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70 Cards in this Set
- Front
- Back
carbamazepine
|
strong CYP inducer
|
|
adriamycin
|
P-glycoprotein – substrate
|
|
amiodarone
|
2D6 – moderate inhibitor
use sotalol 2C9 – moderate inhibitor use sotalol P-glycoprotein – inhibitor |
|
amphetamines
|
2D6 – major substrate
|
|
atypical antipsychotics
|
2D6 – major substrate
|
|
benzodiazepines (alprazolam, triazolam, diazepam, midazolam)
|
3A4 – major substrate
use lorazepam or oxazepam for triazolam esp. |
|
caffeine
|
1A2 – major substrate
|
|
carvedilol
|
2C9 – major substrate
|
|
CCB (amlodipine, felodipine, diltiazem, verapamil)
|
3A4 – major substrate
|
|
celecoxib
|
2C9 – major substrate
|
|
charcoal-broiled foods
|
1A2 – moderate inhibitor
|
|
cigarette smoke
|
1A2 – moderate inhibitor
|
|
cimetidine
|
1A2 – moderate inhibitor
use famotidine 2C19 – moderate inhibitor use famotidine 2D6 – moderate inhibitor use famotidine 3A4 – moderate inhibitor |
|
ciprofloxacin
|
1A2 – strong inhibitor
use another FQ |
|
citalopram
|
2C19 – major substrate
|
|
clarithromycin
|
1A2 – moderate inhibitor
use azithromycin 3A4 – strong inhibitor P-glycoprotein – substrate P-glycoprotein – inhibitor |
|
clozapine
|
1A2 – major substrate
|
|
codeine --> morphine
|
2D6 – major substrate
|
|
daunorubicin
|
P-glycoprotein – substrate
|
|
diazepam
|
2C19 – major substrate
use lora-/oxa-/tema-zepam |
|
digoxin
|
P-glycoprotein – substrate
|
|
erythromycin
|
1A2 – moderate inhibitor
use azithromycin 3A4 – moderate inhibitor P-glycoprotein – substrate P-glycoprotein – inhibitor |
|
fluconazole
|
2C19 – strong inhibitor
use voriconazole 3A4 – moderate inhibitor 2C9 – strong inhibitor use voriconazole |
|
fluoxetine
|
2C19 – moderate inhibitor
2C9 – major substrate 2D6 – strong inhibitor use escitalopram |
|
fluvastatin
|
2C9 – major substrate
2C9 – moderate inhibitor |
|
fluvoxamine
|
1A2 – major substrate
1A2 – strong inhibitor use escitalopram 2C19 – strong inhibitor |
|
garlic (allicin)
|
strong CYP inducer
|
|
gemfibrozil
|
2C19 – strong inhibitor
use fenofibrate 2C9 – strong inhibitor |
|
glimepiride
|
2C9 – major substrate
|
|
glipizide
|
2C9 – major substrate
|
|
grapefruit juice
|
3A4 – strong inhibitor
|
|
haloperidol
|
2D6 – major substrate
|
|
hydro-/oxy-codone
|
2D6 – major substrate
|
|
hypericum (St. John’s Wort)
|
strong CYP inducer
|
|
ibuprofen
|
2C9 – strong inhibitor
use APAP |
|
isoniazid
|
2C19 – strong inhibitor
3A4 – strong inhibitor |
|
itraconazole
|
3A4 – strong inhibitor
|
|
ketoconazole
|
1A2 – strong inhibitor
use fluconazole 2D6 – moderate inhibitor use fluconazole 3A4 – strong inhibitor 2C9 – strong inhibitor P-glycoprotein – inhibitor |
|
losartan
|
2C9 – major substrate
|
|
methadone
|
2D6 – major substrate
|
|
metoprolol
|
2D6 – major substrate
|
|
metronidazole
|
3A4 – moderate inhibitor
|
|
mirtazapine
|
1A2 – major substrate
|
|
omeprazole
|
2C9 – moderate inhibitor
use lansoprazole or famotidine |
|
oral contraceptive
|
1A2 – major substrate
3A4 – major substrate |
|
paclitaxel
|
P-glycoprotein – substrate
|
|
paroxetine
|
2D6 – strong inhibitor
use escitalopram |
|
PDE5-I (sildenafil, tadalafil, & vardenafil)
|
3A4 – major substrate
|
|
phenobarbital
|
strong CYP inducer
2C19 – major substrate |
|
phenytoin
|
strong CYP inducer
2C19 – major substrate 2C9 – major substrate P-glycoprotein – substrate P-glycoprotein – inducer |
|
primidone
|
strong CYP inducer
|
|
propranolol
|
1A2 – major substrate
2D6 – major substrate |
|
protease inhibitors
|
3A4 – major substrate
P-glycoprotein – substrate |
|
quinidine
|
2D6 – strong inhibitor
3A4 – strong inhibitor P-glycoprotein – inhibitor |
|
rifampin
|
strong CYP inducer
P-glycoprotein – inducer |
|
ritonavir
|
2D6 – strong inhibitor
3A4 – strong inhibitor |
|
sertraline
|
2C19 – major substrate
2D6 – moderate inhibitor |
|
SSRIs
|
2D6 – major substrate
|
|
St. John’s Wort
|
P-glycoprotein – inducer
|
|
statins (atorvastatin, lovastatin, simvastatin)
|
3A4 – major substrate
use pravastatin or rosuvastatin |
|
TCA
|
2D6 – major substrate
|
|
telithromycin
|
3A4 – strong inhibitor
|
|
theophylline
|
1A2 – major substrate
|
|
TMP/SMX
|
2C9 – major substrate
2C9 – strong inhibitor |
|
tramadol
|
2D6 – major substrate
|
|
verapamil
|
P-glycoprotein – inhibitor
|
|
vinca alkaloids
|
P-glycoprotein – substrate
|
|
voriconazole
|
3A4 – moderate inhibitor
2C9 – major substrate |
|
warfarin
|
2C9 – major substrate
|
|
zileuton
|
1A2 – moderate inhibitor
use montelukast |