Neurotransmitter Receptor Agonists And Antagonists

Front 1

Acetylocholine ionotropic receptor agonists

Back 1

Nicotinic

Front 2

Acetylcholine metabotropic receptor agonists

Back 2

Muscarinic

Front 3

Acetylcholine Ionotropic/nicotinic receptor antagonists

Back 3

decamethonium (partial agonists)
succinylcholine (partial agonists)

Front 4

Acetylcholine metabotropic/muscarinic receptor antagonists

Back 4

Atropine
pirenzepine
AF-DX 116

Front 5

Glutamate ionotropic receptor subcategories

Back 5

NMDA
AMPA
Kainate

Front 6

Glutamate receptor agonists

Back 6

NMDA
AMPA
Kainate

Front 7

Glutamate receptor antagonist

Back 7

APV
CNQX

Front 8

GABA receptor agonists

Back 8

GABA

Front 9

GABA receptor antagonists

Back 9

picrotoxin
Bicuculline

Front 10

Barbituate/steroid effect of GABA receptor

Back 10

increases conductance of chlorine even without GABA bound

Front 11

Benzodiazapine

Back 11

Increases effect of GABA.

Front 12

Open channel blocker

Back 12

PCP - Glutamate Channel

Front 13

Glycine Agonist

Back 13

Glycine

Front 14

glycine agonist

Back 14

glycine
Ethanol

Front 15

Nucleotide and cyclic nucleotides agonist

Back 15

adenosine

Front 16

Nucleotide antagonist

Back 16

caffeine

Front 17

Caffeine prevents__________ of _______ ________ producing the same effect as

Back 17

inhibition of inhibitory receptors
strychnine

Front 18

Glycine antagonist

Back 18

strychnine

Front 19

Glycine precursor

Back 19

serine

Front 20

Acetylcholine precursor

Back 20

acetyl CoA and choline

Front 21

Glutamate precursor

Back 21

glutamine

Front 22

GABA precursor is

Back 22

bicuculine

Front 23

Nucleotide/cyclic nucleotide precursor is

Back 23

ATP

Front 24

Catecholamine neurotransmitters

Back 24

Dopamine
Epinephrine
Norepinephrine
Serotonin

Front 25

Dopmine agonist

Back 25

Dopamine
Cocaine
Morphine
MPTP

Front 26

Dopamine antagonist

Back 26

Haldol
Thorazine

Front 27

Haldol and Thorazine are

Back 27

sedatives

Front 28

Dopamine precursor is

Back 28

tyrosine

Front 29

Epinephrine agonist is

Back 29

ephedrine

Front 30

Ephedrine is

Back 30

source of methamphetamines which are stimulants

Front 31

Epinephrine antagonists are

Back 31

B blockers - block the B form of receptors in heart

Front 32

Epinephrine precursor is

Back 32

tyrosine to dopamine

Front 33

Norepinephrine agonist

Back 33

Welbutrin

Front 34

Norepinephrine antagonist for brain

Back 34

Pb and Hg

Front 35

Norepinephrine precursor is

Back 35

tyrosine to dopamine to epinephrine to norepinephrine

Front 36

Serotonin is a

Back 36

biogenic amine

Front 37

Loss of serotonin leads to

Back 37

depression

Front 38

Serotonin agonist is

Back 38

Buspar - Prozac

Front 39

Serotonin antagonist is _______ which blocks

Back 39

Phen-Phen
reward sensation of eating food

Front 40

Neuropeptides include

Back 40

endorphins
anandamides

Front 41

Endorphin means

Back 41

endogenous morphine

Front 42

We found the ________ _______ before we found ________.

