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127 Cards in this Set
- Front
- Back
botulinum toxin
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ACh Release Inhibitor, Snap25, Cosmetic and Spasm
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vancomycin
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Active only against gram+ bacteria, Inhibits the enzyme, peptidoglycan synthetase, responsible for adding the dissacharide, RED MAN
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Esmolol
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Adernergic “Selective” B1-blockers, ( 8 min) short half life, emrgencies
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Atenolol
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Adernergic “Selective” B1-blockers
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Clonidine
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Adernergic A-2 agonist, chemical sympthectome
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Methyldopa
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Adernergic A-2 agonist, methyldopa safe in pregnancy, some autoimmune response, chemical sympthectome
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Dopamine
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Adernergic agonist - [low] B1>B2, [high] all
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Dobutamine
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Adernergic agonist - [low] B1>B2, [high] all *Selective for contractility without affecting rate
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Epinephrine
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Adernergic agonist - [low] Betas, [high] all
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Phenoxybenzamine
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Adernergic Alpha(1>2) blockers (irreversible)
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Phenylephrine
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Adernergic Alpha1 Agonist. decongestant, pupilary dilator
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Norepinephrine
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Adernergic Alpha1 and Beta1 Agonist
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Terbutaline
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Adernergic B2 Selective agonist. Athsma
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Albuterol
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Adernergic Beta 2 Agonist
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Isoproterenol
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Adernergic Beta only Agonist
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Cocaine (Mechanism Only)
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Adernergic Blocks NET
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Imipramine (Mechanism Only)
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Adernergic Blocks NET
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Atomoxetine (Mechanism Only)
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Adernergic Blocks NET
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Reserpine (Mechanism Only)
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Adernergic Blocks VMAT(into vessical transporter) Cause depleation of NE Presynaptic
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Ephedrine
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Adernergic CNS stimulant (weak A and B agonist, and also a releaser of NE). nasal decongestant and a pressor
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Methylphenidate
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Adernergic CNS Stimulant for ADHD
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Amphetamine
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Adernergic displacement of NE (FED) ->sympathomimetic effects
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Guanethidine (Mechanism Only)
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Adernergic Displaces NE in Vessicles, reducing availabel concentration, enters via NET, Historic Anti-HTN
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Tyramine (Mechanism Only)
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Adernergic Metabolixed by Monoamine oxidase, On MAOI, it displaces the NE and NE Exits vis FED --> Hypertensive
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Phentolamine
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Adernergic Non-selective alpha blocker
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Propanolol
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Adernergic Non-selective Beta Blocker
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Timolol
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Adernergic non-selective beta blocker, glaucoma
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Prazosin
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Adernergic Selective alpha-1 blocker (reversible)
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Conivaptan
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ADH Antagonist, CD-V1a and V2 ADH Receptors
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Streptomycin
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Aminoglycosides,
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Gentamicin
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Aminoglycosides,
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Amikacin
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Aminoglycosides,
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Neomycin
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Aminoglycosides, poorly absorbed from gut (used as bowel sterilant)
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Question
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Answer
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Nifedipine
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Anti-Anginal, Dihydropyradine, Ca++ Blocker
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Nimodipine
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Anti-Anginal, Dihydropyradine, Ca++ Blocker
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Verapamil
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Anti-Anginal, Non-Dihydropyradine, Ca++ Blocker
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Diltiazem
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Anti-Anginal, Non-Dihydropyradine, Ca++ Blocker
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Nitroglycerin
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Anti-Anginal, Organic Nitrate
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Isosorbide dinitrate
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Anti-Anginal, Organic Nitrate
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amlodipine
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Anti-Hypertensive, Dihydropyridine Calcium Channel Blockers - Reflex Tachy
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captopril
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Anti-Hypertensive, (ACE) Inhibitors
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propranolol
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Anti-Hypertensive, All Beta blocker
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losartan
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Anti-Hypertensive, Angiotension Receptor Blockers
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hydrochlorothiazide
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Anti-Hypertensive, Diuretic -distal convoluted tubule - inhibit Na-Cl co-transport
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methyldopa
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Anti-Hypertensive, Inhibitors of Central adrenergic function- depletes norepinephrine, SAFE IN PREG
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guanethidine
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Anti-Hypertensive, Inhibitors of peripheral adrenergic function- depletes norepinephrine
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reserpine
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Anti-Hypertensive, Inhibitors of peripheral adrenergic function- depletes norepinephrine
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amiloride
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Anti-Hypertensive, K-sparing diuretics
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verapamil
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Anti-Hypertensive, Non-dihydropyridine calcium channel blockers
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clonidine
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Anti-Hypertensive, α2 agonist
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prazosin
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Anti-Hypertensive, α-blockers, “first does phenomenon”
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imipenem-cilastatin
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Carbapenemases, imipenem to prevent breakdown, Seizures
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meropenem
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carbapenems
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Acetazolamide
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Carbonic Anhydrase Inhibitor, PT and CD
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penicillin G
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Cell Wall Inhibitor
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amoxicillin
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Cell Wall Inhibitor, Extended Spectrum, Better GI Absorb
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ampicillin
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Cell Wall Inhibitor, Extended Spectrum, GI Probs
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piperacillin
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Cell Wall Inhibitor, Extended Spectrum, Only given IV or IM
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bacitracin
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Cell wall inhibitor, inhibits recycling of the lipid carrier
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cycloserine
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Cell wall inhibitor, inhibits the racemase and synthetase, 2nd line TB
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nafcillin
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Cell Wall Inhibitor, IV use mainly
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cefazolin
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Cephalosporin, 1st Gen,
