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106 Cards in this Set
- Front
- Back
Norepinephrine
|
α adrenergic agonist
|
|
Phenylephrine
|
α adrenergic agonist
(α1) |
|
Methoxamine
|
α adrenergic agonist
(α1) |
|
Metaraminol
|
α adrenergic agonist
(α1 >> β1) |
|
Tetrahydrozoline
|
α adrenergic agonist
(α1) |
|
Clonidine
|
α adrenergic agonist
anti-hypertension --> central nervious system |
|
Phentolamine
|
α adrenergic antagonist
|
|
Tolazoline
|
α adrenergic antagonist
|
|
Phenoxybenzamine
|
α adrenergic antagonist
|
|
Prazosin
|
α adrenergic antagonist
anti-hypertension --> adrenergic receptor blockade |
|
Isoproterenol
|
β adrenergic agonist
anti-asthma |
|
Dobutamine
|
β adrenergic agonist
(β1 >> β2) treatment for congestive heart failure --> direct cardiotonic agent |
|
Terbutaline
|
β adrenergic agonist
(β2 >> β1) |
|
Albuterol
|
β adrenergic agonist
(β2 >> β1) anti-asthma |
|
Metaproterenol
|
β adrenergic agonist
(β2 >> β1) |
|
Propanolol
|
β adrenergic antagonist
treatment for congestive heart failure antiarrhythmia (class II) --> β blocker antianginal anti-hypertension |
|
Metoprolol
|
β adrenergic antagonist
anti-hypertension |
|
Nadolol
|
β adrenergic antagonist
|
|
Timolol
|
β adrenergic antagonist
anti-hypertension |
|
Epinephrine
|
α & β adrenergic agonist
antihistamine (not a receptor antagonist) antiasthma |
|
Ephedrine
|
α & β adrenergic agonist
(β > α) |
|
Dopamine
|
α & β adrenergic agonist
|
|
Amphetamine
|
α & β adrenergic agonist
|
|
Cocaine
|
affects adrenergic neurotransmitter metabolism
|
|
Tyramine
|
affects adrenergic neurotransmitter metabolism
|
|
Reserpine
|
affects adrenergic neurotransmitter metabolism
anti-hypertension --> central nervous system anti-hypertension --> neurotransmitter depletion |
|
Guanethidine
|
affects adrenergic neurotransmitter metabolism
anti-hypertension --> neuronal blockade |
|
α-methyldopa
|
affects adrenergic neurotransmitter metabolism
anti-hypertension --> central nervous system |
|
Pilocarpine
|
muscarinic agonist
|
|
Bethanecol
|
muscarinic agonist
|
|
Carbachol
|
muscarinic agonist
|
|
Atropine
|
muscarinic antagonist
anti-asthma |
|
Scopolamine
|
muscarinic antagonist
|
|
Succinylcholine
|
cholinergic depolarizing agent
|
|
Tubocurarine
|
competitive cholinergic blocker
|
|
Pancuronium
|
competitive cholinergic blocker
|
|
Vecuronium
|
competitive cholinergic blocker
|
|
Physostigmine
|
anticholinesterase
|
|
Neostigmine
|
anticholinesterase
|
|
Pyridostigmine
|
anticholinesterase
|
|
Edrophonium
|
anticholinesterase
|
|
Isoflurophate (DFP)
|
anticholinesterase
|
|
Pralidoxime (2-PAM)
|
anticholinesterase
|
|
Mannitol
|
osmotic diuretic
|
|
Acetazolamide
|
diuretic --> carbonic anhydrase inhibitor
|
|
Hydrochlorothiazide
|
anti-hypertension --> thiazide diuretic
|
|
Furosemide
|
anti-hypertension --> loop diuretic
|
|
Ethacrynic acid
|
anti-hypertension --> loop diuretic
|
|
Torsemide
|
anti-hypertension --> loop diuretic
|
|
Triamterine
|
anti-hypertension --> K+ sparing diuretic
|
|
Spironolactone
|
anti-hypertension --> K+ sparing diuretic
|
|
Amiloride
|
anti-hypertension --> K+ sparing diuretic
|
|
Desmopressin
|
anti-diuretic
|
|
Verapamil
|
anti-arrhythmia (class IV) --> calcium channel blocker
|
|
Diltiazem
|
calcium channel blocker
|
|
Nifedipine
|
anti-hypertension --> calcium channel blocker
antianginal --> calcium channel blocker |
|
Amlodipine
|
