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295 Cards in this Set

  • Front
  • Back
Acetylcholine
Direct Acting Cholinergic Agonist
Bethanechol
Direct acting cholinergic agonist
carbachol
direct acting cholinergic agonist
cevimeline
direct acting cholinergic agonist
ambenomium
Acetylcholinesterase inhibitor
Donepezil
Acetylcholinesterase inhibitor
edrophonium
acetylcholinesterase inhibitor
galantamine
acetylcholinesterase inhibitor
neostigmine
acetylcholinesterase inhibitor
physostigmiine
acetylcholinesterase inhibitor
physostigmine
acetylcholinesterase inhibitor
pyridostigmine
acetylcholinesterase inhibitor
rivastigmine
acetylcholinesterase inhibitor
tacrine
acetylcholinesterase inhibitor
echothiophate
anticholinesterase irreversible
isoflurophate
anticholinesterase irreversible
pralidoxime
reactivation of acetylcholine esterase
atropine
antimuscarinic agents
ipratropium
antimuscarinic agents
scopolamine
antimuscarinic agent
mecamylamine
ganglionic blockers
nicotine
ganglionic blocker
trimethaphan
ganglionic blocker
atracurium
neuromuscular blockers
cisatracurium
neuromuscular blocker
doxacurium
neuromuscular blocker
metocurine
neuromuscular blocker
mivacurium
neuromuscular blocker
pancuronium
neuromuscular blocker
rocuronium
neuromuscular blocker
succinylcholine
neuromuscular blocker
tubocurarine
neuromuscular blocker
vecuronium
neuromuscular blocker
antimuscarinic agents
block muscarinic receptors causing inhibition of all muscarinic functions
ganglionic blocker
act on the nicontinic receptors of both parasympathetic and sympathetic autonomic ganglia not effective at neuromuscular antagonist
albuterol
adrenergic agonist direct acting
clonidine
adrenergic agonist direct acting
dobutamine
adrenergic agonist direct acting
dopamine
adrenergic agonist direct acting
epinephrine
adrenergic agonist direct acting
formoterol
adrenergic agonist direct acting
isoproterenol
adrenergic agonist direct acting
metaproterenol
adrenergic agonist direct acting
methoxamine
adrenergic agonist direct acting
norepinephrine
adrenergic agonist direct acting
phenylephrine
adrenergic agonist direct acting
piruterol
adrenergic agonist direct acting
salmeterol
adrenergic agonist direct acting
tamsulosine
adrenergic agonist direct acting
terbutaline
adrenergic agonist direct acting
amphetamine
adrenergic agonist indirect acting
tyramine
adrenergic agonist indirect acting
ephedrine
adrenergic agonist direct and indirect(mixed action)
drug of choice for shock
dopamine
drug of choice for type 1 hypersensitivity reactions allergens
epinephrine
doxazosin
alpha blocker
phenoxybenzamine
alpha blocker
phentolamine
alpha blocker
prazosin
alpha blocker
tamsulosin
alpha blocker
terazosin
alpha blocker
acebutolol
beta blocker
atenolol
beta blocker
carvedilol
beta blocker
esmolol
beta blocker
labetalol
beta blocker
metoprolol
beta blocker
nadolol
beta blocker
pindolol
beta blocker
propranolol
beta blocker
timolol
beta blocker
cocaine
drugs affecting neurotransmitter uptake or release
guanethidine
blocks realese of stored epinephrine
reserpine
block atp dependent transport of biogenic amines
loss of cholinergic neurons in the nucleus basalis of maynert
alzheimer disease
loss of dopaminergic neurons in substatia nigra
parkinsons
amantadine
anti-parkinson drugs
benzotropine
anti-parkinson drugs
biperiden
anti-parkinson drugs
bromocriptine
anti-parkinson drugs
carbidopa
anti-parkinson drugs
entacapone
anti-parkinson drugs
levodopa
anti-parkinson drugs
pergolide
anti-parkinson drugs
pramipexole
anti-parkinson drugs
ropinirole
anti-parkinson drugs
selegiline(deprenyl)
anti-parkinson drugs
tolcapone
anti-parkinson drugs
trihexphenidyl
anti-parkinson drugs
donepezil
anti-alzeheimer
galantamine
anti-alzeheimer
memantine
anti-alzeheimer
rivastigmine
anti-alzeheimer
tacrine
anti-alzeheimer
alprazolam
benzodiazepines
