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22 Cards in this Set
- Front
- Back
3A4 substrates
antiarrythmics (3) |
amiodarone, quinidine, lidocaine
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3A4 substrates
antidepressants (4) |
TCAs, fluoxetine, sertraline, nefazadone
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3A4 substrates
allergy meds (2) |
loratadine, terfenadine
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3A4 substrates
Benzos (3) |
alprazolam, midzolam, triazolam
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3A4 substrates
CCBs |
nifedipine, verapamil, diltiazem
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3A4 substrates
antiepileptic |
CBZ
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3A4 substrates
antilipidemic |
statins (except pravastatin)
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3A4 inhibitors (7)
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Ketoconazole, itraconazole, clarithromycin, erythromycin, nefazodone, ritonavir, grapefruit juice
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3A4 inducers (5)
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CBZ, phenytoin, phenobarbitol, rifampin, rifabutin
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2C9 substrates (7)
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warfarin, phenytoin, nsaids, tolbutamide, VPA, glipizide, glyburide
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2C9 inhibitors (3, all weak)
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fluvoxamine, fluoxetine, norfluoxetine
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2C19 substrates (6)
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PPI's, phenytoin, diazepam, citalopram, amitriptyline, imipramine
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2C19 inhibitors (3)
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fluvoxamine > fluoxetine, sertraline
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1A2 substrates (8)
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caffeine, theophylline, clozapine, haldol, TCAs, phenacetin, tacrine, cipro
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1A2 inhibitors (2)
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fluvoxamine (potent), FQs
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1A2 inducers (2)
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smoking, charbroiled food
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2D6 substrates
analgesics (3) |
DM, codeine, tramadol
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2D6 substrates
antidepressants (4) |
paroxetine, fluoxetine, venlafaxine, desipramine
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2D6 substrates
antiarrythmics (2) |
propafenone, fleicanide
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2D6 substrates
antipsychotics (2) |
risperidone, thioridazine
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2D6 inhibitors (8)
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quinidine, paroxetine, fluoxetine, norfluoxetine, haldol, fluphenazine, darvocet, buproprion
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2D6 inducers (2)
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rifampin, cbz
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