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26 Cards in this Set

  • Front
  • Back
TCA's
CYP2D6
FLUOXETINE
METABOLIZED BY CYP2D6
DECENT INHIBITOR OF CYP2C9
POTENT INHIBITOR OF CYP2D6
FLUVOXAMINE
METABOLIZED BY CYP2D6, 1A2
INHIBITS CYP3A4
MIRTAZAPINE
METABOLIZED BT CYP2D6
PAROXETINE
METABOLIZED BT CYP2D6
SERTRALINE
METABOLIZED BT CYP2D6?
ALSO 2C9/2C19
TRAZODONE
METABOLIZED BT CYP2D6
VENLAFAXINE
METABOLIZED BT CYP2D6
CITALOPRAM
METABOLIZED BY CYP3A4
NEFAZODONE
INHIBITS 3A4-INTERACTS WITH PROTEASE INHIBITORS
BUPROPRION
METABOLIZES CYP 2B6
INHIBITS CYP2D6
MOST BENZODIAZEPINES
METABOLIZED BY CYP3A4
BENZODIAZEPINES THAT ARE NOT METABOLIZED BY CYP P450
LORAZEPAM, OXAZEPAM, TEMAZEPAM
DIAZEPAM
METABOLIZED BY CYP2C9 AND 2C19
MOST TYPICAL NEUROLEPTICS
METABOLIZED BY CYP2D6
TYPICAL NEUROLEPTIC METABOLIZED BY CYP3A4
PIMOZIDE
CLOZAPINE
CYP1A2
OLANZAPINE
METABOLIZED BY CYP1A2
RISPERIDONE
CYP2D6
QUETIAPINE
METABOLIZED BY CYP3A4
ZIPRASIDONE
METABOLIZED BY CYP3A4
CARBAMEZAPINE
POTENT INDUCER OF CYP3A4
(ALSO METABOLIZED BY THE SAME; HENCE IT INDUCES ITS OWN METABOLISM, IE CHEWS ITSELF UP).
PREFERRED ANTIDEPRESSANTS FOR HAART PATIENTS
REMERON
EFFEXOR
CELEXA
LEXAPRO
CAUTION THESE ANTIDEPRESSANTS ARE RELATIVELY CONTRAINDICATED IN HIV HAART PATIENTS
WELLBUTRIN
PROZAC
TCAS
HAART POTENT INHIBITOR OF CYP P450 2B6, 2D6, AND 3A4
RITONAVIR
EFAVIRENZ
POTENT INHIBITOR OF 2B6