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126 Cards in this Set

  • Front
  • Back
Bupivacaine
Local anesthetic
amide
Lidocaine
Local anesthetic
amide
Ropivacaine
Local anesthetic
amide
Chloroprocaine
Local anesthetic
ester
Procaine
Local anesthetic
ester
Tetracaine
Local anesthetic
ester

long acting
subarachnoid use?
Cocaine
Local anesthetic
Benzoic Acid Ester
Benzocaine
Local anesthetic
Non-ester

topical use (except eye)
Tetrodotoxin
(TTX)
Local anesthetic
Toxin/tool
Acetylcholine
Muscarinic Cholinergic Agonist
Nicotinic Cholinergic Agonist
M = N
Bethanechol
Muscarinic Cholinergic Agonist
M > N - doesnt activate muscles

-used for atony/urinary retention in bladder
-treatment for GERD
Pilocarpine
Muscarinic Cholinergic Agonist
Carbamylcholine
Muscarinic Cholinergic Agonist
N > M
Atracurium
Nicotinic NMBA
Cholinergic Antagonist

intermediate acting
histamine release
Mivacurium
Nicotinic NMBA
Cholinergic Antagonist
Pancuronium
Nicotinic NMBA
Cholinergic Antagonist
Rocuronium
Nicotinic NMBA
Cholinergic Antagonist
Succinylcholine
Nicotinic NMBA
Cholinergic Antagonist
d-Tubocurarine
Nicotinic NMBA
Cholinergic Antagonist
Vecuronium
Nicotinic NMBA
Cholinergic Antagonist
Varenicline
Nicotinic - central
Cholinergic Antagonist

*smoking cessation*
Bupropion
Nicotinic - central
Cholinergic Antagonist

= wellbutrin
*smoking cessation*
Pirenzapine
Muscarinic - M1
Cholinergic Antagonist
Trihexyphenidyl
Muscarinic - M1
Cholinergic Antagonist
Darifenacin
Muscarinic - M3
Cholinergic Antagonist
Tolteridine
Muscarinic - M3
Cholinergic Antagonist
Atropine
non-specific muscarinic
Cholinergic Antagonist
Benztropine
non-specific muscarinic
Cholinergic Antagonist
Cyclopentolate
non-specific muscarinic
Cholinergic Antagonist
Glyccopyrrolate
non-specific muscarinic
Cholinergic Antagonist
Ipratropium
non-specific muscarinic
Cholinergic Antagonist

GI or GU use
Scopolamine
non-specific muscarinic
Cholinergic Antagonist

ophthalmologic use
GI, GU use
Tropicamide
non-specific muscarinic
Cholinergic Antagonist

ophthalmologic use
Tiotropium
M1/M3 muscarinic
Cholinergic Antagonist
Edrophonium
Ionic Anti-ChE
Neostigmine
Carbamate Anti-ChE

uses:
-MG
atony of bladder

- can cause cholinergic crisis
Pyridostigmine
Carbamate Anti-ChE
Physostigmine
Carbamate Anti-ChE
Carbaryl
Carbamate Anti-ChE
Velnacrine
Carbamate Anti-ChE

Alzheimers treatment
Tacrine
Noncarbamate Anti-ChE
Diazinon
OP Anti-ChE
Malathion
OP Anti-ChE
Parathion
OP Anti-ChE
Sarin (GA)
OP Anti-ChE
Soman(GB)
OP Anti-ChE
nerve gas
Tabun (GD)
OP Anti-ChE
nerve gas
VX
OP Anti-ChE
nerve gas
Pralidoxime
AChE reactivators
Antibiotics
- aminoglycosides
- tetracyclines
distruptors of cholinergic transmission
- amikacin, gentamicin, kanamycin
- doxycycline, tetracycline
Norepinephrine
Sympathomimetic amine
- catecholamine
- A1,2; B1
Epinephrine
Sympathomimetic amine
- catecholamine
- A1,2; B1,2
Isoproterenol
Sympathomimetic amine
- catecholamine
- B1,2
Dopamine
Sympathomimetic amine
- catecholamine
- D1 - renal dose
Dobutamine
Sympathomimetic amine
- catecholamine
- B1
Tyramine
Sympathomimetic amine
- Non-catecholamine
- Indirect-acting (NE-releaser)
Amphetamine
Sympathomimetic amine
- Non-catecholamine
- Indirect-acting (NE-releaser)
Ephedrine
Sympathomimetic amine
- Non-catecholamine
- Indirect-acting (NE-releaser)
Cocaine
Sympathomimetic amine
- Non-catecholamine
- NE/DA uptake blocker
Methoxamine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- A1 agonist
Phenylephrine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- A1 agonist
Clonidine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- A2 agonist
Brimonidine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- A2 agonist

