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173 Cards in this Set
- Front
- Back
HTN drugs
|
-sympatholytics
-ACEI's -ARB's -diurectics -Ca2+ channel blockers -vasodilators |
|
Sympatholytics
|
-b-blockers
-a1 antagonists |
|
B-blockers
|
-pindolol
-carteolol -labetalol -celiprolol -nebivolol |
|
b-blockers: non B selective, MSA, increased lipid solubility
|
propanolol
|
|
b-blockers: cardioselective
|
-metoprolol
-bisoprolol -acebutolol |
|
b-blockers: cardioselective, decreased lipid solubility
|
atenolol
|
|
b-blockers: a1/b selective
|
carvedilol
|
|
a1-antagonists
|
-doxazosin
-tetrazosin |
|
a1-antagonist: prostate hyperplasia
|
-tamusulosin
-alfuzosin |
|
alpha 2 agonists
|
-clonidine
-a-methyldopa -moxonidine |
|
alpah 2 agonists: glaucoma
|
-aproclonidine
-bromonidine |
|
ACEI's
|
-lisonopril
-captopril -quinapril -enalapril -ramipril -benazepril -fosinopril |
|
AT1 receptor antagonists (ARB's)
|
-losartan
-irbesartan -valsartan -candesartan -olmesartan -telmisartan |
|
renin inhibitors
|
aliskiren
|
|
Diuretics
|
-thiazide diuretics
-loop diuretics -K-sparing diuretics |
|
Thiazide diuretics
|
-chlorothiazide
-hydrochlorothiazide -chlorthalidone -bendroflumethiazide -metolazone -indapamide |
|
Loop Diuretics
|
-furosemid
-torsemide -ethacrynic acid -bumetanide |
|
K-sparing Diuretics: Na channel blocker
|
-triamterine
-amiloride |
|
K-sparing diuretics: aldosterone antagonists
|
-spironolactone
-eplernone -drospirenone |
|
Vasodilators
|
-calcium channel blockers
-nitrates -K+ channel openers |
|
Direct Vasodilators
|
-nitrates
-K+ channel openers |
|
Calcium channel blockers
|
-nifedipine
-amlodipine -felodipine -nisoldipine -verapamil -diltiazem |
|
direct vasodilator alternatives
|
-hydralazine
-sodium nitroprusside -minoxidil |
|
Angina Pectoris Drugs
|
-Nitrates
-Ca2 channel Blockers -Inhibitors of platelet aggregation -Beta blockers -Novel channel blockers -Thrombin modulators -Other |
|
Congestive Heart Failure Drugs
|
-ACEI's
-Beta Blockers -Cardiac Glycosides -PDEI's -Beta1 adrenoceptor agonists -Vasodilators -Diuretics |
|
Arrhythima Drugs
|
-Fast Na Channels inhibitors (membrane stabilizers)
-Beta Blockers -Prolong action potential duration -Nonselective Ca2 channel blockers -Cardiac glycosides -Other |
|
Angina Pectoris: Nitrates
|
-NO
-isosorbide dinitrate -nitroglycerin -sodium nitroprusside -micorandil |
|
Angina Pectoris: Ca2+ Channel Blcokers
|
-amlodipine
-nifedipine -felodipine -verpamil -diltiazem |
|
Angina Pectoris: Beta Blockers
|
-propranolol
|
|
Angina Pectoris: Inhibitors of platelet aggregation
|
-aspirin
-clopidogrel -glycoprotein IIB/IIIA |
|
Angina Pectoris: Thrombin modulators
|
-heparin
-warfarin |
|
-Angina Pectoris: Other
|
-morphine
-tx hypercholesteremia, hypertension |
|
CCF: ACEI's
|
?
|
|
CCF: Beta Blockers
|
-carvedilol
-metiprolol -bisoprolol -nebivolol |
|
CCF: cardiac glycosides
|
-digoxin
-digitoxin |
|
CCF: PDEI's
|
-amrinone
-vesnarinone |
|
CCF: Beta1 agonists
|
-dobutamine
|
|
CCF: vasodilators
|
-nitrovasodilators
-hydralazine |
|
CCF: nitrovasodilators
|
-sodium nitroprusside
-isosorbide dinitrate -nitroglycerin |
|
CCF: diurectics
|
?
