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161 Cards in this Set
- Front
- Back
Epinephrine
|
a1, a2, b1, b2 agonist
|
|
Norepinephrine
|
a1, a2, b1, b3 agonist
Limited b2 |
|
Isoproterenol
|
b1, b2 agonist
|
|
Dopamine
|
D1, D2, a1, b1, b2 agonist
|
|
Ephedrine
Pseudoephedrine |
a1, b1, b2 agonist; releases NE
|
|
Amphetamine
|
Releases NE and DA
|
|
Phenylephrine
|
a1 agonist
|
|
Methoxamine
|
a1 agonist
|
|
Tetrahydrozoline
|
a1 agonist
|
|
Oxymetazoline
|
a1 agonist
|
|
Clonidine
|
a2 agonist; has imidazoline activity
|
|
Guanfacine
|
a2 agonist
|
|
Guanabenz
|
a2 agonist
|
|
Dobutamine
|
b1 agonist
|
|
Terbutaline
|
b2 agonist
|
|
Albuterol
|
b2 agonist
|
|
Metaproterenol
|
b2 agonist
|
|
Salmeterol
|
b2 agonist
|
|
Formoterol
|
b2 agonist
|
|
Ritodrine
|
b2 agonist
|
|
Phenoxybenzamine
|
a1, a2 antagonist
|
|
Phentolamine
|
a1, a2 antagonist
|
|
Prazosin
|
a1 antagonist
|
|
Terazosin
|
a1 antagonist
|
|
Doxazosin
|
a1 antagonist
|
|
Alfuzosin
|
a1 antagonist
|
|
Tamsulosin
|
a1a antagonist
|
|
Yohimbine
|
a2 antagonist
|
|
Propranolol
|
b1, b2 antagonist
|
|
Pindolol
|
b1, b2 antagonist
|
|
Timolol
|
b1, b2 antagonist
|
|
Nadolol
|
b1, b2 antagonist
|
|
Sotalol
|
b1, b2 antagonist
|
|
Metoprolol
|
b1 antagonist
|
|
Atenolol
|
b1 antagonist
|
|
Esmolol
|
b1 antagonist
|
|
Acebutolol
|
b1 antagonist
|
|
Bisoprolol
|
b1 antagonist
|
|
Butoxamine
|
b2 antagonist
|
|
Labetalol
|
Mixed a1, b1, b2 actions
|
|
Carvedilol
|
Mixed a1, b1, b2 actions
|
|
Acetylcholine
|
Direct nicotinic and muscarinic agonist
|
|
Nicotine
|
Direct nicotinic agonist
|
|
Methacholine
|
Direct M3 agonist
|
|
Carbachol
|
Direct nicotinic and muscarinic agonist
|
|
Bethanechol
|
Direct muscarinic agonist
|
|
Arecholine
|
Direct nicotinic and muscarinic agonist
|
|
Muscarine
|
Direct muscarinic agonist
|
|
Pilocarpine
|
Direct muscarinic agonist
|
|
Physostigmine
|
Inhibits AChE
|
|
Neostigmine
|
Inhibits AChE
|
|
Pyridostigmine
|
Inhibits AChE
|
|
Edrophonium
|
Inhibits AChE
|
|
Tacrine
|
Inhibits AChE
|
|
Donepezil
|
Inhibits AChE
|
|
Galantamine
|
Inhibits AChE
|
|
Rivastigmine
|
Inhibits AChE
|
|
Atropine
|
Non-selective muscarinic antagonist
|
|
Scopolamine
|
Muscarinic antagonist
|
|
Ipratropium
|
M1, M2, M3 antagonist
|
|
Tiotropium
|
M1, M3 antagonist
|
|
Tolterodine
|
Muscarinic antagonist
|
|
Oxybutynin
|
Muscarinic antagonist
|
|
Solfenacin
|
M3 antagonist
|
|
Darifenacin
|
M3 antagonist
|
|
Benztropine
|
Muscarinic antagonist
|
|
Trihexyphenidyl
|
Muscarinic antagonist
|
|
Pirenzipine
|
M1 antagonist
|
|
Mecamylamine
|
Ganglionic blocker
|
|
Succinylcholine
|
Depolarizing blocker
|
|
D-tubocurarine
|
Neuromuscular blocker
Non-depolarizing antagonist |
|
Pancuronium
|
Neuromuscular blocker
|
|
Doxacurium
|
Neuromuscular blocker
|
|
Levalbuterol
|
b2 agonist
|
|
Pirbuterol
|
b2 agonist
|
|
Theophylline
|
Phosphodiesterase inhibitor
Adenosine receptor antagonist |
|
Zafirlukast
|
Leukotriene antagonist
|
|
Montelukast
|
Leukotriene antagonist
|
|
Zileuton
|
5-lipooxygenase inhibitor
|
|
Omalizumab
|
IgE monoclonal antibody
|
|
Furosemide
|
Loop diuretic
|
|
Bumetanide
|
Loop diuretic
|
|
Torsemide
|
Loop diuretic
|
|
Ethacrynic acid
|
Loop diuretic
|
|
Bendroflumethiazide
|
Thiazide diuretics
|
|
Chlorothiazide
|
Thiazide diuretics