chlordiazepoxide
benzodiazepines
diazepam
benzodiazepines
flurazepam
benzodiazepines
oxazepam
benzodiazepines
temazepam
benzodiazepines
triazolam
benzodiazepines
buspirone
hypnotic, rifampin shortened half life, erthromycin lengthens half life
eszopiclone
non benzodiazepine, used for insomnia
hydroxyzine
antihistamine with antiemetic
zaleplon
hypnotic
zolpidem
hypnotic, avoid rifampin
flumazenil
benzodiazepine antagonist
amobarbital
barbiturates
phenobarbital
barbiturates
secobarbital
barbiturates
thipental
barbiturates
antihistamines
nonbarbiturate sedatives
chloral hydrate
nonbarbiturate sedatives
ethanol
nonbarbiturate sedatives
modafinil
antinarcoleptic drugs
citalopram
ssri
escitalopram
ssri
fluoxetine
ssri
fluoxamin
ssri
paroxetine
ssri
sertraline
ssri
venlafaxine
seratonin norepinephrine re-uptake inhibitor
duloxetine
seratonin norepinephrine re-uptake inhibitor
bupropion
atypical antidepressant
mirtazapine
atypical antidepressants
nefazodone
atypical antidepressant
trazodone
atypical antidepressant
amitriptyline
tricyclic antidepressants
amoxapine
tricyclic antidepressants
clomipramine
tricyclic antidepressants
doxepin
tricyclic antidepressants
imipramine
tricyclic antidepressants
maprotiline
tricyclic antidepressants
nortriptyline
tricyclic antidepressants
protriptyline
tricyclic antidepressants
trimipramine
tricyclic antidepressants
phenelzine
moa inhibitor
tranylcypromine
moa inhibitor
carbamazepine
treat mania
litium salts
drugs to treat mania
valproic acid
drugs to treat mania
chlorpromazine
typical neuroleptic(low potency)
prochlorpromazine
typical neuroleptic (low potency)
promethazone
typical neuroleptic (low potency)
thioridazine
typical neuroleptic (low potency)
fluphenazine
neuroleptic (high potency)
haloperidol
neuroleptic (high potency)
pimozide
neuroleptic (high potency)
thiothixene
neuroleptic (high potency)
aripiprazole
atypical neuroleptic
clozapine
atypical neuroleptic
olanzapine
atypical neuroleptic
quetiapine
atypical neuroleptic
risperidone
atypical neuroleptic
ziprasidone
atypical neuroleptic
drug associated with blood dyscrasias
clozapine
drug of choice to treat motion sickness
scopolamine
treat intractable hiccups
chlorpromazine
drugs that block dopamine receptors can cause mimic symptoms similar to what
parkinson
alfentanil
opiod strong agonist
fentanyl
opiod strong agonist
heroin
opiod strong agonist
meperidine
opiod strong agonist
methadone
opiod strong agonist
morphine
opiod strong agonist
remifentanil
opiod strong agonist
sufentanil
opiod strong agonist
codeine
opiod moderate/low agonist
oxycodone
opiod moderate/low agonist
propoxyphene
opiod moderate/low agonist
buprenorphine
opiod partial agonist acts like morphine in naive patients can pricipitate withdrawal in morphine users
two drugs used to treat opiod dependence
1. methadone 2. buprenophine
nalbuphine and butorphanol
partial opiod agonist
pentazocine
opiod agonist on Kappa receptors weak antagonist at mu and delta
tramadol
centrally acting analgesic binds to mu opiod receptor
naloxone
competitive opiod antagonist
naltrexone
opiod antagonist longer duration of action than naloxone
suppress tonic clonic seizures
phenytoin
treatment of partial seizures
carbamazepine
valproic acid
2ndary anticonvulsant
ethosuximide
anticonvulsant
felbamate
anticonvulsant reserved for refractory epilepsies (lennox-gestaut)
gabapentin
anticonvulsant used for partial seizures
lamotrigine
wide spectrum anticonvulsant
levetiracetam
anticonvulsant
tigabine
anticonvulsant
topiramate
anticonvulsant
zonisamide
anticonvulsant
captopril
ace inhibitor
enalapril
ace inhibitor
fosinopril
ace inhibitor
lisinopril
ace inhibitor
quinapril
ace inhibitor
ramipril
ace inhibitor
candesartan
arb blocker
losartan
arb blocker
telmisartan
arb blocker
valsartan
arb blocker
hydralazine
direct vasodialators
