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111 Cards in this Set

  • Front
  • Back
Midazolam
short acting benzo
Zolpidem
treat insomia (but not muscle relaxant)
Buspirone
5HT1a partial agonist. Anxiolytic.
B carboline
MAO-I
Alprazolam
benzo; treat agoraphobia
Diazapam
benzo
Phenytoin
stabilizes inactive state of Na channels. saturation of the liver cuases it to go from 1st to 0 order pharmacokinetics
Carbamazepine
mood stabilizer and anti convulsant, same mechanism of phenytoin
Gabapentin
mimics GABA
Lorazepam
benzo. treat status epilepticus. Prevents EtOH withdrawl
Vaproic Acid
used to treat absence and partial sezures
Modafinil
promotes awakeness
Flumazenil
benzo antagonist
Thiopental
short acting barbituate
L-Name
inhibitor of NO synthase
Atropine
competitive muscarinic antagonist
Physostigmine
reversible ChE-I
Bethanechol
muscarinic agonist, ChE resistant
Hexamethonium
Nn antagonist
Pilocarpine
muscarinic agonist, can treat glaucoma
Neostigmine
ChE-I, can treat glaucoma
Atenolol
B1 blocker
Prazosin
Reversible A1 antagonist. Lowers BP while increasing HR.
Propranolol
B1/B2 antagonist
Phenylephrine
A1 agonist
Dobutamine
B1 agonist
Tolazoline
reversible A antagonist
Phentolamine
reversible A antagonist
Phenoxybenzamine
irreversible A antagonist
Tamsulosin
A1 antagonist. Used to treat benign hypertrophy of prostate
Memantine
AZ dz drug that blocks NMDA-glutamate receptors
Fluoxetine
SSRI
Imipramine
TCA
Tranylcypromine
MAO-I, contraindicated with decongestants, meperidine
Bupropion
atypical anti-D
Halothane
produces decrease in CO and BP
Etomidate
GABA anesthetic
Isoflurane
can cuase MI or resp irritation
Ketamine
NMDA receptor antagonist, dissociative anesthesia. Bind u and sigma opiod receptors
Fluvoxamine
SSRI
Phenelzine
MAOI
Venlafaxine
SNRI
Citalopram
SSRI
Sertraline
SSRI
Sibutramine
oral anorexiant
Propofol
hypnotic/anesthetic. Short acting
Ropinirole
non-ergot DA agonist
Benztropine
anticholinergic
Selegiline
MAOb-I
Nefazadone
5HT2 antagonist
Fomepizole
CAD inhibitor. Antidote to methanol and ethylene glycol poisoning
Phencyclidine
PCP
Curare
nicotinic antagonist
Hemicholinum
blocks choline transporter
Vseamicol
blocks entry of Ach into secretory granule
Trimethaphan
Ach antagonist
Novibol
B1 antagonist
Pindolol
partial agonist on B1 and B2
Bradykinin
ACE inhibitor
Chlorpromazine
antagonist for A1, A2, H1, 5HT2a, D1, D2, M1
Ondansetron
5HT3 antagonist and anti-emetic
Haloperidol
D2 antagonist
Pirenzepine
M1 antagonist
Telenzepine
M1 antagonist
Edrophonium
short acting ChE-I
Organophosphates
irreversible ChE-I
Baclofen
GABA agonist used spinal cord injury leading to spasticity.
Dantrolene
inhibits Ca++ from sarcoplasmic reticulum. Liver tox risk. Used to treat malignant hyperthermia
Chlorpromazine
D2 antagonist
Thioridazine
D2 antagonist
Fluphenazine
D2 antagonist
Haloperidol
D2 antagonist
Risperidone
D2 and 5HT2a antagonist
Paliperidone
D2 and 5HT2a antagonist
Clozapine
D2 and 5HT2a antagonist
Olanzapine
D2 and 5HT2a antagonist
Quetiapine
D2 and 5HT2a antagonist
Ziprasidone
D2 and 5HT2a antagonist
Aripiprazole
D2 and 5HT2a antagonist
Bromocriptine
DA agonist, ergot
Pergolide
DA agonist, ergot
Pramipexole
DA agonist, non ergot
Ropinirole
DA agonist, non ergot
Apormorphine
DA agonist, non ergot
Trihexiphenidyl
anti - M
Diphenhydramine
anti - M
Stalevo
entacopone, carbidopa, L DOPA
Valproic Acid
affects Na channels, inhibits GABA-T, blocks T-type Ca++ channels; causes alopecia
Zaleplon
Sonata, benzo, BDZ1-R
Solpidem
Ambien, benzo, BDZ1-R
Eszoiclone
Lunesta, benzo, BDZ1-R
Naloxone
opioid antagonist
Naltrexone
opioid antagonist
Nalmefene
opioid antagonist
Tramadol
mu receptor agonist, inhibitor of 5HT and NE reuptake
Pentazocine
kappa agonist, mu antagonist
Nalbuphine
kappa agonist, mu antagonist
Buprenorphine
kappa agonist, mu antagonist
Butorphanol
kappa agonist, mu antagonist
Mirtazapine
A2 and 5HT2a antagonist
Trazadone
5HT2A antagonist
Isocarboxazide
MAO-I
Droperidol
anti emetic.
Cimedtidine
H2 antagonist
Ranitidine
H2 antagonist
Famotidine
H2 antagonist
Metoclopramide
prokinetic
Disulfiram
inhibits acetaldehyde dehydrogenase
Acamprostate
inhibit NMDA glutamate recetpors.
Anandamide
endocannabinoid
Rimonobant
CB1 antagonist. Devo to treat obesity.