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119 Cards in this Set

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penicillin G
gram (+) [uncomplicated], esp S viridians, S pyogenes EXC S aureus
N meningitidis (-)
N gonorrhoeae (-)
H influenzae (-)
penicillin
penicillin V
Strep (+) [exc S pneumoniae]
L. monocytogenes (+)
C. perfringens (+)
B. anthracis (+)
some gram (-)
penicillin
methicillin
Staph (+) known to make beta-lactamase
penicillin (penicillinase-resistant)
nafcillin
MSSA/MSSE expressing beta-lactamase
penicillin (penicillinase-resistant)
oxacillin
Staph a / e expressing beta-lactamase
penicillin (penicillinase-resistant)
cloxacillin
Staph a / e expressing beta-lactamase
penicillin (penicillinase-resistant)
dicloxacillin
Staph a / e expressing beta-lactamase
penicillin (penicillinase-resistant)
ampicillin
gram (+) and (-) not expressing beta-lactamase
aminopenicillin
amoxicillin
gram (+) and (-) not expressing beta-lactamase
esp H pylori, H. influenzae
aminopenicillin
bacampicillin
gram (+) and (-) not expressing beta-lactamase
aminopenicillin
amoxicillin / clavulanic acid
gram (+) and (-)
aminopenicillin / beta-lactamase inhibitor
ampicillin / sulbactam
gram (+) and (-)
aminopenicillin / beta-lactamase inhibitor
carbenicillin
gram (+) and (-), esp P aeruginosa, P. vulgaris, Enterobacter
exc S aureus
carboxypenicillin (antipseudomonal)
ticarcillin
gram (+) and (-), esp P aeruginosa, P. vulgaris, Enterobacter
exc S aureus
carboxypenicillin (antipseudomonal)
ticarcillin / clavulanic acid
gram (+) and (-), esp P aeruginosa, P. vulgaris, Enterobacter
exc S aureus
carboxypenicillin (antipseudomonal)
mezlocillin
gram (+) and (-), esp (-) like P aeruginosa, K. pneumoniae, wound infection, UTI
ureidopenicillin (antipseudomonal)
piperacillin
gram (+) and (-), esp (-) like P aeruginosa, K. pneumoniae, wound infection, UTI
ureidopenicillin (antipseudomonal)
piperacillin / tazobactam
gram (+) and (-), esp (-) like P aeruginosa, B. fragilis
ureidopenicillin (antipseudomonal)
cefazolin
most gram(+) cocci
okay at E coli, K pneum., P mirabilis
cephalosporin G1
cephalexin
most gram(+) cocci
okay at E coli, K pneum., P mirabilis
cephalosporin G1
cefadroxil
most gram(+) cocci
okay at E coli, K pneum., P mirabilis
cephalosporin G1
cefuroxime (parenteral)
most gram(+) cocci
H. influenzae, N. meningitidis, and S. pneumoniae
cephalosporin G2
cefuroxime axetil
most gram(+) cocci
H. influenzae, N. meningitidis, and S. pneumoniae
cephalosporin G2
cefoxitin
most gram(+) cocci
some g(-): H. influenzae, N. meningitidis, and S. pneumoniae
esp B fragilis!
cephalosporin G2
cefotetin
most gram(+) cocci
some g(-): H. influenzae, N. meningitidis, and S. pneumoniae
esp B fragilis!
cephalosporin G2
cefaclor
most gram(+) cocci
less gram(-), but H influenzae, E coli
cephalosporin G2
cefprozil
some gram(+) eg S pyogenes, S aureus
some (-), eg B fragilis, E coli, H influenzae
cephalosporin G2
loracarbef
most gram(+) cocci
less gram(-), but H influenzae, E coli
carbacephem
cefotaxime
broad spectrum
good gram(-): Enterobacteriaceae, H. influenzae, E. coli, N. gonorrhoeae, N. meningitidis, Klebsiella sp, Serratia marcescens, Salmonella sp., Proteus sp.