isosorbide dinitrate
direct vasodialators
sodium nitroprusside
direct vasodilators
amrinone
inotropic agents
digitoxin
inotropic agents
digoxin
inotropic agents
dobutamine
inotropic agents
milrinone
inotropic agents
spironolactone
aldosterone antagonist K+ sparing diuretic
disopyramide
class Ia antiarrhythmic (na+ channel blocker)
flecainide
class Ic antiarrhythmic (na+ channel blocker)
lidocaine
class Ib antiarrhythmic (na+ channel blocker)
mexiletine
class Ib antiarrhythmic (na+ channel blocker)
procainamide
class Ia antiarrhythmic (na+ channel blocker)
propafenone
class Ic antiarrhythmic (na+ channel blocker)
quinidine
class Ia antiarrhythmic (na+ channel blocker)
tocainide
class Ib antiarrhythmic (na+ channel blocker)
class II antiarrhythmic
beta blockeres
amiodarone
class III antiarrhythmic K+ channel blocker
dofetilide
class III antiarrhythmic K+ channel blocker
sotalol
class III antiarrhythmic K+ channel blocker
class IV antiarrhythmic
ca2+ channel blocker
adenosine
treatment for acute supraventricular tachycardia 15 second duration
treatment for angina attacks
organic nitrates, beta blockers, calcium channel blockers
amlodipine
ca channel blocker
diltiazem
ca channel blocker
felodipine
ca channel blocker
isradipine
ca channel blocker
nicardipine
ca channel blocker
nifedipine
ca channel blocker
nisoldipine
ca channel blocker
verapamil
ca channel blocker
bumetanide
loop diuretic
ethacrynic acid
loop diuretic
furosemide
loop diuretic
torsemide
loop diuretic
chlorothiazide
thiazide diuretic
chlorthalidone
thiazide diuretic
hydrochlorothiazide
thiazide diuretic
indapamide
thiazide diuretic
metolazone
thiazide diuretic
amiloride
K+ sparing diuretic
triamterene
K+ sparing diuretic
acetazolamide
carbonic anhydrase inhibitor
mannitol
osmotic diuretic
urea
osmotic diuretic
atorvastatin
statin - hmg coa reductase inhibitor
fluvastatin
statin - hmg coa reductase inhibitor
lovastatin
statin - hmg coa reductase inhibitor
pravastatin
statin - hmg coa reductase inhibitor
rosuvastatin
statin - hmg coa reductase inhibitor
simvastatin
statin - hmg coa reductase inhibitor
fenofibrate
fibrate
gemfibrozil
fibrate
niacin
lowers ldl and best for raising good hdl can be used in combo with statins
colesevelam
bile acid sequestrant
colesevelam
bile acid sequestrant
cholestryamine
bile acid sequestrant
ezetimibe
cholesterol absorption inhibitors
abciximab
platelet inhibitor
aspirin
platelet inhibitor
clopidogrel
platelet inhibitor
dipyridamole
platelet inhibitor
eptifibatide
platelet inhibitor
ticlopidine
platelet inhibitor
tirofiban
platelet inhibitor
danaparoid
anticoagulant
enoxaprin
anticoagulant
heparin
anticoagulant binds to antithrombin III
lepirudin
anticoagulant
warfarin
anticoagulant vitamin K antagonist
alteplase
thrombolytic agents
streptokinase
thrombolytic agents
aminocaproic acid
treatment of bleeding
aprotinin
treatment of bleeding
protamine sulfate
treatment of bleeding
tranexamic acid
treatment of bleeding
vitamin k
treatment of bleeding
cyanocoblamin (b12 vitamin)
anemia tx
erythropoietin
anemia tx
folic acid
anemia tx
iron
anemia tx
hydroxyurea
tx sickle cell anemia
in a hypergylcemic emergency what should be injected
regular insulin
rapid onset and ultra short acting insulin
1. regular insulin 2. insulin lispro 3. insulin aspart 4. insulin glulisine
intermediate acting insulin
lente insulin, isophane nph insulin
prolonged acting insulin
ultralente insulin, insulin glargine, insulin detimir
sulfonylureas
insulin secretegogues
repaglinide
meglitinide analogs
nateglinide
meglitinide analogs
metformin
binguanides insulin sensitizer, decreases cardiovascular mortalitiy
glitazones
insulin sensitizers
troglitazone
insulin sensitizers
pioglitazone
insulin sensitizer
rosiglitazone
insulin sensitizer
acarbose
decrease digestion of carbohydrates
miglitol
decrease digestion of carbohydrates