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97 Cards in this Set
- Front
- Back
Heparin |
Complexes with AT and inhibits factors Xa and IIa
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LMW Heparin
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Complexes with AT and inhibits factors Xa and IIa
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Fondaparinux
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Complexes with AT and inhibits factor Xa
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Argatroban
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Directly inhibits IIa
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Bivalirudin
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Directly inhibits IIa
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Hirudin
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Directly inhibits IIa
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Antithrombin
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Directly inhibits IIa
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Protamine sulfate
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Heparin antagonist
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Warfarin
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(oral) Competitive antagonist of Vitamin K and suppresses factors II, VII, IX and X
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Vitamin K
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(oral) Cofactor in the synthesis of factors II, VII, IX and X
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Rivaroxaban
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(oral) Inhibits factor Xa
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Apixaban
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(oral) Inhibits factor Xa
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Dabigatran
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(oral) Inhibits thrombin
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Clopidogrel
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(AP) ADP receptor inhibitor
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Prasugrel
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(AP) ADP receptor inhibitor
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Ticagrelor
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(AP) ADP receptor inhibitor
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Dipyridamole
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(AP) Phosphodiesterase inhibitor
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Cilostazol
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(AP) Phosphodiesterase inhibitor
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Abciximab
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(AP) GP IIb/IIIa inhibitor
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Eptifibatide
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(AP) GP IIb/IIIa inhibitor
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Tirofiban
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(AP) GP IIb/IIIa inhibitor
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Monteleukast
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(AP) Leukotriene receptor inhibitor
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Zafirleukast
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(AP) Leukotriene receptor inhibitor
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Zieuton
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(AP) Lipoxygenase inhibitor
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Streptokinase
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Fibrinolytic
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Urokinase
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Fibrinolytic
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t-PA
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Fibrinolytic
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Epsilon amino acid acaproic acid
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Anti-fibrinolytic
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Aprotonin
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Anti-fibrinolytic
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Ancrod
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Fibrinolytic
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Tranexamic acid
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Anti-fibrinolytic
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Statins
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Inhibit HMG CoA reductase and triggers SREBP transcription factor which leads to an increase in LDL receptor expression
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Bile-acid binding resins
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Binds bile acids and prevents reabsorption
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Ezetimibe
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Inhibits intestinal absorption of cholesterol
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Niacin
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Decreases lipolysis, inhibits DGAT2, increases apoA1 and converts ApoCIII to LPL
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Fibrates
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Decreases ApoC3 expression, increases LPL expression, increases fatty acid oxidation and increases apoA1 expression
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Nitric Oxide
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Covalent modification of proteins
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Nitroglycerine
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NO donor
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Hydralazine
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NO donor, vasodilator
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Sildenafil
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Phosphodiesterase inhibitor
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L-arginine
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NO donor
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Captopril
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ACE inhibitor
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Enalapril
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ACE inhibitor
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Losartan
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Angiotensin receptor inhibitor
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Valsartan
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Angiotensin receptor inhibitor
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Icatibant
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Bradykinin receptor inhibitor
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Desmopressin (DDAVP)
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Vasopressin analogue
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Bosentan
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Endothelin receptor inhibitor
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Acetazolamide
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Inhibits carbonic anhydrase
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Mannitol
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Osmotic diuretic
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Dichlorphenamide
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Inhibits carbonic anhydrase
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Methazolamide
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Inhibits carbonic anhydrase
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Dorzolamide
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Inhibits carbonic anhydrase
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Furosemide
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Blocks Na/K/2Cl cotransporter in the TAL
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Bumetanide
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Blocks Na/K/2Cl cotransporter in the TAL
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Torsemide
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Blocks Na/K/2Cl cotransporter in the TAL
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Ethacrynic Acide
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Blocks Na/K/2Cl cotransporter in the TAL
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Hydrochlorothiazide
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Inhibits Na/Cl cotransporter in distal tubule
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Chlorothiazide
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Inhibits Na/Cl cotransporter in distal tubule
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Metolazone
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Inhibits Na/Cl cotransporter in distal tubule
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Indapamide
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Inhibits Na/Cl cotransporter in distal tubule
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Chlorthalidone
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Inhibits Na/Cl cotransporter in distal tubule
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Spironolactone
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Competitively inhibits the aldosterone receptor
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Eplerenone
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Competitively inhibits the aldosterone receptor
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Amiloride
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Blocks Na channels in principal cells
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Triamterene
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Blocks Na channels in principal cells
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Demeclocycline
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ADH antagonist
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Lithium
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ADH antagonist
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Tolvaptan
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Selective antagonist of vasopressin v2 receptor
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Mozavaptan
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Selective antagonist of vasopressin v2 receptor
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Lixivaptan
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Selective antagonist of vasopressin v2 receptor
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Conivaptan
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Antagonist of v1a and v2 vasopressin receptors
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Nifedipine
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Calcium channel antagonist |
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Diltiazem
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Calcium channel antagonist |
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Verapamil
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Calcium channel antagonist |
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Clonidine
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A2 agonist
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Guanfacine
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A2 agonist
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Methyldopa
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A2 agonist
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Reserpine
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Depletes monoamine from storage vesicles
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Phenoxybenzamine
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A blocker
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Prazosin
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A blocker
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Terazosin
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A1 blocker
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Doxazosin
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A1 blocker |
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Labetolol
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Mixed alpha/beta receptor antagonist
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Carvedilol
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Mixed alpha/beta receptor antagonist and NO generator
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Minoxidil
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Vasodilator
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Nitroprusside
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Vasodilator
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Lisinopril
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ACE inhibitor
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Nicardipine
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Calcium channel antagonist
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Amlodipine
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Calcium channel antagonist
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Ranolazine
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Inhibits fatty acid beta oxidation in cardiac myocyte mitochondria
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Isosorbide dinitrate
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NO donor, vasodilation
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Erythrityl tetranitrate
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NO donor, vasodilation
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Digoxin
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Partially inhibits Na/K atpase, increases SR calcium stores
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Irbesartan
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Angiotensin Receptor blocker
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Candesartan |
Angiotensin Receptor blocker
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Bucindolol
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B blocker |