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38 Cards in this Set

  • Front
  • Back
Nonspecific sympathetic agonist
Epinephrine – bronchodilation, local vasoconstriction, hypotension, shock, allergy
α receptor agonist
Methylphenidate (Ritalin) – for ADHD
Amphetamine (Adderall) – for ADHD
Presynaptic α2 agonist (inverse agonist)
Clondine (Catapres) - HTN
β2 Agonist
Albuterol (Proventil) – bronchodilator
α blocker
Terazosin (Hytrin) - α1- benign prostatic hyperplasia, HTN, CHF, post MI, arrhythmias, IHD
Tamsulosin (Flomax) - α1A and α1D - benign prostatic hyperplasia
β blocker
Metoprolol (Toprol) – selective for β1-HTN, CHF, post MI, arrhythmias, IHD
Propranolol (Inderal) – nonselective-HTN, CHF, post MI, arrhythmias, IHD
Carvedilol (Coreg) - β1 and α1, HTN-CHF, post MI, arrhythmias, IHD
Cholinesterase inhibitor
Tacrine (Cognex) – Alzheimer’s, Parkinson’s w/ dementia
Anticholinergic
Ipratropium(Atrovent) – bronchodilation
Tiotropium(Spiriva) - bronchodilation
Tolterodine (Detrol) - dysuria
Darifenacin (Enablex) – dysuria
muscarinic antagonist & short acting beta 2 adrenergic agonist
Ipratropium /albuterol (Combivent)
Partial nicotine agonist
Varenicline (Chantix)
Typical Antipsychotic
Haloperidol (Haldol) – dopamine antagonist - Schizophrenia
Atypical Antipsychotic
Clozapine (Clozaril) - Schizophrenia
Olanzapine (Zyprexa) - Schizophrenia
Risperidone (Risperdal) - Schizophrenia
Quetiapine (Seroquel) - Schizophrenia
Ziprasidone (Geodon) - Schizophrenia
Aripiprazole (Abilify) – Schizophrenia, bipolar disorder, depression
Dopamine procursors
Sinemet (Carbidopa/Levodopa) - Parkinson’s
Dopamine receptor agonist
Ropinirole (Requip)- Parkinson’s
dopamine metabolism inhibitor
Entacapone (Comtan) - inhibits COMT - Parkinson’s
Rasagiline (Azilect) – inhibits MAO-B - Parkinson’s
MAOI
Selegiline (Emsam) –inhibits serotonin degredation - depression
TCA
Amitriptyline (Elavil) – NE and serotonin reuptake inhibitors – depression, chronic pain
Benzodiazepam
Diazepam (Valium) - Antianxiety, sedative-hypnotic, amnesic, anticonvulsant, skeletal muscle relaxant, alcohol withdrawal
Benzo receptor antagonist (antidote)
Flumazenil (Romazicon) – for benzo overdose
GABA receptor modulator
Zolpidem (Ambien) central sites on benzo receptor - insomnia
*Eszopiclone (Lunesta) – sites close to benzo receptor - insomnia
SNRIs
Venlafaxine (Effexor) - depression
Duloxetine (Cymbalta) – depression, neuropathic pain
Bupropion (Wellbutrin) – depression, nicotine withdrawal
SSRIs
Fluoxetine (Prozac) – depression
*Sertraline (Zoloft)
*Paroxetine (Paxil)
*Citalopram (Celexa)
*Escitalopram (Lexapro)
SARI
Trazodone (Desyrel) – depression w/ sleep disturbances
GABA b Receptor Agonist
Baclofen - MS, Spinal cord injuries, Pts who have had strokes, spasticity, flexor spasm and concomitant pain, muscular rigidity
Calcium channel inhibitor
Gabapentin (Neurontin) – seizures, pain
Pregabalin (Lyrica)
Antimania
Lithium carbonate – alters sodium transport – mania, depression
Sodium channel inhibitor
Carbamazepine (Tegretol) - Seizure disorders, bi-polar, neuralgias, migraines
*Phenytoin (Dilantin)
*Valporic Acid (Depakote)
*Topiramate (Topamax)
Anticonvulsant/mood stabilizer
Lamotrigine (Lamictal)
Levetiracetam (Keppra)
NMDA receptor blocker
Memantine (Namenda) - Alzheimer’s
Amantadine - Parkinson’s disease
NSAID
Ibuprofen
Aspirin
Celebrex – COX-2
Acetaminophen
Tylenol
Opioid
Codeine
Hydrocodone
Non-opioid centrally acting analgesic
Tramadol
Muscle relaxant – CNS depressant
Tizanidine (Zanaflex) – α2 inverse agonist
Cyclobenzaprine (Flexeril)
Metaxalone (Skelaxin)
Steroid
Steroids – anti-inflammatory
General anesthetic
Ketamine Patch
Topical analgesic
Capsaicin
Lidoderm
Serotonin 5-HT 1B/1D receptor agonists
Sumatriptan (Imitrex) - migraine