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48 Cards in this Set

  • Front
  • Back

Metacholine

Muscarinic agonist (bronchoconstriction)



Pilocarpine

Muscarinic agonist (pupillary constriction)

Atropine

Muscarinic antagonist

Tolterodine

Muscarinic antagonist (urinary incontinence)

Botulinum Toxin

Prevents AcH release

Neostigmine

Cholinesterase inhibitor

Physostigmine

Cholinesterase inhibitor (myasthenia gravis)

Pyridostigmine

Cholinesterase inhbiitor

Sevin

Cholinesterase inhibitor

Ephedrine

Increases NE release from postsynaptic terminal

Epineprine

(a1, a2, b1, b2) Low dose: b2>a1, high dose: a1>b2

Norepinephrine

(a1, a2, b1) Inc CO and TPR

Isoproterenol

(b1, b2) Inc CO dec TPR

Dopamine

(a1, a2, b1, b2), a1>b2, net ^ TPR

Dobutamine

(a1,a2,b1,b2), a1 = b2, net <--> TPR

Phenylephrine

a1 agonist

Albuterol

b2 agonist

Methyldopa

Central a2 agonist (pregnancy hypertension)

Clonidine

Central a2 agonist (sedative)

Dexmedetomidine

A2 agonist (muscle relaxant)

Reserpine

Inhibits NE uptake, depletes NE, dec TPR and Force

Prazosin

Peripheral a1 blocker (HTN, BPH)

Doxazocin

Peripheral a1 blocker (HTN, BPH)

Tamulosin

Peripheral a1 blocker (HTN, BPH)

Phenoxybenzamine

Nonselective alpha blockade (pheochromocytoma)

phentolomine

Nonselective alpha blockade (pheochromocytoma)

Labetalol

Beta1, 2 with alpha 1 blocker

Carvedilol

Beta1, 2 with alpha 1 blocker

Atenolol

B1 blocker (renal)

Metoprolol

B1 blocker

Esmolol

B1 blocker

Propanolol

nonselective beta blocker

Nadolol

Nonselective beta blocker

Catopril

Ace inhibitor

Lisinopril

Ace inhibitor

Losartan

ARB

Aliskiren

Renin inhibitor

Nitroprusside

Arterial + venous dilater

Hydralazine

Direct arterial vasodilator (drug induced lupus)

Adenosine

Coronary vasodilator, slows heart rate and conduction, bronchoconstriction

Neseritide

Recombinant BNP

Sildenafil

PD5 inhibitor (PAH)

Verapamil

Central and peripheral Ca2+ channel blocker

Diltiazem

Central and peripheral Ca2+ channel blocker

Nifedipine

Peripheral Ca2+ channel blocker

NTG

Vasodilation (increased cGMP)

Isosorbide dinitrite

Vasodilation (increased cGMP)

Isosorbide mononitrate

Vasodilation (increased cGMP)