Back 42

endorphin receptor
endorphin

Front 43

Endorphin agonist is

Back 43

opium

Front 44

Anandamides bind

Back 44

endogenous cannabinoid receptor

Front 45

Adenosine receptors are bound antagonistically by

Back 45

xanthines
caffeine
theophylline

Front 46

Theophylline is the precursor for

Back 46

theobromine in chocolate

Front 47

Theobromine binds ___________ along with ________

Back 47

love receptors
caffeine

Front 48

Dopamine activates __________ and acts as a ___________

Back 48

motor control
stimulant

Front 49

Epinephrine will bind

Back 49

specific adenergic receptors

Front 50

amphetamines will bind

Back 50

all catecholamine or serotonine receptors

Front 51

Methamphetamine binds

Back 51

all seratonergic, dopanergic, peinergic, and norepinergic receptors

Front 52

Benzedrine binds _________

Back 52

adrenergic beta epinergic receptors

Front 53

Amphetamine not only binds ________ and _______. But also binds

Back 53

epinergic and dopanergic receptors,
presynaptic reuptake receptors

Front 54

Amphetamine preferentially binds

Back 54

dopamine receptors

Front 55

Methamphetamine binds

Back 55

dopanergic, epinergic, norepinergic and seronergic receptors

Front 56

Cocaine reverses flow of

Back 56

presynaptic receptor

Front 57

Pharmaceutical grade amphetamines bind

Back 57

specific receptors because of manufacturing control of chiral carbons

Front 58

Street drugs bind

Back 58

all receptors because of various forms of chiral carbons

Front 59

Cocaine binds ________ and ________

Back 59

epinephrine, dopamine (preferentially) and serotenergic reuptake receptors causing uncontrolled dopamine release

Front 60

Amphetamines

Back 60

activate adrenergic receptors in the PNS

Front 61

Adderall chemical name

Back 61

dextroamphetamine

Front 62

Benzodiazapines for _________ receptors

Back 62

Xanax
Rohypnol
Valium
GABA

Front 63

Barbituates for _________ receptors

Back 63

Seconal
Nembutal

Front 64

COMT:

Back 64

Catechol-O-Methyl Transferase

Front 65

MAO

Back 65

Mono Amine Oxidases

Front 66

MAO's have _____ subtypes based on ______ _______ they affect

Back 66

2
Neurotransmitter
MAO-A and MAO-B

Front 67

First generation antidepressants

Back 67

Phenelzine (Nardil)
Isocarboxazide (Marplan)

Front 68

Nardil

Back 68

anti-depressant
anti-anxiety
anti-phobic

Front 69

marplan

Back 69

anti-depressant but also affects GABA

Front 70

Second Generation antidepressants

Back 70

Tofranil
Norpramin

Front 71

Third Generation Antidepressants

Back 71

Prozac
Zoloft
Cypramil
Paxil

Front 72

The serotonin binding site includes

Back 72

an ionic site, and polar ring site, and a polar site

Front 73

COMT can break down ________ without reducing the amount of _________

Back 73

dopamine
norepinephrine

Front 74

First generation anti-depressants were _____ ____ and affected the

Back 74

MAO inhibitors
Norepinephrine pathways

Front 75

First generation anti-depressants also affected the

Back 75

GABA reversing effect - inhibiting pathways.

Front 76

Second generation antidepressants increased ______, and decreased

Back 76

release of norepinephrine,
reuptake of norepinephrine

Front 77

Third generation anti-depressants affect

Back 77

Serotonin reputake receptors

Front 78

Prozac dosage has to be

Back 78

increased over time because of new receptors being produced

Front 79

Hallucinogens bind

Back 79

serotonin receptors better than serotonin

Front 80

When we first wake our serotonin levels are at their

Back 80

lowest

Front 81

Serotonin is also important in

Back 81

wakefullness

Front 82

These compounds bridge the gap between consciousness and unconsiousness

Back 82

Serotonin, Mescaline, Lysergic Acid, and Psilocybin

Front 83

THC causes

Back 83

retrograde inhibition of Ca++ pathway

Front 84

Endocannabinoids affect the

Back 84

pain pathway