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35 Cards in this Set
- Front
- Back
Norepinephrine
|
A1,A2,B1
|
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Epinephrine
|
A1,A2,B1,B2
|
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Phenylephrine
|
A1 agonist
|
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Clonidine
|
A2 agonist
|
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Dobutamine
|
B1 agonist
|
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Terbutaline
|
B2 agonist
|
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Albuterol
|
B2 agonist
|
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metaproterenol
|
B2 agonist
|
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isoproterenol
|
B1 and B2 agonist
|
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oxymetazoline
|
A1 and A2 agonist
|
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ephedrine
|
mixed-agonist activity
epenphrine +CNS effects |
|
amphetamine
|
Causes catchecholamine release
|
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dextroamphetamine
methamphetamine methylphenidate |
Causes catchecholamine release
|
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tyramine
|
Causes catchecholamine release
|
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Phenoxybenzamine
|
"irreversible" a1-a2 antagonist
|
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phentolamine
|
non-selective competitive alpha antagonist
|
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tolazoline
|
non-selective competitive alpha antagonist
|
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prazosin
|
alpha1 antagonist
|
|
doxazosin
|
alpha1 antagonist
|
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terazosin
|
alpha1 antagonist
|
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tamsulosin
|
selective alpha1(a-d) antagonist
-BPH, prostatic hyperplasia treatment |
|
yohimbine
|
a2 antagonist
|
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Nebivolol
|
B1 blocker, NO potentiator
|
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timolol
|
non-selective beta blocker
-glaucoma treatment |
|
propanolol
|
non-selective beta blocker
|
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labetalol
|
non-selective beta blocker(partial agonist)
alpha 1 antagonist |
|
carvedilol
|
non-selective beta blocker
ca entry blocker, alpha 1 antagonist |
|
pindolol
|
non-selective beta blocker(partial agonist)
|
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gunadrel
|
adrenergic neuronal blocker
-false transmitter- blocks NE uptake, NE release, and depletes NE as a false transmitter |
|
guanethidine
|
-adrenergicneuronal blocker
-false transmitter- blocks NE uptake, NE release, and depletes NE as a false transmitter |
|
Reserpine
|
Adrenergic neuronal blocker
-prevents vesicle uptake of NE |
|
methyldopa
|
indirect a2 antagonist
|
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a-methyltyrosine
|
adrenergic neuronal blocker
|
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Neuropeptide Y
|
non-adrenegic non-cholinergic
-NE constrictor effects |
|
cocaine
|
prevents reuptake of catcholamines
|