Reading...
Play button
Play button
Use LEFT and RIGHT arrow keys to navigate between flashcards;
Use UP and DOWN arrow keys to flip the card;
H to show hint;
A reads text to speech;
10 Cards in this Set
- Front
- Back
|
Morphine
|
Strong Full Agonist
MS Contin, Kadian High affinity for Mu receptor |
|
|
Hydromorphone
|
Strong Full Agonist
Dilaudid |
|
|
Oxycodone
|
Strong Full Agonist
Oxycontin |
|
|
Methadone
|
Dolophine
Strong Full Agonist Most often used to treat addiction, sometimes used for severe pain NMDA antagonist and blocks SERT and NET T 1/2 = 8-59 hours. |
|
|
Fentanyl
|
Duragesic, Sublimaze
Strong Full Agonist |
|
|
Levorphanol
|
Levo Dromoran
Strong Full Agonist T 1/2 = 12-15 hours May block NMDA receptor Used in neuropathic pain. |
|
|
Meperidine
|
Demerol
Strong Full Agonist Less potent than morphine. Rapid onset, short duration. (T1/2 = 3 hours) Neurotoxic metabolite - normeperidine that is not reversed by naloxone! |
|
|
Hydrocodone
|
Vicodin, Lortab, Lorcet
Mild to Moderate Full Agonist In combo with APAP (N-acetyl-para-aminophenol) |
|
|
Codeine
|
Weak Mu receptor agonist
Low analgesic potency, low ceiling. Possess anti-tussive activity. |
|
|
Propoxyphene
|
Darvon, Darvon N, Darvocet
Mild to Moderate Full Agonist Low analgesic activity (1/2 as potent as codeine) Neurotoxic metabolite - norpropoxyphene |