- ophthalmic
Fenoldopam
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- D1 agonist
Albuterol
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- B2 agonist
Ritodrine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- B2 agonist
Salmeterol
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- B2 agonist
Ergonovine
Ergotamine
Sympathomimetic amine
- Non-catecholamine
- Direct-acting
- A1 partial agonist
Caffeine
Sympathomimetic-like amine
- phosphodiesterase inhibitor
Theophylline
Sympathomimetic-like amine
- phosphodiesterase inhibitor
Sildenafil
Sympathomimetic-like amine
- phosphodiesterase inhibitor
Cocaine
Sympathomimetic-like amine
- NE/DA uptake blocker
Dimercaprol
Heavy metal chelator
- acute Pb, Inorg Hg, or As intoxication
DMTC
dimethyldithiocarbamate
Heavy metal chelator
- acute Cd intoxication
D-penicillamine
Heavy metal chelator
- persistant Pb intoxication
EDTA
Edetate Ca diNa
Heavy metal chelator
- acute Pb intoxication
Succimer
Heavy metal chelator
- Acute Pb, Hg, or As intoxication
Phenoxybenzamine
- Adrenergic Antagonist
- A1,2 receptor blocker
Phentolamine
- Adrenergic Antagonist
- A1,2 receptor blocker
Prazosin
- Adrenergic Antagonist
- A1 receptor blocker
Terazosin
- Adrenergic Antagonist
- A1 receptor blocker
Yohimbine
- Adrenergic Antagonist
- A2 receptor blocker
Propranolol
- Adrenergic Antagonist
- B1,2 receptor blocker
Timolol
- Adrenergic Antagonist
- B1,2 receptor blocker
Metoprolol
- Adrenergic Antagonist
- B1 receptor blocker
Labetalol
- Adrenergic Antagonist
- A/B receptor blocker
Cetirizine
Antihistamine

used for resp tract disorders
Desloratidine
Antihistamine

used for resp tract disorders
Diphenhydramine
Antihistamine

used for resp tract disorders
Fexofenadine
Antihistamine

used for resp tract disorders
Hydroxyzine
Antihistamine

used for resp tract disorders
Levocetirizine
Antihistamine

used for resp tract disorders
Loratidine
Antihistamine

used for resp tract disorders
Ipratropium
(Atrovent)
Resp Tract Treatment

Vasoconstrictor
Pseudoephedrine
(Sudafed)
Resp Tract Treatment

Vasoconstrictor
Flunisolide
Resp Tract Treatment

Anti-Inflammatory
Fluticasone
(flonase)
Resp Tract Treatment

Anti-Inflammatory
Mometason
(Nasonex)
Resp Tract Treatment

Anti-Inflammatory
D-methorphan
(Robitussin)
Resp Tract Treatment

Anti-tussive
B-IFN-1a
MS immunomodulator
B-IFN-1b
MS Immunomodulator
Glatiramer acetete
MS Immunomodulator
Mitoxantrone
MS Immunomodulator
Natalizumab
MS Immunomodulator
monoclonal antibody
Phytoin
(dilantin)
Anticonvulsant

Hydantoin
Carbamazepine
Anticonvulsant

Iminostilbene
Pheobarbital
Anticonvulsant

Barbiturate/desozybarbiturate
Valproic Acid
Anticonvulsant - GABA-ergic
- aids glutamic acid decarbozylase
- broad spectrum - can be used in all seizure types

Valproate
Ethosuximide
Anticonvulsant

Succinimide
Diazepam
(valium)
Anticonvulsant

Benzodiazepine
Clonazepam
Anticonvulsant

Benzodiazepine
Gabapentin
Anticonvulsant

GABA-ergic drug
Vigabatrin
Anticonvulsant

GABA-ergic drug
Acetazolamide
Anticonvulsant

other
Lamotrigine
(Lamictal)
Anticonvulsant

other
Ethanol
CNS Depressant

alcohol
Methanol
CNS Depressant

alcohol
Acamprosate
CNS Depressant

Antidote/Support
Disulfiram
(Antabuse)
CNS Depressant

Antidote/Support
Fomepizole
CNS Depressant

Antidote/Support
Aspirin
CVD drug

Antithrombotic
ASA/Dipyramidole XR
CVD drug

Antithrombotic
Clopidogrel
(Plavix)
CVD drug

Antithrombotic
Warfarin
(Coumadin)
CVD drug

Anticoagulant
- Vit K Antagonist
rt-PA
CVD Drug

Thrombolytic
Alteplase
CVD Drug

Thrombolytic