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cephalexin
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Cephalosporin, 1st Gen,
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cefoxitin
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Cephalosporin, 2nd Gen, IV,
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ceftriaxone
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Cephalosporin, 3rd Gen, Crosses BBB
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ceftazidime
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Cephalosporin, 3rd Gen, Crosses BBB
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pralidoxime
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Cholinesterase Reactivator
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amoxicillin + clavulanic acid
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Clavulanic acid- inhibitor of bacterial beta lactamase, Improves activity
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daptomycin
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Cyclic lipopeptide, Forms ion conducting pore, Needs Calcium
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clindamycin
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Derivative of lincomycin L in MLS, Pseudomembranous colitis
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acetylcholine
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Direct-Acting Cholenergic Agonist
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bethanechol
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Direct-Acting Cholenergic Agonist
Metabolized by acetylcholinesterase? No Muscarinic Cholenergic? Any Dose Nicotinic Cholenergic? NO |
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nicotine
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Direct-Acting Cholenergic Agonists
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varenicline
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Direct-Acting Cholenergic Agonists
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carbachol
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Direct-Acting Cholenergics, Metabolized by
acetylcholinesterase? NO Muscarinic Cholenergic? Any Dose Nicotinic Cholenergic? High Dose Treatment of Glaucoma |
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Ciprofloxacin
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Fluoroquinolones
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Diphenhydramine
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H1 Antagonist 1st Gen (Benadryl®) Motion and Sleep
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Chlorpheniramine
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H1 Antagonist 1st Gen (Chlortrimeton®), OTC Cold Meds
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Dimenhydrinate
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H1 Antagonist 1st Gen (Dramamine®) Motion
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Loratadine
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H1 Antagonist 2nd Gen (Claritin®)
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Fexofenadine
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H1 Antagonist 2nd Gen (Allegra®)
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Cetirizine
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H1 Antagonist 2nd Gen (Zyrtec ®)
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Cimetidine
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H2 Antagonists (Tagamet®), Hormonal Effects(gynomastia, Impotence), Big CYP interactions
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Ranitidine
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H2 Antagonists (Zantac®)
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Famotidine
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H2 Antagonists (Pepcid®)
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donepezil
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Alzheimers
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rivastigmine
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Alzheimers
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galantamine
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Alzheimers
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sarin
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Death
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physostigmine
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Glaucoma
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edrophonium
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Myestinia Gravis Diag, Illius
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neostigmine
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Indirect-Acting Cholenergic Agonists, Anticholenesterase, Myestinia Gravis, Illius
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telithromycin
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Ketolide, 50% by CYP 3A4,
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Furoseminde
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Loop Diuretic, Na/K/2Cl (Acending loop)
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erythromycin
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Macrolide antibiotic
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azithromycin
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Macrolide antibiotic, Azithromycin penetrates tissues well (CNS exception), T1/2=3Days, Does not inhibit cytochrome P-450
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clarithromycin
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Macrolide antibiotic, More stable to acid than erythromycin
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Cromolyn Sodium
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Mast Cell Stabilizer (Nasalcrom®)
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Spirolactone
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Mineralcorticode antagonist, Aldosterone Antagonist (Competetive), CD, K+ Sparing
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Eplerenone
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Mineralcorticode antagonist, Aldosterone Antagonist (Competetive), CD, K+ Sparing
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aztreonam
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Monobactam
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atropine
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Muscarinic Antagonists, Crosses BBB, Used Pre Surgery
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ipratropium
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Muscarinic Antagonists, Used for COPD
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Amiloride
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Na+ Channel Blocker, K+ Sparing, CD
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hexamethonium
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Nicotinic Antagonists, Disected aorta, a3b2
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vecuronium
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Nicotinic Antagonists, Paralysis
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tubocurarine
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Nicotinic Antagonists, Paralysis, Hypotension(mast Cells)
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succinylcholine
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Nicotinic Antagonists, Quick Paralysis, faculations first, metabolized by ACHase-don’t use neo
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Mannitol
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Osmotic Diuretic, PT-Decending Loop-CD
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linezolid
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Oxazolidinone class, inhibitor of monoamine oxidase - avaoid tyrosine,
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H1 Antagonist Side Effects
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Sedation, CNS Effects, Non specific hit other receptors (anti-ach)
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Cotrimazole
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Sulfonamide
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Dapsone
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Sulfonamide, treatment of leprosy (w/rifampin)
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Sulfisoxazole
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Sulfonamide, urinary tract infections
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Sulfamethoxazole
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Sulfonamide, urinary tract infections (combo w/ trimethoprim)
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Tetracycline
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Tetracyclines,
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Doxycycline
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Tetracyclines,
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Minocycline
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Tetracyclines,
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Tigecycline
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Tetracyclines, IV only
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Hydrochlorothiazide
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Thiazide Diuretic, Na/Cl Cotransporter (DCT)
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Chloramphenicol
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topical usage for bacterial conjunctivitis - interfere with eukaryotic, mitochondrial ribosomes BAD, Gray Baby Syndrome
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Methenamine
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Urinary Antiseptic Agent, low pH (<5.5) to yield formaldehyde
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Nitrofurantoin
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Urinary Antiseptic Agent, reduction in bacteria (not humans)
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metronidazole
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With nitroreductase forms radicals. anaerobic infections and for pseudomembranous colitis due to C. difficile. Anabuse like, Inhibit P450. Brown Pee
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Caffeine
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Xanthine Blocks Phostdiesterase metabolism of cAMP, Andenosine Antagonist
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Theophylline
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Xanthine Relaxes Bronchi
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