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33 Cards in this Set
- Front
- Back
What are dugs that STIMULATE UTERINE contractions called?
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OXYTOCICS
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What are drugs that SUPPRESS Contractions called?
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TOCOLYTICS
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What are the 3 applications of OXYTOCIC drugs?
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1. INDUCTION/AUGMENTATION of labor
2. CONTROL Postpardum BLEEDING 3. INCUCE ABORTION |
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What is the ONE MAJOR use of TOCOLYTIC drugs?
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SUPPRESS PRETERM LABOR
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What are some TOCOLYTIC (uterine relaxants) drugs?
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-MG. SULFATE
-BETA2-SELECTIVE ADRENERGIC AGONIST(Ritodrin} -Terbutaline{Brethine} -NIFEDIPINE(procardia, adalat, nifedical) -Indomethacin (Indocin) |
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What is the treatment OF CHOICE to treat PREterm Labor?
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MG. SULFATE IV
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How does Mg. Sulfate work?
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Inhibits ACETYLCHOLINE RELEASE @ UTERINE NEUROMUSCULAR JUNCTION.
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What else is MG. SULFATE used for?
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PREFERRED for PREVENTION of TREATMENT of SEIZURES associated with ECLAMPSIA & PRE-ECLAMPSIA
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What should you ASSESS OFTEN if giving MG. SULFATE?
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RESPERATIONS
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What are some BETA2-SELECTIVE ADRENERGIC AGONIST?
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RITODRINE
TERBUTALINE(BRETHINE) |
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What are the affects of RITODRINE?
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It affects BETA CELLS, RELAXES uterus smooth muscles therby DECREASING Frequency and Intensity of contractions.
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What are the ADVERSE EFFECTS of RITODRINE?
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PULMONARY EDEMA, HYPOTENSTION, HYPERGLYCEMIA, TACHYCARDIA in FETUS.
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Which is better for the mother RITODRINE or MG. SULFATE?
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MG. SULFATE.
RITODRINE is as effective as MG. SULFATE but poses a MUCH greater risk on the mother. |
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What is TERBUTALINE(BRETHINE) used for? is it FDA approved?
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ASTHMA but used to delay preterm labor(NOT FDA approved)
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What is NIFEDIPINE? (procardia, adalat, nifedical) Whats it used for?
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CALCIUM CHANNEL BLOCKER--suppress PRETERM Labor
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What is INDOMETHICIN(INDOCIN) used for?
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-2nd line drug for SUPPRESSING PRETERM labor.
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When is INDOMETHICIN(INDOCIN) reserved for?
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WOMEN UNRESPONSIVE/INTOLERENT to preferred agents.
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What are OXYTOCIC used to do?
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STIMULATES uterine contractions, INDUCTION/Augmentation of labor, Control of POSTpartum bleeding, INDUCTION of ABORTION.
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What are TOCOLYTIC used for?
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SUPPRESS CONTRACTIONS, SUPPRESS PREtem labor.
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What are the drugs in the OXYTOCICS family?
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OXYTOCIN(PITOCIN),ERGOT ALKALOIDS(ergonovine&methlergonovine), CARBOPROST TROMETHAMINE(HEMABATE)
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what kind of hormone is OXYTOCIN(PITOCIN)? Where is OXYTOCIN(PITOCIN) produced?
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POLYPEPTIDE hormone produced by the POSTERIOR PITUITARY.
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What is OXYTOCIN(PITOCIN) used for?
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INDUCE labor, PROMOTE UTERINE CONTRACTIONS, MILK EJECTION, WATER RETENTION(similar to ADH)
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What women SHOULD NOT use OXYTOCIN(PITOCIN)?
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Women who have active GENITAL HERPES, uterine rupture possibility.
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What should you do if while taking OXYTOCIN(PITOCIN) contractions are >60sec.?
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DISCONTINUE!!
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What are the ADVERSE effects of taking OXYTOCIN(PITOCIN)?
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WATER INTOXICATION d/t anti diuretic affects.
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What are ERGOT ALKALOIDS(ergonovine&methylergonovine used for?
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POSTPARTUM BLEEDING, MIGRAINE,AUGMENTAION of labot(NOT recommended)
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What are teh ADVERSE effects of IV ERGOT ALKOLOIDS(ergonovine&methylergonovine)?
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HTN d/t constiction of arterioler & veins.
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What are ERGOT ALKALOIDS reserved for?
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HEMORRHAGIC EMERGENCIES.
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When in ERGONOVINE used?
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In the presence of BOGGY uterus & VAGINAL bleeding.
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What is the preferred agent used for controlling POSTPARTUM HEMORRHAGE?
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CARBOPROST THROMETHAMINE(hemabate)--causes INTENSE uterine contractions
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what are the ADVERSEeffects of CARBOPROST TROMETHAMINE(hemabate)
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GI reactions, V&D, Fever, Vasoconstrition, Constriction of Bronchi.
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What is DINOPROSTONE(Prepidil/Ceridil) used for?
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Promote Cervical Ripining BEFORE INDUCTION of labor w/ Oxytocin(Pitocin).
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What are the 3 different types of DINOPROSTONE(prepidil/Cervidil)?
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DINOPROSTONE GEL
DINOPROSTONE VAGINAL INSERTS(cervidil) MISOPROSTOL(cytotec)-NOT APPROVED for CERVICAL RIPENING |