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14 Cards in this Set
- Front
- Back
Conjugated Estrogens
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Estradiol
Ethinyl estradiol |
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SERM
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Raloxifene
|
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Estrogen Inhibitor
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Anastrozole
|
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Progestins
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Medroxyprogesterone
Norethindrone Levonorgestrel Progesterone |
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GnRH agonists
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Leuprolide
Goserelin Nafarellin |
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Anti-Androgen
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Flutamide
Finasteride Spironolactone |
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Estradiol
Ethinyl estradiol |
MOA - receptor interaction -> gene transcription
Uses - postmenopausal HRT (prevent vasomotor sxs), hormonal contraception CI - estrogen dep neoplasms, endometriosis, adolescent girls, pregs |
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Raloxifene
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MOA - agonists/antagonists on estrogen receptor - agonist in bone, antagonists in breast/uterus
Uses - prevention of breast cancer Tox - menopausal sxs, bone loss! |
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Anastrozole
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MOA - selective inhibitor of aromatase
Uses - post menopausal women w/ hormone receptor pos for breast cancer, relieves postmenopausal ab pain from endometriosis AE - hot flases, osteoporosis |
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Medroxyprogesterone
Norethindrone Levonorgestrel Progesterone |
Dx uses - test for estrogen secretion
Tx uses - hormonal contraception, endometriosis, DUB, dysmenorrhea, inc fertility, advanced breast and endometrial carcinoma |
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Leuprolide
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-> gonadal suppression
Uses - tx of prostatic carcinoma, rapid relief from endometriosis AE - bone loss |
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Flutamide (antagonist)
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MOA - competitive antagonist at androgen receptor
Uses - prostatic cancer |
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Finasteride (inhibitor)
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MOA - inhibits the 5-alpha reductase
Uses - BPH, hirsutism |
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Spironolactone
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Uses - hirsutism in females w/ PCOS
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