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18 Cards in this Set
- Front
- Back
Erythromycin
|
(Macrolide - 50S)
DOC: Mycoplasma pneumonia, legionella infections, diptheria infections. Tox: dec. P450 |
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Clarithromycin
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(Macrolide - 50S)
TX: H. influenzae, Mycoplasma avium complex, H. Pylori Tox: dec. P450 |
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Azithromycin
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(Macrolide - 50S)
TX: Mycoplasma avium complex, toxoplasmosis encephalitis, chlamydia trachomatis |
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Clindamycin
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Lincosamide (50S)
-DOC: Anaerobes -Tox: pseudomembranous enterocolitis |
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Chloramphenicol
|
50S
-DOC: salmonella typhosa -Tox: "GRAY BABY SYNDROME", aplastic anemia, pancytopenia, transient bone marrow depression |
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Tetracyclines
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(30S)
DOC: Cholera, rickettsia, coxiella, relapsing fever, chalamydial diseases, ROCKY MOUNTAIN SPOTTED FEVER, rickettsiae, mycoplasma, lymphogranuloma Tox: Discolor/damage teeth, bones, nails b/c chelation of Ca, Mg, Al; Fanconi syndrome |
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Aminoglycosides, general
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(30S)
-blocks initiation -promotes misreading -poor GI absorption -excreted unchanged in urine -Concentration dependent - administer one large dose daily Tox: Ototox, nephrotox, curare-like syndrome, electroylte imbalance |
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Streptomycin
|
Aminoglycoside (30S)
-Used IN COMBO for tx of TB, strep faecalis, endocarditis, plague |
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Neomycin
|
Aminoglycoside (30S)
-VERY toxic -topical use or bowel sterilization ONLY -for G+/G- including mycobacteria |
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Kanamycin
|
Aminoglycoside (30S)
-very high misreading of mRNA -very toxic -seldomly used |
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Gentamicin
|
Aminoglycoside (30S)
-active against many G- (P-PEck) |
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Tobramycin
|
New Aminoglycoside (30S)
-for bacteremia by G- Bacilli |
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Amikacin
|
New Aminoglycoside (30S)
-for resistent strains |
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Netilmicin
|
New Aminoglycoside (30S)
-against G- bacilli -less toxic |
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Viomycin
|
New Aminoglycoside (30S)
-second line drug for TB |
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Spectinomycin
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AminoCYCLITOL (30S)
-only for acute gonococcal urethritis, proctitis, cervicitis -LOW renal tox -NO ototoxicity |
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Streptogramins A+B
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Quinupristin and Dalfopristin
-inhibit 50S, bactericidal -for resistant bacteria -SE: arthralgia-myalgia, inc. P450 |
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Oxazoladinones
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Linezolid
-for G+ multiple drug resistant -TOX: GI, headache, thrombocytopenia, MAOI |