|
|
Arrythmias: Fast Na channel inhibitors
|
-quinidine
-procainamide -disopyramide -lidocaine -flecainide -propafenone |
|
Arrythmias: Beta blockers
|
-propanolol
-solalol |
|
Arrythmias: prolong action potential
|
-amiodarone
-dronedarone -dofetilide -sotalol -ibutilide |
|
Arrythmias: Nonselective CA2+ channel blockers
|
-verapamil
-diltiazem |
|
-Arrythmias: cardiac glycosides
|
-verampil
-beta blockers |
|
-arrythmia: new drugs
|
-ivabradine
-adenosine -potassium |
|
Ophthalmic (topical) corticosteroids
|
-prednisolone
-dexamethasone -fluorometholone -rimexolone -loteprednol -medrysone |
|
Systemic Corticosteroids
|
-dexamethasone
-prednisolone -hydrocortisone -tramcinolone -fluticasone -mometasone -bethamethasone -budesonide -flucinolone -disonide |
|
Diagnostic Dyes
|
-fluorescein (fluorexon)
-rose bengal -lissamine green B -indocyanine green -trypan blue |
|
DMARDs
|
-methotrexate
-sulfasalazine -chloroquine derivatives -cyclophosphamide -azathioprine -leflunomide -inliximab/etanercept -sirolimus (rapamycin) -calcineuron inhibitors -daclizumab -anakinra |
|
Major subgroups of anti-inflammatory drugs
|
-NSAIDs
-corticosteroids -SAARDs -DMARDs |
|
Immunosuppressants: cytotoxic/antimetabolites/small molecules
|
-cyclophosphamide
-leflunomide -methotrexate -azathioprine -colchicine |
|
Immunosuppressants: immune modulators
|
-calcineuron
-sirolimus -infliximab -daclizumab |
|
Systemic immunosuppressants: uveitis
|
-azathiprine
-methotrexate -cyclosporine -daclizumab -infliximab |
|
systemic immunosuppressants: cicatricia pemphigoid
|
-dapson
-azathioprine -cyclophosphamide |
|
topical immunosuppressants: corneal ulcers
|
-galardin
|
|
systemic immunosuppressants: behcet syndrome
|
-chlorambucil
-cochicine |
|
osteoporosis drugs
|
-alendronate
-chondroitin -glucosamine |
|
Gout drugs
|
-uricosuric agents
-metabolic inhibitors -cochicine -NSAIDs -steroids |
|
Gout: metabolic inhibitors
|
allopurinol
|
|
Gout: uricosuric agents
|
-probenacid
-sulfinpyrazone -high dose aspirin |
|
Asthma Drugs
|
-Bronchodilators
-anti inflammatory drugs -allergic component Tx -other |
|
Asthma: bronchodilators
|
-beta2 agonists
-non selective beta agonists -non selective alpha/beta agonists -PDEI's -anti muscarinics |
|
Asthma: anti-inflammatory drugs
|
-inhaled coritcosteroids
-leukotriene antagonists |
|
Asthma: allergic component Tx
|
-mast cell stabilizers
-anti-histamines -anti-IgE monoclonal antibodies: omalizumab -acupuncture |
|
Asthma: other drugs
|
-treat symptoms: cough/sore throat/runny nose
|
|
Bronchodilators: beta2 agonists
|
-albuterol
-terbutaline -salmeterol -pirbuterol -fometerol |
|
Bronchodilators: non selective beta agonists
|
-isoproterenol
|
|
Bronchodilators: non selective alpha/beta agonists
|
-ephedrine
-epinephrine |
|
Bronchodilators: PDEI's
|
-theophlylline
-oxtriphylline -aminophylline -3-prophylxanthine |
|
Bronchodilators: anti-muscarinics
|
-ipratropium bromide
-tiotropium |
|
Anti-inflammatory: Steroids
|
-beclomethasone
-triamcinolone -fluticasone -mometasone -flunisolide -budesonide -dexamethasone -prednisolone -ciclesonide |
|
Anti-inflammatory: Leukotriene antagonists
|
-montelukast
-zafrilukast -pranlukast -zileuton |
|
Treating allergic component of asthma
|
-mast cell stabilizers
-anti-histamines -immunotherapy -anti-IgE monoclonal antibodies -acupuncture |
|
Anti-IgE monoclonal Antibodies
|
omalizumab
|
|
Cystic fibrosis Drugs
|
-amiloride
-expectorants -mucolytics -Antibodies -DNAases -targeted gene therapy |
|
treatments for COPD mucus/cough
|
-decongestants
-mucolytic agents -expectorants -cough suppressants (anti-tussive) -analgesics and antipyretics -loop diuretics -gene therapy |
