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30 Cards in this Set

  • Front
  • Back
Atenolol
B1 Antagonist

50-100mg

Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness
Metoprolol
B1 Antagonist

25-100mg

Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness
Bisoprolol
B1 Antagonist

2.5-10mg

Could cause: Bradycardia, ED, insomnia, heart palpitation, dizziness
Clonidine
a2 agonist

Tablet: 0.1-0.8mg
Patch: 0.1-0.3mg

Could cause: orthostatic hypotension, drowsiness, dizziness
Hydrochlorothiazide
DCT diuretic (thiazide)

12-25mg

Compete for the Cl binding site and thus inhibit the Na, Cl symporter causing increased excretion of Na, Cl, H2O and K

This symporter is responsible for ~ 5% of Na reabsorption
Furosemide
Lasix (Loop Diuretic)

20-80mg/day

Compete for the Cl binding site of the Na, K, 2Cl symporter causing increased excretion of Na, Cl, H2O, K, Ca, Mg

This symporter is responsible for ~ 25% of Na reabsorption

THESE AGENTS ARE NOT TO BE USED FOR THE TREATMENT OF HYPERTENSION ALONE!
Amiloride
K sparing diuretic

5-10mg/day

Block Na channels in the late distal tubule and collecting duct
Triamterene
K sparing diuretic

50-100mg/day

Block Na channels in the late distal tubule and collecting duct
Spironolactone
K sparing diuretic

25-50mg/day

Aldosterone inhibitors bind the mineralocorticoid receptor in the late distal tubule and collecting duct

Net result is blockade of Na movement from luminal to interstitial space through Na channels and pumps
Captopril
ACEI

25-100mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Lisinopril
ACEI

10-40mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Ramipril
ACEI

2.5-20mg/dat

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Trandolapril
ACEI

1-4mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Enalapril
ACEI

5-20mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Quinapril
ACEI

10-40mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Perindopril
ACEI

4-8mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Fosinopril
ACEI

10-40mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Benazepril
ACEI

10-40mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, cough, dizziness
Losartan
ARB

25-100mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Olmesartan
ARB

20-40mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Candesartan
ARB

8-32mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Valsartan
ARB

80-320mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Irbesartan
ARB

150-300mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Telmisartan
ARB

20-80mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Eprosartan
ARB

400-800mg/day

Could cause: Hyperkalemia, transient SCr increase, renal insufficiency, dizziness
Aliskerin
Direct Renin Inhibitor

150-300mg/day

Inhibits the conversion of angiotensinogen to angiotensin I via direct renin inhibition

Could cause: Diarrhea, cough, dizziness
Amlodipine
Dihydropyridine CCB

5-10mg/day

In general, more selective for vascular smooth muscle

Could cause: Edema, HA
Felodipine
Dihydropyridine CCB

5-10mg/day

In general, more selective for vascular smooth muscle

Could cause: HA, dizziness
Diltiazem
Non-Dihydropyridine CCB

120-540mg/day

Less selectivity for vascular smooth muscle (relatively equal affinity for cardiac and vascular calcium channels) (edema caused by vasodilation)

More likely to have a depressant effect on the heart

Could cause: Hypotension, bradycardia
Verapamil
Non-Dihydropyridine CCB

80-480mg/day

Less selectivity for vascular smooth muscle (relatively equal affinity for cardiac and vascular calcium channels) (edema caused by vasodilation)

More likely to have a depressant effect on the heart

Could cause: Hypotension, constipation, edema