Use LEFT and RIGHT arrow keys to navigate between flashcards;
Use UP and DOWN arrow keys to flip the card;
H to show hint;
A reads text to speech;
65 Cards in this Set
- Front
- Back
Acetylcholine
|
Cholinomimetic
-Stimulates Muscarinic & Nicotinic receptor |
|
Behanechol
|
Cholinomimetic
-ONLY muscarinic -Long acting |
|
Carbachol
|
Cholinomimetic
-BOTH muscarinic & nicotinic -Long acting |
|
Pilocarpine
|
Cholinomimetic
Muscarinic |
|
Cevimeline
|
Cholinomimetic
M3 selective |
|
Edrophonium
|
Cholinomimetic
ChE inhibitor Brief duration |
|
Ambenonim
|
Cholinomimetic
ChE inhibitor Brief duration (hrs) |
|
Neostigmine
|
Cholinomimetic
ChE inhibitor |
|
Physostigmine
|
Cholinomimetic
ChE inhibitor Crosses BBB |
|
Pyridostigmine
|
Cholinomimetic
ChE inhibitor |
|
Isoflurophate
|
Cholinomimetic
ChE inhibitor Organophosphate Non-competitive (Slow reversal) |
|
Echothiophate
|
Cholinomimetic
ChE inhibitor Organophoshpate non-competitive (slow reversal) |
|
Tacrine
|
Cholinomimetic
ChE inhibitor not used widely |
|
Donepezil
|
Cholinomimetic
ChE inhibitor more selective to CNS Alzheimers drug w/ long duration |
|
Rivastigmine
|
Cholinomimetic
ChE inhibitor Alzheimer drug |
|
Galantamine
|
Cholinomimetic
ChE inhibitor Alzheimer drug |
|
Atropine
|
Antimuscarinic
Selective for Muscarinic receptors Long acting Crosses BBB only @ high dose |
|
Scopolamine
|
Antimuscarinic
Selective for Muscarinic receptors crosses BBB |
|
Tropicamide
|
Antimuscarinic
Ophthalmological exam short acting Use w/ pheynlephrine |
|
Pralidoxime
|
Antimuscarinic
ChE reactivator (w/in 24 hrs) |
|
Tolterodine
|
Antimuscarinic
M3 selective Relaxes detrusor tightens sphincter Urinary urgency & freq |
|
Solifenacin
|
Antimuscarinic
M3 antagonist, some muscarinc receptors |
|
Ipratropium
|
Antimuscarinic
noselective For asthma, COPD |
|
Tiotroprium
|
Antimuscarinic
Selective longer duration 24 hrs |
|
Succinylcholine
|
Neuromuscular Blocker
Nicotinic receptor Depolarizing |
|
Atarcrium
|
Neuromuscular Blocker
nicotinic receptor Non-depolarizing |
|
Cisatracurium
|
Neuromuscular Blocker
Nicotinic receptor Non-depolarizing |
|
Pancuronium
|
Neuromuscular Blocker
Nicotinic Non-depolarizing |
|
Rocuronium
|
Neuromusclular Blocker
Nicotinic Nondepolarizing |
|
Vecuronium
|
Neuromusclular Blocker
Nicotinic Nondepolarizing |
|
Nicotine
|
Depolarizing Ganglion Blocker
|
|
Epinephrine
|
Catecholamine
BOTH alpha & beta |
|
Norepinephrine
|
Catecholamine
Alpha & Beta w/ MORE B-1 |
|
Dopamine
|
Catecholamine
D1 & D2 > B > a |
|
Phenylephrine
|
Sympathomietic
Alpha 1 Agonist |
|
Midodrine
|
Sympathomietic
Alpha-1 Agonists |
|
Brimonidine
|
Sympathomietic
Alpha-2 Agonist Glaucoma |
|
Oxymetazoline
|
Sympathomimetic
Alpha-1 agonist |
|
Isoproterenol
|
Sympathomietic
Beta Agonist Non-selective |
|
Albuterol
|
Sympathomietic
B-2 selective Agonist |
|
Levalbuterol
|
Sympathomietic
B-2 selective Agonist |
|
Terbutaline
|
Sympathomietic
B-2 selective Agonist |
|
Formoterol
|
Sympathomietic
B-2 selective Agonist |
|
Dobutamine
|
Sympathomietic
Mixed Agonist (a & B) B-1 predominate |
|
Ephedrine
|
Sympathomietic
Mixed Agonist |
|
Pseudoephedrine
|
Sympathomietic
Mixed Agonist |
|
Fenoldopam
|
Sympathomietic
D-1 Receptor Agonist |
|
Methylphenidate
|
Sympathomietic
Indirect agonist: blocks reuptake of catecholamines |
|
Cocaine
|
Sympathomietic
Indirect Agonists: blocks reuptake of catecholamines Local anesthetic effect (non-adrenergic) |
|
Tyramine
|
Sympathomietic
By-product of tyrosine metabolism Releases NE from storage vesicles |
|
Phenoxybenzamine
|
Antiadrenergic
Mixed alpha antagonist |
|
Phentolamine
|
Antiadrenergic
Mixed alpha antagonist |
|
Doxazosin
|
Antiadrenergic
a-1 antagonist |
|
Terazosin
|
Antiadrenergic
a-1 antagonist |
|
Tamsulosin
|
Antiadrenergic
a-1 antagonist |
|
Propranolol
|
Antiadrenergic
Non-selective beta antagonist |
|
Nadolol
|
Antiadrenergic
B-1 & B-2 antagonist |
|
Timolol
|
Antiadrenergic
Non-selective Beta Antagonist |
|
Metoprolol
|
Antiadrenergic
B-1 selective antagonist |
|
Atenolol
|
Antiadrenergic
B-1 selective antagonist |
|
Esmolol
|
Antiadrenergic
B-1 Selective antagonist |
|
Betaxolol
|
Antiadrenergic
B-1 seclective for glaucoma |
|
Carvedilol
|
Antiadrenergic
Mixed a-1 & B antagonist |
|
Clonidine
|
Antiadrenergic
a-2 agonists |
|
Reserpine
|
Antiadrenergic
Deplete NE stores |