|
COPD: decongestants
|
-oxymetazoline
-phenylephrine -xylometazoline -pseudophredrine -ephedrine -methol/vapor tx |
|
COPD: mucolytic agents
|
-acetylcysteine
-brombexine |
|
COPD: expectorants
|
-licorice
-ammonium salts -guaniphenesin -guaicacolsulphate -eucalyptus oil |
|
COPD: cough suppressants
|
-codeine
-dihydrocodone -dexatromethorphan -menthol/vapor tx |
|
COPD: analgesics and antipyretics
|
-codiene
-aspirin and other salicylates -ibuprofen |
|
Angina: novel channel blockers
|
-Ivarbadine
-ranolazine |
|
principal CNS nt's
|
-gluatmate
-GABA |
|
Classicnt's
|
-Ach
-DA -5-HT -NE |
|
Anti-anxiety drugs
|
-benzodiazepines
-buspirone -antidepressants (TCA's, SSRI's, MAIO's) -beta blockers |
|
Benzodiazepines
|
-diazepam
-temazepam -oxazepam -lorazepam -triazolam |
|
Depression drugs
|
-TCA's
-SSRI's -MAOI's |
|
TCA's
|
-impiramine
-amitriptyline -nortiptyline |
|
SSRI's/SNRI's
|
-fluoxetine
-fluvoxamine -sertraline -citalopram -praoxetine +anit mus -venlafaxine +NE -nefazodone (inhibits 5-HT2) |
|
MAOI's - nonselective
|
-phenelzine
|
|
MAOI's - selective
|
-moclobemide
|
|
Other therapies for depression
|
-light
-st john's wort -ECT/TMS -combo drugs for mixed disorders |
|
mania and bipolar drugs
|
-lithium
-carbamazepine -valproate |
|
schizophrenia drugs
|
-phenothiazine
-butyrophenones -thioxanthenes -atypical |
|
-phenothiazines
|
-chlorpromazine
-thiroridazine -prochlorperazine |
|
vutyrophenones
|
-haloperidol
|
|
-thioxanthenes
|
-flupentixol
|
|
-atypical schizo drugs
|
-risperidone
-clozapine -olanzapine |
|
anti-perkinson's drugs
|
-reverse DA defiency/increase DA activity
-antimuscarinic |
|
-parkinson's - reverse DA deficiency
|
-DA precursor
-DOPA decarboxylase -MAO-B -COMT 1 -DA agonists -increase release/uptake inhibiors |
|
DA precursor
|
-levodopa
|
|
DOPA decarboxylase i
|
-carbidopa
-benserazide |
|
Parkinson's - MAO-B I
|
-selegiline
|
|
Parkinson's - COMT I
|
-entacopone
-tolcapone |
|
Parkinson's - DA agonists
|
-apomorphine
-bromocryptine -pergolide |
|
Parkinson's - Increase release/uptake inhibitor
|
-amantidine
|
|
Parkinson's - antimuscarinics
|
-benztropine
-trihexyphenidyl HCl |
|
Anti - epiliepsy drugs
|
-carbamazepine
-phenytoin -lamotrigine -valproate/divalproex -gabapentin -ethosuximide -topiramate -vigabatrin -clonazepam (BZ) -clozabam (BZ) |
|
Alzheimer's drugs
|
-cholinesterase inhibitors
-memantine |
|
Cholinesterase inhibitors
|
-donepezil
-rivastigmine -galantamine |
|
ADHD drugs
|
-stimulants
-misc non stimulative |
|
ADHD - stimulants
|
-dextroamphetamine
-methamphetamine -dextroamphetamine/amphetamine -dextromethylphenidate |
|
ADHD misc
|
-atomoxetine
-buproprion -guanfacine -clonidine |
|
Autistic spectrum disorders drugs
|
-risperidone
-methylphenidate (ritalin, concerta) |
|
Jet lag drugs
|
-melatonin
-short acting hypnotics -stimulants (narcolepsy) |
|
Jet lag - short acting hypnotics
|
-triazolam
-zolpidem -zalepion |
|
Jet lag - stimulants
|
-caffiene
-armodafinil |
|
Acid-peptic drugs
|
-neutralize acid
-reduce acid secretion -protect tissue -enhance cytoprotective mechanism -eradicate heiobactor pylori |
|
Acid peptic - neutralize acid
|
-antacid
|
|
Acid peptic - reduce acid secretion
|
-anticholinergics
-H2 receptor antagnoists -proton pump inhibitors -prostaglandins |
|
Acid peptic - protect tissue
|
-bismuth
-sucralfate |
|
Acid peptic - enhance cytoprotective mechanism
|
-prostaglandins (misoprostol)
|
|
acid peptic - Antacids
|
-Systemic: NaHCO3
-Nonsystemic |
|
Antacids - non systemic
|
-CaCO3
-Mg(OH)2 -Al(OH)2 |
|
Acid-peptic - anticholinergics (M1 antagonists)
|
-pirenziepine
-telenezepine |
|