calcium channel blocker
|
|
Captopril
|
treatment for congestive heart failure --> ACE inhibitor
anti-hypertension --> ACE inhibitor |
|
Enalapril (prodrug)
|
treatment for congestive heart failure --> ACE inhibitor
anti-hypertension --> ACE inhibitor |
|
Enalaprilat (active drug)
|
treatment for congestive heart failure --> ACE inhibitor
anti-hypertension --> ACE inhibitor |
|
Lisinopril
|
treatment for congestive heart failure --> ACE inhibitor
anti-hypertension --> ACE inhibitor |
|
Benazepril
|
treatment for congestive heart failure --> ACE inhibitor
anti-hypertension --> ACE inhibitor |
|
Losartan
|
anti-hypertension --> angiotensin II receptor antagonist
|
|
Digoxin
|
treatment for congestive heart failure --> cardiac glycoside
|
|
Digitoxin
|
treatment for congestive heart failure --> cardiac glycoside
antiarrhythmia |
|
Amrinone
|
treatment for congestive heart failure --> PDE inhibitor
|
|
Milrinone
|
treatment for congestive heart failure --> PDE inhibitor
|
|
Sotolol
|
treatment for congestive heart failure --> β blocker
antiarrhytmia (class II) --> β blocker |
|
Carvedilol
|
treatment for congestive heart failure --> α & β blocker
anti-hypertension --> adrenergic receptor blockade |
|
Neseritide
|
treatment for congestive heart failure
|
|
Quinidine
|
antiarrhythmia (class I) --> sodium channel blocker
|
|
Procainamide
|
antiarrhythmia (class I) --> sodium channel blocker
|
|
Lidocaine
|
antiarrhythmia (class I) --> sodium channel blocker
|
|
Phenytoin
|
antiarrhythmia (class I) --> sodium channel blocker
|
|
Esmolol
|
antiarrhythmia (class II) --> β blocker
|
|
Acebutolol
|
antiarrhythmia (class II) --> β blocker
|
|
Bretyllium
|
antiarrhythmia (class III) --> AP prolongation
|
|
Amiodarone
|
antiarrhythmia (class III) --> AP prolongation
|
|
Adenosine
|
antiarrhythmia
|
|
Nitroglycerine
|
antianginal (no precursors)
|
|
Isosorbide dinitrate
|
antianginal (no precursors)
|
|
Hydralazine
|
anti-hypertension --> vasodilator
|
|
Minoxidil
|
anti-hypertension --> vasodilator
|
|
Nitroprusside
|
anti-hypertension --> vasodilator
|
|
Pindolol
|
anti-hypertension --> adrenergic receptor blockade
|
|
Diphenhydramine (ex. Benadryl)
|
antihistamine --> 1st generation H1 antagonist
|
|
Chlorpheniramine (ex. Chlor-trimetron)
|
antihistamine --> 1st generation H1 antagonist
|
|
Promethazine (ex. Phenergan)
|
antihistamine --> 1st generation H1 antagonist
antiemetic and motion sickness --> antihistamine |
|
Meclizine (ex. Bonine)
|
antiemetic and motion sickness --> antihistamine
|
|
Dimenhydrinate (ex. Dramamine)
|
antiemetic and motion sickness --> antihistamine
|
|
Loratadine
|
antihistamine --> 2nd generation H1 antagonist
|
|
Fexofenadine
|
antihistamine --> 2nd generation H1 antagonist
|
|
Cimetidine
|
antihistamine --> H2 antagonist
|
|
Famotidine
|
antihistamine --> H2 antagonist
|
|
Ranitidine
|
antihistamine --> H2 antagonist
|
|
Cromolyn
|
antihistamine (not a receptor antagonist)
antiasthma |
|
Levalbuterol
|
antiasthma --> β2 agonist
|
|
Formoterol
|
antiasthma --> β2 agonist
|
|
Salmeterol
|
antiasthma --> β2 agonist
|
|
Beclomethasone
|
antiasthma --> inhaled corticosteroid
|
|
Flunisolide
|
antiasthma --> inhaled corticosteroid
|
|
Montelukast
|
antiasthma --> leukotriene antagonist
|
|
Zafirlukast
|
antiasthma --> leukotriene antagonist
|
|
Theophyline
|
antiasthma
|
|
Ipratropium
|
antiasthma
|
|
Zileuton
|
antiasthma
|