|
|
Hydrochlorothiazide
|
Thiazide diuretics
|
|
Methylclothiazide
|
Thiazide diuretics
|
|
Polythiazide
|
Thiazide diuretics
|
|
Thichlormethiazide
|
Thiazide diuretics
|
|
Chlorthalindone
|
Thiazide-like diuretic
|
|
Metolazone
|
Thiazide-like diuretic
|
|
Indapamide
|
Thiazide-like diuretic
|
|
Amiloride
|
K+ sparing diuretic
|
|
Triamterene
|
K+ sparing diuretic
|
|
Spironolactone
|
Aldosterone antagonist
|
|
Eplerenone
|
Aldosterone antagonist
|
|
Acetazolamide
|
Carbonic anhydrase inhibitor
|
|
Dichlorphenamide
|
Carbonic anhydrase inhibitor
|
|
Methazolamide
|
Carbonic anhydrase inhibitor
|
|
Mannitol
|
Osmotic diuretic
|
|
Glycerin
|
Osmotic diuretic
|
|
Isosorbide
|
Osmotic diuretic
|
|
Urea
|
Osmotic diuretic
|
|
Captopril
|
ACE inhibitor
|
|
Lisinopril
|
ACE inhibitor
|
|
Enalapril
|
ACE inhibitor
|
|
Benazepril
|
ACE inhibitor
|
|
Fosinopril
|
ACE inhibitor
|
|
Trandolapril
|
ACE inhibitor
|
|
Quinapril
|
ACE inhibitor
|
|
Ramipril
|
ACE inhibitor
|
|
Perindopril
|
ACE inhibitor
|
|
Moexipril
|
ACE inhibitor
|
|
Candesartan
|
Angiotensin receptor blocker
|
|
Olmesartan
|
Angiotensin receptor blocker
|
|
Losartan
|
Angiotensin receptor blocker
|
|
Eprosartan
|
Angiotensin receptor blocker
|
|
Irbesartan
|
Angiotensin receptor blocker
|
|
Telmisartan
|
Angiotensin receptor blocker
|
|
Valsartan
|
Angiotensin receptor blocker
|
|
Aliskiren
|
Renin inhibitor
|
|
Diltiazem
|
Benzothiazepine calcium channel blocker
|
|
Verapamil
|
Phenylalkylamine calcium channel blocker
|
|
Amlodipine (and every drug ending in -pine)
|
DHP calcium channel blocker
|
|
Cholestyramine
|
Bile acid sequestrant
|
|
Colestipol
|
Bile acid sequestrant
|
|
Colesevelam
|
Bile acid sequestrant
|
|
Simvastatin (and every drug ending in -statin)
|
HMG-CoA reductase inhibitors
|
|
Ezetimibe
|
NPC1L1 inhibitor
|
|
Fenofibrate
|
Fibric acid derivative
|
|
Gemfibrozil
|
Fibric acid derivative
|
|
Niacin
|
B-complex vitamin
|
|
a-methyldopa
|
a2 agonist
|
|
Rilmenidine
|
Imidazoline agonist
|
|
Reserpine
|
Blocks transport into vesicles, synthesis of vesicles
|
|
Hydralazine
|
Increases cGMP and NO
|
|
Minoxidil
|
Activates K+ channels
|
|
Nitroprusside
|
Activates cGMP, decreases intracellular Ca++
|
|
Diazoxide
|
Prolongs K+ channel opening
|
|
Fenoldopam
|
D1 and a2 agonist
|
|
Sildenafil
|
Phosphodiesterase 5 inhibitor
|
|
Tadalafil
|
Phosphodiesterase 5 inhibitor
|
|
Vardenafil
|
Phosphodiesterase 5 inhibitor
|
|
Digoxin
|
Positive inotrope
Decreases sympathetic tone Increases parasympathetic tone |
|
Milrinone
|
cAMP phosphodiesterase 3 inhibitors
|
|
Inaminrone
|
cAMP phosphodiesterase 3 inhibitors
|
|
Quinidine
|
Class 1a Na+ channel blocker
|
|
Procainamide
|
Class 1a Na+ channel blocker
|
|
Disopyramide
|
Class 1a Na+ channel blocker
|
|
Lidocaine
|
Class 1b Na+ channel blocker
|
|
Mexiletine
|
Class 1b Na+ channel blocker
|
|
Flecainide
|
Class 1c Na+ channel blocker
|
|
Propafenone
|
Class 1c Na+ channel blocker
|
|
Amiodarone
|
Class 3 K+ channel blocker
|
|
Dronedarone
|
Class 3 K+ channel blocker
|
|
Ibutilide
|
Class 3 K+ channel blocker
|
|
Dofetilide
|
Class 3 K+ channel blocker
|
|
Adenosine
|
Activates K+ channels
Blocks Ca++ channels |
|
Phenytoin
|
Blocks inactivated Na+ channels
|
|
Moricizine
|
Na+ channel blocker
|