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65 Cards in this Set

  • Front
  • Back
Acetylcholine
Cholinomimetic
-Stimulates Muscarinic & Nicotinic receptor
Behanechol
Cholinomimetic
-ONLY muscarinic
-Long acting
Carbachol
Cholinomimetic
-BOTH muscarinic & nicotinic
-Long acting
Pilocarpine
Cholinomimetic
Muscarinic
Cevimeline
Cholinomimetic
M3 selective
Edrophonium
Cholinomimetic
ChE inhibitor
Brief duration
Ambenonim
Cholinomimetic
ChE inhibitor
Brief duration (hrs)
Neostigmine
Cholinomimetic
ChE inhibitor
Physostigmine
Cholinomimetic
ChE inhibitor
Crosses BBB
Pyridostigmine
Cholinomimetic
ChE inhibitor
Isoflurophate
Cholinomimetic
ChE inhibitor
Organophosphate
Non-competitive (Slow reversal)
Echothiophate
Cholinomimetic
ChE inhibitor
Organophoshpate
non-competitive (slow reversal)
Tacrine
Cholinomimetic
ChE inhibitor
not used widely
Donepezil
Cholinomimetic
ChE inhibitor
more selective to CNS
Alzheimers drug w/ long duration
Rivastigmine
Cholinomimetic
ChE inhibitor
Alzheimer drug
Galantamine
Cholinomimetic
ChE inhibitor
Alzheimer drug
Atropine
Antimuscarinic
Selective for Muscarinic receptors
Long acting
Crosses BBB only @ high dose
Scopolamine
Antimuscarinic
Selective for Muscarinic receptors
crosses BBB
Tropicamide
Antimuscarinic
Ophthalmological exam
short acting
Use w/ pheynlephrine
Pralidoxime
Antimuscarinic
ChE reactivator (w/in 24 hrs)
Tolterodine
Antimuscarinic
M3 selective
Relaxes detrusor tightens sphincter
Urinary urgency & freq
Solifenacin
Antimuscarinic
M3 antagonist, some muscarinc receptors
Ipratropium
Antimuscarinic
noselective
For asthma, COPD
Tiotroprium
Antimuscarinic
Selective
longer duration 24 hrs
Succinylcholine
Neuromuscular Blocker
Nicotinic receptor
Depolarizing
Atarcrium
Neuromuscular Blocker
nicotinic receptor
Non-depolarizing
Cisatracurium
Neuromuscular Blocker
Nicotinic receptor
Non-depolarizing
Pancuronium
Neuromuscular Blocker
Nicotinic
Non-depolarizing
Rocuronium
Neuromusclular Blocker
Nicotinic
Nondepolarizing
Vecuronium
Neuromusclular Blocker
Nicotinic
Nondepolarizing
Nicotine
Depolarizing Ganglion Blocker
Epinephrine
Catecholamine
BOTH alpha & beta
Norepinephrine
Catecholamine
Alpha & Beta w/ MORE B-1
Dopamine
Catecholamine
D1 & D2 > B > a
Phenylephrine
Sympathomietic
Alpha 1 Agonist
Midodrine
Sympathomietic
Alpha-1 Agonists
Brimonidine
Sympathomietic
Alpha-2 Agonist
Glaucoma
Oxymetazoline
Sympathomimetic
Alpha-1 agonist
Isoproterenol
Sympathomietic
Beta Agonist Non-selective
Albuterol
Sympathomietic
B-2 selective Agonist
Levalbuterol
Sympathomietic
B-2 selective Agonist
Terbutaline
Sympathomietic
B-2 selective Agonist
Formoterol
Sympathomietic
B-2 selective Agonist
Dobutamine
Sympathomietic
Mixed Agonist (a & B)
B-1 predominate
Ephedrine
Sympathomietic
Mixed Agonist
Pseudoephedrine
Sympathomietic
Mixed Agonist
Fenoldopam
Sympathomietic
D-1 Receptor Agonist
Methylphenidate
Sympathomietic
Indirect agonist: blocks reuptake of catecholamines
Cocaine
Sympathomietic
Indirect Agonists: blocks reuptake of catecholamines
Local anesthetic effect (non-adrenergic)
Tyramine
Sympathomietic
By-product of tyrosine metabolism
Releases NE from storage vesicles
Phenoxybenzamine
Antiadrenergic
Mixed alpha antagonist
Phentolamine
Antiadrenergic
Mixed alpha antagonist
Doxazosin
Antiadrenergic
a-1 antagonist
Terazosin
Antiadrenergic
a-1 antagonist
Tamsulosin
Antiadrenergic
a-1 antagonist
Propranolol
Antiadrenergic
Non-selective beta antagonist
Nadolol
Antiadrenergic
B-1 & B-2 antagonist
Timolol
Antiadrenergic
Non-selective Beta Antagonist
Metoprolol
Antiadrenergic
B-1 selective antagonist
Atenolol
Antiadrenergic
B-1 selective antagonist
Esmolol
Antiadrenergic
B-1 Selective antagonist
Betaxolol
Antiadrenergic
B-1 seclective for glaucoma
Carvedilol
Antiadrenergic
Mixed a-1 & B antagonist
Clonidine
Antiadrenergic
a-2 agonists
Reserpine
Antiadrenergic
Deplete NE stores