cephalosporin G3
ceftizoxime
broad spectrum
good gram(-): Enterobacteriaceae, H. influenzae, E. coli, N. gonorrhoeae, N. meningitidis, Klebsiella, Serratia marcescens, Salmonella, Proteus
cephalosporin G3
ceftriaxone
broad spectrum, esp for meningitis
Enterobacteriacaea, N. gonorrhoeae, N. meningitidis, H. influenzae
Streptococcus
cephalosporin G3
cefixime
broad spectrum, esp for N gonorrhoeae
H. influenzae, Enterobacteriacaea, Salmonella, Shigella
Streptococcus
cephalosporin G3
cefdinir
H influenzae
S pneumoniae; S aureus and S pyogenes in skin
cephalosporin G3
cefpodoxime proxetil
H influenzae
S pneumoniae
S aureus and S pyogenes in skin
cephalosporin G3
cefditoren
H influenzae
S pneumoniae
S aureus and S pyogenes in skin
cephalosporin G3
ceftibuten
S pyogenes
cephalosporin G3
ceftazidime
gram(-), esp Pseudomonas
weaker at gram(+)
cephalosporin G3
cefepime
broad spectrum
distinguished by Staph, Strep
P aeruginosa, Enterobacteriaceae
cephalosporin G4
ceftaroline fosamil
broad spectrum
resistant S aureus, resistant Strep
Pseudomonas, Enterobacteriacaea
cephalosporin G5
imipenem / cilastatin
wide gram(+), potent gram (-) special use
for ESBLs
carbapenem
meropenem
wide gram(+), potent gram (-) special use
for ESBLs
carbapenem
ertapenem
wide gram(+), potent gram (-) special use
for ESBLs
NO P aeruginosa
carbapenem
doripenem
wide gram(+), potent gram (-) special use
for ESBLs
carbapenem
aztreoman
mostly gram(-)
monolactam
vancomycin
gram (+)
lipoglycopeptide
telavancin
gram (+)
lipoglycopeptide
bacitracin
gram (+)
Neisseria (-)
H. influenzae (-)
peptidoglycan transport disruptor
polymixin B
gram(-), incl P aeruginosa
cell membrane disruptor
colistin (polymixin E)
gram (-)
esp P. aeruginosa
cell membrane disruptor
colistimethate (polymixin E)
gram (-)
cell membrane disruptor
daptomycin
gram (+)
incl MRSA, VRE
cell membrane disruptor
streptomycin
gram(-), esp tuberculosis (with another agent), Y pestis
aminoglycoside
gentamicin
gram(-), esp P aeruginosa
Listeria monocytogenes (g+) with another agent
aminoglycoside
tobramycin
gram(-), esp P aeruginosa (with ticarcillin)
aminoglycoside
amikacin
gram(-), broadest spectrum of aminoglycosides
esp Mycobacterium avium, TB
aminoglycoside
neomycin
gram(-) plus E faecalis, S aureus
NO P aeruginosa
aminoglycoside
tetracycline
H pylori, Borrelia, V cholerae, C diff
tetracycline
oxytetracycline
H pylori, Borrelia, V cholerae, C diff
tetracycline
minocycline
treponema pallidum, n gonorrhoeae, Rickettsia, Borrelia
tetracycline
doxycycline
treponema pallidum, n gonorrhoeae, Rickettsia, Borrelia
tetracycline
tigecycline
extended spectrum tcn
glycylcycline (tetracycline)
erythromycin base
gram(+) RTI,
plus Legionella pneumophila (g-)
macrolide
erythromycin estolate
gram(+)RTI ,
plus Legionella pneumophila (g-)
macrolide
erythromycin ethysuccinate
gram(+) RTI,
plus Legionella pneumophila (g-)
macrolide
clarithromycin
gram(+)
some (-) esp H pylori, H influenzae, MAC
macrolide
azithromycin
gram(+) RTI,
some gram(-) esp H influenzae, otitis media
macrolide
fidaxomicin
C. diff ONLY
macrolide
telithromycin
esp MDR S pneumoniae
ketolide (macrolide)
clindamycin
broad spectrum, esp P acnes
P jiroveci
but causes C diff
lincosamide
lincomycin
streptococci (+)
lincosamide
linezolid
gram(+) only, esp MRSA, VISA, VRSA
oxolidinone
quinupristin / dalfopristin
MDR E. faecium
skin inf: MSSA, S pyogenes
straptogramins
chloramphenicol
wide spectrum, last line
covers meningitis bugs
protein synthesis inhibitor [no class]
sulfanilamide
broad spectrum - not used (pKa 10.5)
sulfonamide
sulfadiazine / sulfamerazine / sulfamethazine
broad spectrum, esp UTI (E coli, K pneumoniae, Salmonella)
sulfonamide
silver / sulfadiazine
broad spectrum topical, esp P aeruginosa
also fungi
sulfonamide
sulfisoxazole
broad spectrum, mostly used for gram (-) e.g. UTI (E coli, Salmonella, Shigella), Klebsiella, H influenzae, Proteus
sulfonamide
sulfisoxazole / phenazopyridine
broad spectrum, mostly used for gram (-) e.g. UTI (E coli, Salmonella, Shigella), Klebsiella, H influenzae, Proteus
Azo - local UT analgesic
sulfonamide
sulfisoxazole acetyl / E.E.S.
