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26 Cards in this Set
- Front
- Back
TCA's
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CYP2D6
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FLUOXETINE
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METABOLIZED BY CYP2D6
DECENT INHIBITOR OF CYP2C9 POTENT INHIBITOR OF CYP2D6 |
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FLUVOXAMINE
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METABOLIZED BY CYP2D6, 1A2
INHIBITS CYP3A4 |
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MIRTAZAPINE
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METABOLIZED BT CYP2D6
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PAROXETINE
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METABOLIZED BT CYP2D6
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SERTRALINE
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METABOLIZED BT CYP2D6?
ALSO 2C9/2C19 |
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TRAZODONE
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METABOLIZED BT CYP2D6
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VENLAFAXINE
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METABOLIZED BT CYP2D6
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CITALOPRAM
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METABOLIZED BY CYP3A4
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NEFAZODONE
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INHIBITS 3A4-INTERACTS WITH PROTEASE INHIBITORS
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BUPROPRION
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METABOLIZES CYP 2B6
INHIBITS CYP2D6 |
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MOST BENZODIAZEPINES
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METABOLIZED BY CYP3A4
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BENZODIAZEPINES THAT ARE NOT METABOLIZED BY CYP P450
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LORAZEPAM, OXAZEPAM, TEMAZEPAM
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DIAZEPAM
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METABOLIZED BY CYP2C9 AND 2C19
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MOST TYPICAL NEUROLEPTICS
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METABOLIZED BY CYP2D6
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TYPICAL NEUROLEPTIC METABOLIZED BY CYP3A4
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PIMOZIDE
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CLOZAPINE
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CYP1A2
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OLANZAPINE
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METABOLIZED BY CYP1A2
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RISPERIDONE
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CYP2D6
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QUETIAPINE
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METABOLIZED BY CYP3A4
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ZIPRASIDONE
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METABOLIZED BY CYP3A4
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CARBAMEZAPINE
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POTENT INDUCER OF CYP3A4
(ALSO METABOLIZED BY THE SAME; HENCE IT INDUCES ITS OWN METABOLISM, IE CHEWS ITSELF UP). |
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PREFERRED ANTIDEPRESSANTS FOR HAART PATIENTS
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REMERON
EFFEXOR CELEXA LEXAPRO |
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CAUTION THESE ANTIDEPRESSANTS ARE RELATIVELY CONTRAINDICATED IN HIV HAART PATIENTS
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WELLBUTRIN
PROZAC TCAS |
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HAART POTENT INHIBITOR OF CYP P450 2B6, 2D6, AND 3A4
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RITONAVIR
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EFAVIRENZ
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POTENT INHIBITOR OF 2B6
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