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20 Cards in this Set

  • Front
  • Back

2 groups of myorelaxants?

1. Spasmolytics


2. Neuromuscular blockers

Main spasmolytic groups?

1. Benzodiazepines


2. GABA agonists


3. Alpha2-agonist


4. Antiepileptics


5. Others

What benzodiazepines are used as spasmolytics?

- Tetrazepam


- Diazepam

What GABA agonist are used as spasmolytic?

Baclofen

What alpha2-agonist is used as spasmolytic?

Tizanidine

What antiepileptic is used as spasmolytic?

Gabapentin

What are the other spasmolytics?

- Mephenoxalone


- Tolperison


- Carisoprodol


- Dantrolene

2 groups of neuromuscular blockers?

1. Nondepolarizing (curare)


2. Depolarizing (succinylcholine)

3 types of classifications of nondepolarizing neuromuscular blockers?

1. Benzylisocholines vs. steroids


2. Type of elimination


3. Duration of action

Which nondepolarizing neuromuscular blockers are benzylisocholines?

- Tubokurarin


- Mivacurium


- Atracurium


- Cisatracurium



(curiums)

Which nondepolarizing neuromuscular blockers are steroid molecules?

- Pancuronium


- Pipecuronium


- Rocuronium


- Vecuronium



(curoniums)

Which nondepolarizing NM blockers are secreted unchanged by kidney? (GF)

Tubokurarin

Which nondepolarizing NM blockers are decomposed by pseudocholineEsterase?

Mivacurium

Which nondepolarizing NM blockers decompose spontaneously in blood?

- Atracurium


- Cis-atracurium

Which nondepolarizing NM blockers are metabolized by liver and secreted in bile?

- Rocuronium


- Vecuronium

Which nondepol NM blockers are long lasting?

- Tubokurarin


- Pancuronium


- Pipecuronium

Which nondepol. NM blockers are medium lasting?

- Atracuronium


- Cis-atracuronium


- Rocuronium


- Vecuronium

Which nondepol. NM blockers are short lasting?

Mivacurium

Which nondepol. NM blocker may be ultra short lasting and may displace succinylcholine?

Rocuronium

What are the depolarizing neuromuscular blockers?

- Suxamethonium (succinylcholine)


- Botulinum toxin (?)