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6 Cards in this Set
- Front
- Back
Fentanyl
mechanism of action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Safe Metabolism: liver; CYP450: 3A4 substrate Excretion: urine (10-25% unchanged); Half-life: 3.7h DEA/FDA: Schedule II Class: Induction/Maintenance |
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Alfentanil
Mechanism Of Action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Probably Safe Metabolism: liver extensively; CYP450: 3A4 substrate Excretion: urine (<1% unchanged); Half-life: 1.5-1.8h DEA/FDA: Schedule II Class: Induction/Maintenance, Narcotics |
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Sufentanil
Mechanism Of Action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Safety Unknown Metabolism: liver, small intestine; CYP450: 3A4 substrate Excretion: urine (<2% unchanged); Half-life: 2.7h DEA/FDA: Schedule II Class: Narcotics, Induction/Maintenance |
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Remifentanil
Mechanism Of Action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Safety Unknown Metabolism: other Excretion: urine DEA/FDA: Schedule II Class: Narcotics, Induction/Maintenance |
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Meperidine
Mechanism Of Action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Safety Unknown Metabolism: liver; CYP450: 2D6 substrate; Info: active metabolite Excretion: urine; Half-life: 2.5-4h (adults), 23h (neonates); 15-30h (normeperidine); Info: active metab. accumulation in renal or hepatic impairment assoc. w/seizures DEA/FDA: Schedule II Class: Narcotics |
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Morphine
Mechanism Of Action |
Mechanism Of Action: binds to various opiate receptors, producing analgesia and sedation (opioid agonist)
Pregnancy: C Lactation: Probably Safe Metabolism: liver Excretion: urine DEA/FDA: Schedule II Class: Narcotics |