecticides and humanocides
|
- atropine (Isopto Atropine)
- pralidoxime (Protopam, 2-PAM) |