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30 Cards in this Set
- Front
- Back
Atenolol
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B1 Antagonist
50-100mg Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness |
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Metoprolol
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B1 Antagonist
25-100mg Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness |
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Bisoprolol
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B1 Antagonist
2.5-10mg Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness |
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Clonidine
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a2 agonist
Tablet: 0.1-0.8mg Patch: 0.1-0.3mg Could cause: orthostatic hypotension, drowsiness, dizziness |
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Hydrochlorothiazide
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DCT diuretic (thiazide)
12-25mg Compete for the Cl binding site and thus inhibit the Na, Cl symporter causing increased excretion of Na, Cl, H2O and K This symporter is responsible for ~ 5% of Na reabsorption |
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Furosemide
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Lasix (Loop Diuretic)
20-80mg/day Compete for the Cl binding site of the Na, K, 2Cl symporter causing increased excretion of Na, Cl, H2O, K, Ca, Mg This symporter is responsible for ~ 25% of Na reabsorption THESE AGENTS ARE NOT TO BE USED FOR THE TREATMENT OF HYPERTENSION ALONE! |
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Amiloride
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K sparing diuretic
5-10mg/day Block Na channels in the late distal tubule and collecting duct |
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Triamterene
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K sparing diuretic
50-100mg/day Block Na channels in the late distal tubule and collecting duct |
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Spironolactone
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K sparing diuretic
25-50mg/day Aldosterone inhibitors bind the mineralocorticoid receptor in the late distal tubule and collecting duct Net result is blockade of Na movement from luminal to interstitial space through Na channels and pumps |
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Captopril
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ACEI
25-100mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Lisinopril
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ACEI
10-40mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Ramipril
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ACEI
2.5-20mg/dat Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Trandolapril
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ACEI
1-4mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Enalapril
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ACEI
5-20mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Quinapril
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ACEI
10-40mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Perindopril
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ACEI
4-8mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Fosinopril
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ACEI
10-40mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Benazepril
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ACEI
10-40mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness |
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Losartan
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ARB
25-100mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Olmesartan
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ARB
20-40mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Candesartan
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ARB
8-32mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Valsartan
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ARB
80-320mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Irbesartan
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ARB
150-300mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Telmisartan
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ARB
20-80mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Eprosartan
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ARB
400-800mg/day Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness |
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Aliskerin
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Direct Renin Inhibitor
150-300mg/day Inhibits the conversion of angiotensinogen to angiotensin I via direct renin inhibition Could cause: Diarrhea, cough, dizziness |
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Amlodipine
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Dihydropyridine CCB
5-10mg/day In general, more selective for vascular smooth muscle Could cause: Edema, HA |
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Felodipine
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Dihydropyridine CCB
5-10mg/day In general, more selective for vascular smooth muscle Could cause: HA, dizziness |
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Diltiazem
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Non-Dihydropyridine CCB
120-540mg/day Less selectivity for vascular smooth muscle (relatively equal affinity for cardiac and vascular calcium channels) (edema caused by vasodilation) More likely to have a depressant effect on the heart Could cause: Hypotension, bradycardia |
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Verapamil
|
Non-Dihydropyridine CCB
80-480mg/day Less selectivity for vascular smooth muscle (relatively equal affinity for cardiac and vascular calcium channels) (edema caused by vasodilation) More likely to have a depressant effect on the heart Could cause: Hypotension, constipation, edema |