Acid-peptic - eradicate helicobacter pylori
|
-antibiotics
|
|
Acid-peptic: misc
|
-metoclopramide
|
|
Diarrhea drugs
|
-opiates
-bismuth subsalicylate (pepto) -kaolin and pectin |
|
diarrhea - opiates
|
-diphenoxylate
-leoperamide |
|
Lipid drugs
|
-statins
-fibrates -bile acid binding resin -ezetimibe -niacin |
|
lipid drugs - statins
|
-atorvastatin
-simvastatin -fluvastatin -lovastatin -rosuvastatin |
|
lipid drugs - fibrates
|
-gemfibrozil
-fenofibrate |
|
lipid drugs - bile acid
|
-cholestyramine
-colestipol |
|
Rapid acting insulins
|
-insulin lispro
-insulin aspart -insulin glusisine |
|
Short acting insulins
|
-velosulin (pump)
-Regular |
|
Intermediate acting insulins
|
-NPH
-lente |
|
Premixed insulins
|
-novolin
-humulin -50/50 NPL, lispro -75/25 NPL, lispro -70/30 NPA, aspart |
|
Long acting insulins
|
-insulin detemir
-insulin glargine |
|
Oral antidiabetic (type II)
|
-insulin secretagoues
-biguanides -thizaolidediones -alpha - glucosidase inhibitors |
|
Oral antidiabetics: insulin secretagogues
|
-sulfonylurea
-meglitinides -D-phenylalanine derivatives |
|
Oral antidiabetics: Thiazolidinediones
|
-Tzd's
-PPAR alpha agonists -rosiglitazone -pioglitazone |
|
Insulin secretagogues: sulfonylureas
|
-tolbutamide
-chlorpropamide -tolazamide -glyburide -glipizide -glimepiride |
|
Insulin secretagogues: Meglitinides
|
-repaglinide
|
|
Biguanides
|
-metformin
-phenoformin |
|
Alpha-glucosidase inhibitors
|
-acarbose
-miglitol |
|
Other diabetes options
|
-pramlintide
-exenatide -glucagon |
|
Topical LA's
|
-beoxinate
-proparacaine -tetracaine -cocaine |
|
Cornea/ Conj problem herbs
|
-cocaine
-chamomile -echinacea |
|
Dry eyes problem herbs
|
-datura
-vitamin A analogs |
|
Mydriasis problem herbs
|
-datura
-cocaine -crystal meth -methylphenidate -ecstacy -marijauna -deadly nightshade |
|
Miosis problem herbs
|
-heroin
|
|
Ciliary muscle/acc problem herbs
|
-datura
-marijuana -insecticides? |
|
EOM problem herbs
|
-cocaine
-crystal meth -marijuana -additives to injectibles |
|
IOP problem herbs
|
-datura
-marijuana -alcohol |
|
Other problem herbs
|
-ecstacy and lsd
-ginkgo -licorice -canthaxanthine echinacea pupurea -niacin |
|
Color vision problem herbs
|
-marijuana
-cocaine -heroin |
|
Cornea problem systemic drugs
|
-crack
-rifabutin -amiodarone -chloroquine -chlorpromazine -tamoxifen |
|
Lens problem systemic drugs
|
-phenathiazines
-SSRI's -steroids |
|
dry eye problem systemic drugs
|
-anti-muscarinic ->depression drugs
-beta blockers -vitamin A analogs -HRT (BCP) -antihistamines -diuretics |
|
Mydriasis problem systemic drugs
|
-CNS drugs (stimulants and depressants)
-antimuscarinics |
|
Miosis problem systemic drugs
|
-opioids
-Achesterase inhibitors -insecticides |
|
floppy iris problem systemic drugs
|
-alpha adrenergic blockers
-tamsulosin |
|
EOM problem systemic drugs
|
-neuraleptics
-anti-epileptic -BZ drugs -lithium -antihistamines |
|
Retina problem systemic drugs
|
-chloroquine
-digoxin -vigabatrin -orobronze (canthaxanthine) -talc retinopathy -cisplatin -steroids -tamoxifen |
|
Optic nerve problem systemic drugs
|
-retinoids
-chloroquine -amiodarone -steroids -clyclosporine -ethambutol -isoniazid -sildenafil -tamoxifen |
|
IOP problem systemic drugs
|
-steroids
-antimuscarinics -beta blockers -alpha 2 agonists -prostaglandins |
|
cycloplegia problem systemic drugs
|
-antimuscarinics
|
|
Myopia problem systemic drugs
|
-elevated IOP
|
|
Conj/Lids problem systemic durgs
|
-xenobiotic - photocopying carbon
-bimatoprost |
|
Leber's Congenital Amaurosis
|
-AAV-RPE65
|
|
Age related macular degeneration
|
-AAV-sFLT01
|
|
First generation optical neuromodulators
|
-ChR2
-NpHR |