broad spectrum, esp otitis media
sulfonamide / macrolide
sulfamethoxazole
wide spectrum
also T gondii (protozoa)
sulfonamide
sulfacetamide
broad spectrum, for ophthalmic use
sulfonamide
trimethoprim
synergism with sulfamethoxazole
dihydrofolate reductase inhibitor
sulfamethoxazole / trimethoprim
very wide spectrum - all the bugs
even some MRSA, T gondii, P jiroveci (protozoal)
sulfonamide
nalidixic acid
gram(-), esp E coli, M morganii, Proteus, P rettgeri
NO P aeroginosa
quinolone
norfloxacin
broadish spectrum, mainly gram(-), esp P aeruginosa
fluoroquinolone (G2)
ciprofloxacin
broadish spectrum, mainly gram(-), esp P aeruginosa, B anthracis, household prevention for meningitis
fluoroquinolone (G2)
ofloxacin
broadish spectrum, incl E coli UTI
fluoroquinolone (G2)
levofloxacin
broader spectrum, incl MDR Strep
fluoroquinolone (G2)
gatifloxacin
broader spectrum, incl S pneumoniae
fluoroquinolone (G3)
moxifloxacin
intracellular / anaerobes, e.g. Bacteroides
esp Strep pneumoniae
NOT for UTI
fluoroquinolone (G4)
gemifloxacin
best gram(+) of FQs, esp MDR S pneumoniae
some gram (-)
anaerobes, e.g. Bacteroides
fluoroquinolone (G4)
besifloxacin
broad spectrum, conjunctivitis
fluoroquinolone
methenamine / hippuric acid
UTI, nearly all bacteria except Proteus
adjunct UTI agent
nitrofurantoin powder
UTI, E coli and Enterococci only
UTI agent
nitrofurantoin macrocrystals
UTI, E coli and Enterococci only
UTI agent
nitrofurantoin macrocrystals / gel polymer
UTI, E coli and Enterococci only
UTI agent
metronidazole
anaerobic cocci and bacilli (e.g. Bacteroides)
amoebiasis, trichomoniasis, giardiasis, C diff DoC
anti-parasitic
quinine
malaria merozoicide (gameticide for vivax, malariae)
NOT DoC
anti-parasitic
quinidine
malaria merozoicide (gameticide for vivax, malariae)
NOT DoC
anti-parasitic
diloxanide furoate
special use (through CDC): entamoeba hystolitica
anti-parasitic
atovaquone
P jiroveci, T gondii
anti-parasitic
atovaquone / proguanil
P falciparum (chloroquine resistant) - prophylaxis and treatment
anti-parasitic
chloroquine
malaria DoC esp relapse suppression
also E hystolitica
anti-parasitic
hydroxychloroquine
malaria DoC esp relapse suppression
also E hystolitica
anti-parasitic
mefloquine
chloroquine-resistant Plasmodium
anti-parasitic
pyrimethamine
chloroquine-resistant Plasmodium
anti-parasitic
paromomycin
E hystolitica
anti-parasitic
trimetrexate
pneumocystis (with Leucovorin)
anti-parasitic
nitazoxanide
special use: giardia lamblia
anti-parasitic
tinidazole
trichomoniasis, giardiasis, amoebiasis
anti-parasitic
γ-benzene hexachloride
Sarcoptes scabiei (Scabies) and Pediculus sp. (lice) in >110lb
anti-ectoparasitic
pyrethryins
Sarcoptes scabiei (Scabies) and Pediculus sp. (lice)
anti-ectoparasitic
permithrin
Sarcoptes scabiei (Scabies - 5%) and Pediculus sp. (lice - 1%)
anti-ectoparasitic
spinosad (spynocin A and D)
pediculus (lice) in > 4yo
anti-ectoparasitic
mebendazole
nematodes
antihelmintic
albendazole
nematodes
antihelmintic
ivermectin
Onchocerciasis DoC
nematode: pinworm, roundworm
antihelmintic
praziquantel
cestode, trematode
antihelmintic
pyrantel pamoate
nematodes
antihelmintic