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20 Cards in this Set
- Front
- Back
2 groups of myorelaxants? |
1. Spasmolytics 2. Neuromuscular blockers |
|
Main spasmolytic groups? |
1. Benzodiazepines 2. GABA agonists 3. Alpha2-agonist 4. Antiepileptics 5. Others |
|
What benzodiazepines are used as spasmolytics? |
- Tetrazepam - Diazepam |
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What GABA agonist are used as spasmolytic? |
Baclofen |
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What alpha2-agonist is used as spasmolytic? |
Tizanidine |
|
What antiepileptic is used as spasmolytic? |
Gabapentin |
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What are the other spasmolytics? |
- Mephenoxalone - Tolperison - Carisoprodol - Dantrolene |
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2 groups of neuromuscular blockers? |
1. Nondepolarizing (curare) 2. Depolarizing (succinylcholine) |
|
3 types of classifications of nondepolarizing neuromuscular blockers? |
1. Benzylisocholines vs. steroids 2. Type of elimination 3. Duration of action |
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Which nondepolarizing neuromuscular blockers are benzylisocholines? |
- Tubokurarin - Mivacurium - Atracurium - Cisatracurium
(curiums) |
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Which nondepolarizing neuromuscular blockers are steroid molecules? |
- Pancuronium - Pipecuronium - Rocuronium - Vecuronium
(curoniums) |
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Which nondepolarizing NM blockers are secreted unchanged by kidney? (GF) |
Tubokurarin |
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Which nondepolarizing NM blockers are decomposed by pseudocholineEsterase? |
Mivacurium |
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Which nondepolarizing NM blockers decompose spontaneously in blood? |
- Atracurium - Cis-atracurium |
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Which nondepolarizing NM blockers are metabolized by liver and secreted in bile? |
- Rocuronium - Vecuronium |
|
Which nondepol NM blockers are long lasting? |
- Tubokurarin - Pancuronium - Pipecuronium |
|
Which nondepol. NM blockers are medium lasting? |
- Atracuronium - Cis-atracuronium - Rocuronium - Vecuronium |
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Which nondepol. NM blockers are short lasting? |
Mivacurium |
|
Which nondepol. NM blocker may be ultra short lasting and may displace succinylcholine? |
Rocuronium |
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What are the depolarizing neuromuscular blockers? |
- Suxamethonium (succinylcholine) - Botulinum toxin (?) |