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35 Cards in this Set

  • Front
  • Back
Norepinephrine
A1,A2,B1
Epinephrine
A1,A2,B1,B2
Phenylephrine
A1 agonist
Clonidine
A2 agonist
Dobutamine
B1 agonist
Terbutaline
B2 agonist
Albuterol
B2 agonist
metaproterenol
B2 agonist
isoproterenol
B1 and B2 agonist
oxymetazoline
A1 and A2 agonist
ephedrine
mixed-agonist activity
epenphrine +CNS effects
amphetamine
Causes catchecholamine release
dextroamphetamine
methamphetamine
methylphenidate
Causes catchecholamine release
tyramine
Causes catchecholamine release
Phenoxybenzamine
"irreversible" a1-a2 antagonist
phentolamine
non-selective competitive alpha antagonist
tolazoline
non-selective competitive alpha antagonist
prazosin
alpha1 antagonist
doxazosin
alpha1 antagonist
terazosin
alpha1 antagonist
tamsulosin
selective alpha1(a-d) antagonist
-BPH, prostatic hyperplasia treatment
yohimbine
a2 antagonist
Nebivolol
B1 blocker, NO potentiator
timolol
non-selective beta blocker
-glaucoma treatment
propanolol
non-selective beta blocker
labetalol
non-selective beta blocker(partial agonist)
alpha 1 antagonist
carvedilol
non-selective beta blocker
ca entry blocker, alpha 1 antagonist
pindolol
non-selective beta blocker(partial agonist)
gunadrel
adrenergic neuronal blocker
-false transmitter- blocks NE uptake, NE release, and depletes NE as a false transmitter
guanethidine
-adrenergicneuronal blocker
-false transmitter- blocks NE uptake, NE release, and depletes NE as a false transmitter
Reserpine
Adrenergic neuronal blocker
-prevents vesicle uptake of NE
methyldopa
indirect a2 antagonist
a-methyltyrosine
adrenergic neuronal blocker
Neuropeptide Y
non-adrenegic non-cholinergic
-NE constrictor effects
cocaine
prevents reuptake of catcholamines